Discovery and Profiling of a Selective and Efficacious Syk Inhibitor
Thoma, Gebhard, Smith, Alexander B, van Eis, Maurice J, Vangrevelinghe, Eric, Blanz, Joachim, Aichholz, Reiner, Littlewood-Evans, Amanda, Lee, Christian C, Liu, Hong, Zerwes, Hans-Günter
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
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Indolyl-naphthyl-maleimides as potent and selective inhibitors of protein kinase C-α/β
van Eis, Maurice J., Evenou, JeanPierre, Schuler, Walter, Zenke, Gerhard, Vangrevelinghe, Eric, Wagner, Juergen, von Matt, Peter
Published in Bioorganic & medicinal chemistry letters (15.02.2017)
Published in Bioorganic & medicinal chemistry letters (15.02.2017)
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Novel ROCK inhibitors for the treatment of pulmonary arterial hypertension
Shaw, Duncan, Hollingworth, Greg, Soldermann, Nicolas, Sprague, Elizabeth, Schuler, Walter, Vangrevelinghe, Eric, Duggan, Nicholas, Thomas, Matthew, Kosaka, Takatoshi, Waters, Nigel, van Eis, Maurice J.
Published in Bioorganic & medicinal chemistry letters (15.10.2014)
Published in Bioorganic & medicinal chemistry letters (15.10.2014)
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Syk inhibitors with high potency in presence of blood
Thoma, Gebhard, Blanz, Joachim, Bühlmayer, Peter, Drückes, Peter, Kittelmann, Matthias, Smith, Alexander B., van Eis, Maurice, Vangrevelinghe, Eric, Zerwes, Hans-Günter, Che, Jianwei (John), He, Xiaohui, Jin, Yunho, Lee, Christian C., Michellys, Pierre-Yves, Uno, Tetsuo, Liu, Hong
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
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Journal Article
2,6-Naphthyridines as potent and selective inhibitors of the novel protein kinase C isozymes
van Eis, Maurice J., Evenou, Jean-Pierre, Floersheim, Philipp, Gaul, Christoph, Cowan-Jacob, Sandra W., Monovich, Lauren, Rummel, Gabriele, Schuler, Walter, Stark, Wilhelm, Strauss, Andre, Matt, Anette von, Vangrevelinghe, Eric, Wagner, Juergen, Soldermann, Nicolas
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
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Synthesis and anomalous structure–reactivity relationship of 8,11-dichloro[5]metacyclophan-3-one
van Es, Daniël S, Gret, Norbert, de Rijke, Marianne, van Eis, Maurice J, de Kanter, Franciscus J.J, de Wolf, Willem H, Bickelhaupt, Friedrich, Menzer, Stephan, Spek, Anthony L
Published in Tetrahedron (23.04.2001)
Published in Tetrahedron (23.04.2001)
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12,15-Dichloro[3.0]orthometacyclophane: A Highly Strained Biphenylophane
van Eis, Maurice J, Bickelhaupt, Friedrich
Published in Journal of the American Chemical Society (15.04.1998)
Published in Journal of the American Chemical Society (15.04.1998)
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Journal Article
Supramolecular Fullerene Chemistry: A Comprehensive Study of Cyclophane-Type Mono- and Bis-Crown Ether Conjugates of C70
van Eis, Maurice J., Seiler, Paul, Muslinkina, Liya A., Badertscher, Martin, Pretsch, Ernö, Diederich, François, Alvarado, Robert J., Echegoyen, Luis, Pérez Núñez, Ignacio
Published in Helvetica chimica acta (01.07.2002)
Published in Helvetica chimica acta (01.07.2002)
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Journal Article
Chiroptical properties of 12,15-dichloro[3.0]orthometacyclophane—correlations between molecular structure and circular dichroism spectra of a biphenylophane
Niederalt, Christoph, Grimme, Stefan, Peyerimhoff, Sigrid D, Sobanski, Adam, Vögtle, Fritz, Lutz, Martin, Spek, Anthony L, van Eis, Maurice J, de Wolf, Willem H, Bickelhaupt, Friedrich
Published in Tetrahedron: asymmetry (04.06.1999)
Published in Tetrahedron: asymmetry (04.06.1999)
