4-원 헤테로시클릭 아미드를 포함하는 JAK 저해제
SMITH CAMERON, KLEINSCHEK MELANIE A, CRATER GLENN D, SULLIVAN STEVEN D.E, VAN ORDEN LORI JEAN, FATHEREE PAUL R, BRANDT GARY E.L
Year of Publication 13.11.2019
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Year of Publication 13.11.2019
Patent
융합된 이미다조-피페리딘 JAK 저해제
SMITH CAMERON, KLEINSCHEK MELANIE A, CRATER GLENN D, SULLIVAN STEVEN D.E, VAN ORDEN LORI JEAN, FATHEREE PAUL R, BRANDT GARY E.L
Year of Publication 13.11.2019
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Year of Publication 13.11.2019
Patent
호흡기 질환의 치료를 위한 JAK 키나제 저해제 화합물
FASS GENE TIMOTHY, BENJAMIN NOAH, BEAUSOLEIL ANNE MARIE, FLEURY MELISSA, COLSON PIERRE JEAN, SULLIVAN STEVEN D.E, VAN ORDEN LORI JEAN, SMITH CAMERON, JACOBSEN JOHN R, THALLADI VENKAT R, JIANG LAN, DABROS MARTA, RAPTA MIROSLAV, FATHEREE PAUL R, BRANDT GARY E.L
Year of Publication 02.07.2018
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Year of Publication 02.07.2018
Patent
ROD-LIKE HEPATITIS C VIRUS INHIBITORS CONTAINING THE FRAGEMENT [2-[4-(BI PHENYL-4-YL)-1H-IMIDAZO-2-YL]PYRROLIDINE-1-CARBONLYMETHYL]AMINE
ZHANG WEIJIANG, HUANG XIAOJUN, LONG DANIEL D, MCKINNELL ROBERT MURRAY, OGAWA GAVIN, JIANG LAN, LOO MANDY, VAN ORDEN LORI JEAN, LEPACK KASSANDRA
Year of Publication 18.07.2014
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Year of Publication 18.07.2014
Patent
S102 - NMRA-140, a Novel and Selective Kappa Opioid Receptor Antagonist: Mode of Action Profiling Studies Demonstrate No Opioid Agonist Properties Implicated in Opioid-Related Abuse
Morrison, Filomene, Van Orden, Lori Jean, Zeitz, Karla, Heal, David, Smith, Sharon, Wallace, Tanya
Published in Drug and alcohol dependence (01.07.2024)
Published in Drug and alcohol dependence (01.07.2024)
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Journal Article
NMRA-140, a Novel and Selective Kappa Opioid Receptor Antagonist: Mode of Action Profiling Studies Demonstrate No Opioid Agonist Properties Implicated in Opioid-Related Abuse
Morrison, Filomene, Van Orden, Lori Jean, Zeitz, Karla, Heal, David, Smith, Sharon, Wallace, Tanya
Published in Drug and alcohol dependence (01.07.2024)
Published in Drug and alcohol dependence (01.07.2024)
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Journal Article
225. NMRA-140, a Novel and Selective Kappa Opioid Receptor Antagonist: Mode of Action Profiling Studies Demonstrate No Opioid Agonist Properties Implicated in Opioid-Related Abuse
Morrison, Filomene, Van Orden, Lori Jean, Zeitz, Karla, Heal, David, Smith, Sharon, Wallace, Tanya L.
Published in Biological psychiatry (1969) (01.05.2023)
Published in Biological psychiatry (1969) (01.05.2023)
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Journal Article
Navacaprant, a novel and selective kappa opioid receptor antagonist, has no agonist properties implicated in opioid-related abuse
Morrison, Filomene G., Van Orden, Lori Jean, Zeitz, Karla, Kuijer, Eloise J., Smith, Sharon L., Heal, David J., Wallace, Tanya L.
