Do active site conformations of small ligands correspond to low free-energy solution structures?
Vieth, M, Hirst, J D, Brooks, 3rd, C L
Published in Journal of computer-aided molecular design (01.11.1998)
Published in Journal of computer-aided molecular design (01.11.1998)
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Journal Article
The discovery of a new structural class of cyclin-dependent kinase inhibitors, aminoimidazo[1,2-a]pyridines
Hamdouchi, Chafiq, Keyser, Heather, Collins, Elizabeth, Jaramillo, Carlos, De Diego, Jose Eugenio, Spencer, Charles D, Dempsey, Jack Alan, Anderson, Bryan D, Leggett, Tillie, Stamm, Nancy B, Schultz, Richard M, Watkins, Scott A, Cocke, Kim, Lemke, Stephanie, Burke, Teresa F, Beckmann, Richard P, Dixon, Jeffrey T, Gurganus, Thomas M, Rankl, Nancy B, Houck, Keith A, Zhang, Faming, Vieth, Michal, Espinosa, Juan, Timm, David E, Campbell, Robert M, Patel, Bharvin K R, Brooks, Harold B
Published in Molecular cancer therapeutics (01.01.2004)
Published in Molecular cancer therapeutics (01.01.2004)
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Journal Article
Prediction of the Folding Pathways and Structure of the GCN4 Leucine Zipper
Vieth, Michal, Kolinski, Andrzej, Brooks, Charles L., Skolnick, Jeffrey
Published in Journal of molecular biology (08.04.1994)
Published in Journal of molecular biology (08.04.1994)
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Journal Article
An Exotic Visitor
Sen Gupta, Robin, Wilke, Karl, Vieth, Michael
Published in Deutsches Ärzteblatt international (23.02.2018)
Published in Deutsches Ärzteblatt international (23.02.2018)
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Journal Article
Design of potent and selective 2-aminobenzimidazole-based p38alpha MAP kinase inhibitors with excellent in vivo efficacy
de Dios, Alfonso, Shih, Chuan, López de Uralde, Beatriz, Sánchez, Concepción, del Prado, Miriam, Martín Cabrejas, Luisa M, Pleite, Sehila, Blanco-Urgoiti, Jaime, Lorite, María José, Nevill, Jr, C Richard, Bonjouklian, Rosanne, York, Jeremy, Vieth, Michal, Wang, Yong, Magnus, Nicholas, Campbell, Robert M, Anderson, Bryan D, McCann, Denis J, Giera, Deborah D, Lee, Paul A, Schultz, Richard M, Li, Li C, Johnson, Lea M, Wolos, Jeffrey A
Published in Journal of medicinal chemistry (07.04.2005)
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Published in Journal of medicinal chemistry (07.04.2005)
Journal Article
A red spot in the gut : The "floater" as a classic pitfall?
Lang-Schwarz, Corinna, Kiene, Ralf, Böcker, Ingo, Sterlacci, William, Oellig, Frank, Vieth, Michael
Published in Pathologie (Heidelberg, Germany) (01.09.2022)
Published in Pathologie (Heidelberg, Germany) (01.09.2022)
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Journal Article
Predicting leucine zipper structures from sequence
Hirst, Jonathan D., Vieth, Michal, Skolnick, Jeffrey, Brooks, Charles L.
Published in Protein engineering (01.08.1996)
Published in Protein engineering (01.08.1996)
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Journal Article
Molecular properties that influence oral drug-like behavior
Lajiness, Michael S, Vieth, Michal, Erickson, Jon
Published in Current opinion in drug discovery & development (01.07.2004)
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Published in Current opinion in drug discovery & development (01.07.2004)
Journal Article
Novel Route to the Synthesis of 4-Quinolyl Isothiocyanates
Zhong, Boyu, Al-Awar, Rima S., Shih, Chuan, Grimes, John H. Jr, Vieth, Michal, Hamdouchi, Chafiq
Published in ChemInform (04.07.2006)
Published in ChemInform (04.07.2006)
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Journal Article
Benzimidazoles and benzothiazoles as inhibitors of map kinase
Bonjouklian, Rosanne, De Diego Gomez, Jose Eugenio, De Dios, Alfonso, Hamdouchi, Chafiq Hamdouchi, Li, Tiecho, De Uralde Garmendia, Beatriz Lopez, Vieth, Michal, York, Jeremy Schulenberg, Dally, Robert Dean, Del Prado Catalina, Miriam Filadelfa, Jaramillo Aguado, Carlos, Martin-Cabrejas, Luisa Maria, Montero Salgado, Carlos, Pleite Selgas, Sheila, Sanchez-Martinez, Concepcion, Shepherd, Timothy Alan, Wikel, James Howard
Year of Publication 22.01.2008
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Year of Publication 22.01.2008
Patent
Benzimidazoles and benzothiazoles as inhibitors of map kinase
PLEITE SELGAS SHEILA, WIKEL JAMES HOWARD, DE DIOS ALFONSO, BONJOUKLIAN ROSANNE, VIETH MICHAL, DEL PRADO CATALINA MIRIAM FILADELFA, DE DIEGO GOMEZ JOSE EUGENIO, DE URALDE GARMENDIA BEATRIZ LOPEZ, MARTIN-CABREJAS LUISA MARIA, SANCHEZ-MARTINEZ CONCEPCION, HAMDOUCHI CHAFIQ HAMDOUCHI, LI TIECHO, MONTERO SALGADO CARLOS, YORK JEREMY SCHULENBERG, SHEPHERD TIMOTHY ALAN, DALLY ROBERT DEAN, JARAMILLO AGUADO CARLOS
Year of Publication 22.01.2008
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Year of Publication 22.01.2008
Patent