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Trapping of the highly strained [5](2,4)quinolinophane system
van Eis, Maurice J., Lutz, Martin, Spek, Anthony L., de Wolf, Willem H., Bickelhaupt, Friedrich
Published in Tetrahedron (12.02.2007)
Published in Tetrahedron (12.02.2007)
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Journal Article
The 2-Vinylphosphirane−3-Phospholene Rearrangement: Biradicaloid and Concerted Features
van Eis, Maurice J, Nijbacker, Tom, de Kanter, Franciscus J. J, de Wolf, Willem H, Lammertsma, Koop, Bickelhaupt, Friedrich
Published in Journal of the American Chemical Society (05.04.2000)
Published in Journal of the American Chemical Society (05.04.2000)
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Journal Article
Dichlorocarbene Addition to [5]Metacyclophane; Experimental and Calculational Evidence for a [1,5] Sigmatropic Chlorine Shift in a Bridged Cycloheptatriene
van Eis, Maurice J, van der Linde, Barbara S. E, de Kanter, Franciscus J. J, de Wolf, Willem H, Bickelhaupt, Friedrich
Published in Journal of organic chemistry (14.07.2000)
Published in Journal of organic chemistry (14.07.2000)
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Journal Article
1,4-Addition of a Terminal Phosphinidene Complex to [5]Metacyclophane
van Eis, Maurice J., Komen, Corine M. D., de Kanter, Franciscus J. J., de Wolf, Willem H., Lammertsma, Koop, Bickelhaupt, Friedrich, Lutz, Martin, Spek, Anthony L.
Published in Angewandte Chemie (International ed.) (19.06.1998)
Published in Angewandte Chemie (International ed.) (19.06.1998)
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The First Free 7λ 3-Phosphanorbornadiene
van Eis, Maurice J, Zappey, Herman, de Kanter, Franciscus J. J, de Wolf, Willem H, Lammertsma, Koop, Bickelhaupt, Friedrich
Published in Journal of the American Chemical Society (12.04.2000)
Published in Journal of the American Chemical Society (12.04.2000)
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Journal Article
7,14-Dichloro[1.1]metacyclophane: A Highly Strained Aromatic Intermediate
van Eis, Maurice J, de Kanter, Franciscus J. J, de Wolf, Willem H, Bickelhaupt, Friedrich
Published in Journal of organic chemistry (17.10.1997)
Published in Journal of organic chemistry (17.10.1997)
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Journal Article
Identification of Orally Available Naphthyridine Protein Kinase D Inhibitors
Meredith, Erik L, Ardayfio, Ophelia, Beattie, Kimberly, Dobler, Markus R, Enyedy, Istvan, Gaul, Christoph, Hosagrahara, Vinayak, Jewell, Charles, Koch, Keith, Lee, Wendy, Lehmann, HansJoerg, McKinsey, Timothy A, Miranda, Karl, Pagratis, Nikos, Pancost, Margaret, Patnaik, Anup, Phan, Dillon, Plato, Craig, Qian, Ming, Rajaraman, Vasumathy, Rao, Chang, Rozhitskaya, Olga, Ruppen, Thomas, Shi, Jie, Siska, Sarah J, Springer, Clayton, van Eis, Maurice, Vega, Richard B, von Matt, Anette, Yang, Lihua, Yoon, Taeyoung, Zhang, Ji-Hu, Zhu, Na, Monovich, Lauren G
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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Journal Article
Identification of Potent and Selective Amidobipyridyl Inhibitors of Protein Kinase D
Meredith, Erik L, Beattie, Kimberly, Burgis, Robin, Capparelli, Michael, Chapo, Joseph, DiPietro, Lucian, Gamber, Gabriel, Enyedy, Istvan, Hood, David B, Hosagrahara, Vinayak, Jewell, Charles, Koch, Keith A, Lee, Wendy, Lemon, Douglas D, McKinsey, Timothy A, Miranda, Karl, Pagratis, Nikos, Phan, Dillon, Plato, Craig, Rao, Chang, Rozhitskaya, Olga, Soldermann, Nicolas, Springer, Clayton, van Eis, Maurice, Vega, Richard B, Yan, Wanlin, Zhu, Qingming, Monovich, Lauren G
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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