Published in Neuropharmacology (01.10.2024)
Published in Neuropharmacology (01.10.2024)
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Journal Article
Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140)
Guerrero, Miguel, Urbano, Mariangela, Kim, Eun-Kyong, Gamo, Ana M, Riley, Sean, Abgaryan, Lusine, Leaf, Nora, Van Orden, Lori Jean, Brown, Steven J, Xie, Jennifer Y, Porreca, Frank, Cameron, Michael D, Rosen, Hugh, Roberts, Edward
Published in Journal of medicinal chemistry (28.02.2019)
Published in Journal of medicinal chemistry (28.02.2019)
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A novel class of 3-(phenoxy-phenyl-methyl)-pyrrolidines as potent and balanced norepinephrine and serotonin reuptake inhibitors: Synthesis and structure–activity relationships
Van Orden, Lori Jean, Van Dyke, Priscilla M., Saito, D. Roland, Church, Timothy J., Chang, Ray, Smith, Jacqueline A.M., Martin, William J., Jaw-Tsai, Sarah, Stangeland, Eric L.
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
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Journal Article
JAK inhibitors containing a 4-membered heterocyclic amide
Fatheree, Paul R, Sullivan, Steven D. E, Smith, Cameron, Van Orden, Lori Jean, Kleinschek, Melanie A, Crater, Glenn D, Brandt, Gary E. L
Year of Publication 23.01.2024
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Year of Publication 23.01.2024
Patent
JAK inhibitors containing a 4-membered heterocyclic amide
Fatheree, Paul R, Sullivan, Steven D. E, Smith, Cameron, Van Orden, Lori Jean, Brandt, Gary E. L
Year of Publication 27.09.2022
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Year of Publication 27.09.2022
Patent
JAK INHIBITORS CONTAINING A 4-MEMBERED HETEROCYCLIC AMIDE
FATHEREE, PAUL R, SMITH, CAMERON, BRANDT, GARY E.L, SULLIVAN, STEVEN D.E, VAN ORDEN, LORI JEAN
Year of Publication 02.09.2021
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Year of Publication 02.09.2021
Patent
Fused imidazo-piperidine JAK inhibitors
Fatheree, Paul R, Sullivan, Steven D. E, Smith, Cameron, Van Orden, Lori Jean, Kleinschek, Melanie A, Crater, Glenn D, Brandt, Gary E. L
Year of Publication 06.06.2023
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Year of Publication 06.06.2023
Patent
JAK INHIBITORS CONTAINING A 4-MEMBERED HETEROCYCLIC AMIDE
FATHEREE, PAUL R, SMITH, CAMERON, CRATER, GLENN D, KLEINSCHEK, MELANIE A, BRANDT, GARY E.L, SULLIVAN, STEVEN D.E, VAN ORDEN, LORI JEAN
Year of Publication 02.03.2023
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Year of Publication 02.03.2023
Patent
Fused imidazo-piperidine JAK inhibitors
Fatheree, Paul R, Sullivan, Steven D. E, Smith, Cameron, Van Orden, Lori Jean, Brandt, Gary E. L
Year of Publication 22.02.2022
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Year of Publication 22.02.2022
Patent
Jak kinase inhibitor compounds for treatment of respiratory disease
Rapta, Miroslav, Benjamin, Noah, Jacobsen, John R, Fatheree, Paul R, Smith, Cameron, Van Orden, Lori Jean, Brandt, Gary E.l, Dabros, Marta, Fleury, Melissa, Beausoleil, Anne-Marie, Jiang, Lan, Colson, Pierre-Jean, Sullivan, Steven D.e, Thalladi, Venkat R, Fass, Gene Timothy
Year of Publication 24.11.2023
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Year of Publication 24.11.2023
Patent
FUSED IMIDAZO-PIPERIDINE JAK INHIBITORS
Fatheree, Paul R, Sullivan, Steven D. E, Smith, Cameron, Van Orden, Lori Jean, Kleinschek, Melanie A, Crater, Glenn D, Brandt, Gary E. L
Year of Publication 15.09.2022
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Year of Publication 15.09.2022
Patent
JAK INHIBITORS CONTAINING A 4-MEMBERED HETEROCYCLIC AMIDE
FATHEREE, PAUL R, SMITH, CAMERON, BRANDT, GARY E.L, SULLIVAN, STEVEN D.E, VAN ORDEN, LORI JEAN
Year of Publication 09.07.2020
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Year of Publication 09.07.2020
Patent