3‘-C-Branched-Chain-Substituted Nucleosides and Nucleotides as Potent Inhibitors of Mycobacterium tuberculosis Thymidine Monophosphate Kinase
VANHEUSDEN, Veerle, MUNIER-LEHMANN, Hélène, FROEYEN, Matheus, DUGUé, Laurence, HEYERICK, Arne, DE KEUKELEIRE, Denis, POCHET, Sylvie, BUSSON, Roger, HERDEWIJN, Piet, VAN CALENBERGH, Serge
Published in Journal of medicinal chemistry (28.08.2003)
Published in Journal of medicinal chemistry (28.08.2003)
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Journal Article
Enzymatic and Structural Analysis of Inhibitors Designed against Mycobacterium tuberculosis Thymidylate Kinase
Haouz, Ahmed, Vanheusden, Veerle, Munier-Lehmann, Hélène, Froeyen, Mattheus, Herdewijn, Piet, Van Calenbergh, Serge, Delarue, Marc
Published in The Journal of biological chemistry (14.02.2003)
Published in The Journal of biological chemistry (14.02.2003)
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Journal Article
Enzymatic and structural analysis of inhibitors designed against Mycobacterium tuberculosis thymidylate kinase. New insights into the phosphoryl transfer mechanism
Haouz, Ahmed, Vanheusden, Veerle, Munier-Lehmann, Hélène, Froeyen, Mattheus, Herdewijn, Piet, Van Calenbergh, Serge, Delarue, Marc
Published in The Journal of biological chemistry (14.02.2003)
Published in The Journal of biological chemistry (14.02.2003)
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Journal Article
Discovery of Bicyclic Thymidine Analogues as Selective and High-Affinity Inhibitors of Mycobacterium tuberculosis Thymidine Monophosphate Kinase
Vanheusden, Veerle, Munier-Lehmann, Hélène, Froeyen, Matheus, Busson, Roger, Rozenski, Jef, Herdewijn, Piet, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
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Synthesis and evaluation of thymidine-5′- O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase
Vanheusden, Veerle, Munier-Lehmann, Hélène, Pochet, Sylvie, Herdewijn, Piet, Van Calenbergh, Serge
Published in Bioorganic & medicinal chemistry letters (07.10.2002)
Published in Bioorganic & medicinal chemistry letters (07.10.2002)
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Journal Article
Thymidine and thymidine-5′- O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase
Vanheusden, Veerle, Van Rompaey, Philippe, Munier-Lehmann, Hélène, Pochet, Sylvie, Herdewijn, Piet, Van Calenbergh, Serge
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
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Journal Article
Thymidine and thymidine-5'-O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase: Recent advances in the design of kinase inhibitors as novel therapeutic agents
VANHEUSDEN, Veerle, VAN ROMPAEY, Philippe, MUNIER-LEHMANN, Hélène, POCHET, Sylvie, HERDEWIJN, Piet, VAN CALENBERGH, Serge
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
Journal Article
Mycobacterium tuberculosis Thymidine Monophosphate Kinase Inhibitors: Biological Evaluation and Conformational Analysis of 2′- and 3′-Modified Thymidine Analogues
Van Rompaey, Philippe, Nauwelaerts, Koen, Vanheusden, Veerle, Rozenski, Jef, Munier-Lehmann, Hélène, Herdewijn, Piet, Van Calenbergh, Serge
Published in European journal of organic chemistry (01.08.2003)
Published in European journal of organic chemistry (01.08.2003)
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Journal Article
3‘-C-Branched-Chain-Substituted Nucleosides and Nucleotides as Potent Inhibitors of Mycobacterium t uberculosis Thymidine Monophosphate Kinase
Vanheusden, Veerle, Munier-Lehmann, Hélène, Froeyen, Matheus, Dugué, Laurence, Heyerick, Arne, De Keukeleire, Denis, Pochet, Sylvie, Busson, Roger, Herdewijn, Piet, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (28.08.2003)
Published in Journal of medicinal chemistry (28.08.2003)
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Journal Article
5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists
Van Calenbergh, Serge, Link, Andreas, Fujikawa, Shelly, de Ligt, Rianne A F, Vanheusden, Veerle, Golisade, Abolfasl, Blaton, Norbert M, Rozenski, Jef, IJzerman, Adriaan P, Herdewijn, Piet
Published in Journal of medicinal chemistry (25.04.2002)
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Published in Journal of medicinal chemistry (25.04.2002)
Journal Article
5‘-Deoxy Congeners of 9-(3-Amido-3-deoxy- β - d -xylofuranosyl)- N 6 -cyclopentyladenine: New Adenosine A 1 Receptor Antagonists and Inverse Agonists
Van Calenbergh, Serge, Link, Andreas, Fujikawa, Shelly, de Ligt, Rianne A. F., Vanheusden, Veerle, Golisade, Abolfasl, Blaton, Norbert M., Rozenski, Jef, IJzerman, Adriaan P., Herdewijn, Piet
Published in Journal of medicinal chemistry (01.04.2002)
Published in Journal of medicinal chemistry (01.04.2002)
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Journal Article
5‘-Deoxy Congeners of 9-(3-Amido-3-deoxy-β-d-xylofuranosyl)-N6-cyclopentyladenine: New Adenosine A1 Receptor Antagonists and Inverse Agonists
VAN CALENBERGH, Serge, LINK, Andreas, FUJIKAWA, Shelly, DE LIGT, Rianne A. F., VANHEUSDEN, Veerle, GOLISADE, Abolfasl, BLATON, Norbert M., ROZENSKI, Jef, IJZERMAN, Adriaan P., HERDEWIJN, Piet
Published in Journal of medicinal chemistry (25.04.2002)
Published in Journal of medicinal chemistry (25.04.2002)
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Journal Article
5‘-Deoxy Congeners of 9-(3-Amido-3-deoxy-β-d-xylofuranosyl)-N 6-cyclopentyladenine: New Adenosine A1 Receptor Antagonists and Inverse Agonists
Van Calenbergh, Serge, Link, Andreas, Fujikawa, Shelly, de Ligt, Rianne A. F, Vanheusden, Veerle, Golisade, Abolfasl, Blaton, Norbert M, Rozenski, Jef, IJzerman, Adriaan P, Herdewijn, Piet
Published in Journal of medicinal chemistry (25.04.2002)
Published in Journal of medicinal chemistry (25.04.2002)
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Journal Article