Two distinct classes of novel pyrazolinecarboxamides as potent cannabinoid CB1 receptor agonists
LANGE, Jos H. M, ATTALI, Amos, VAN DER NEUT, Martina A. W, WALS, Henri C, MULDER, Arie, ZILAOUT, Hicham, DUURSMA, Ate, VAN AKEN, Hans H. M, VAN VLIET, Bernard J
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Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB1 receptor antagonists
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Synthesis and SAR of novel imidazoles as potent and selective cannabinoid CB2 receptor antagonists with high binding efficiencies
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Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Probing the cannabinoid CB1/CB2 receptor subtype selectivity limits of 1,2-diarylimidazole-4-carboxamides by fine-tuning their 5-substitution pattern
LANGE, Jos H. M, VAN DER NEUT, Martina A. W, BORST, Alice J. M, YILDIRIM, Mahmut, VAN STUIVENBERG, Herman H, VAN VLIET, Bernard J, KRUSE, Chris G
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USE OF INDOLE DERIVATIVES AS NURR-1 ACTIVATORS FOR TREATING PARKINSON'S DISEASE
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Year of Publication 07.10.2011
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Year of Publication 07.10.2011
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The novel compound Sul-121 inhibits airway inflammation and hyperresponsiveness in experimental models of chronic obstructive pulmonary disease
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Two distinct classes of novel pyrazolinecarboxamides as potent cannabinoid CB 1 receptor agonists
Lange, Jos H.M., Attali, Amos, van der Neut, Martina A.W., Wals, Henri C., Mulder, Arie, Zilaout, Hicham, Duursma, Ate, van Aken, Hans H.M., van Vliet, Bernard J.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Probing the cannabinoid CB 1/CB 2 receptor subtype selectivity limits of 1,2-diarylimidazole-4-carboxamides by fine-tuning their 5-substitution pattern
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Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB 1 receptor antagonists
Lange, Jos H.M., van der Neut, Martina A.W., den Hartog, Arnold P., Wals, Henri C., Hoogendoorn, Jan, van Stuivenberg, Herman H., van Vliet, Bernard J., Kruse, Chris G.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Probing the cannabinoid CB sub(1)/CB sub(2) receptor subtype selectivity limits of 1,2-diarylimidazole-4-carboxamides by fine-tuning their 5-substitution pattern
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Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Antipsychotic drugs classified by their effects on the release of dopamine and noradrenaline in the prefrontal cortex and striatum
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Published in European journal of pharmacology (26.01.2001)
Published in European journal of pharmacology (26.01.2001)
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