A novel doxorubicin-glucuronide prodrug DOX-GA3 for tumour-selective chemotherapy: distribution and efficacy in experimental human ovarian cancer
HOUBA, P. H. J, BOVEN, E, VAN DER MEULEN-MUILEMAN, I. H, LEENDERS, R. G. G, SCHEEREN, J. W, PINEDO, H. M, HAISMA, H. J
Published in British journal of cancer (01.02.2001)
Published in British journal of cancer (01.02.2001)
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Secreted and tumour targeted human carboxylesterase for activation of irinotecan
OOSTERHOFF, D, PINEDO, H. M, VAN DER MEULEN, I. H, DE GRAAF, M, SONE, T, KRUYT, F. A, VAN BEUSECHEM, V. W, HAISMA, H. J, GERRITSEN, W. R
Published in British journal of cancer (09.09.2002)
Published in British journal of cancer (09.09.2002)
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A fully human anti-Ep-CAM scFv-beta-glucuronidase fusion protein for selective chemotherapy with a glucuronide prodrug
DE GRAAF, M, BOVEN, E, OOSTERHOFF, D, VAN DER MEULEN-MUILEMAN, I. H, HULS, G. A, GERRITSEN, W. R, HAISMA, H. J, PINEDO, H. M
Published in British journal of cancer (04.03.2002)
Published in British journal of cancer (04.03.2002)
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Adenoviral vector-mediated expression of a gene encoding secreted, EpCAM-targeted carboxylesterase-2 sensitises colon cancer spheroids to CPT-11
Oosterhoff, D, Overmeer, R M, de Graaf, M, van der Meulen, I H, Giaccone, G, van Beusechem, V W, Haisma, H J, Pinedo, H M, Gerritsen, W R
Published in British journal of cancer (14.03.2005)
Published in British journal of cancer (14.03.2005)
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Pronounced antitumor efficacy of doxorubicin when given as the prodrug DOX‐GA3 in combination with a monoclonal antibody β‐glucuronidase conjugate
Houba, P.H.J., Boven, E., van der Meulen‐Muileman, I.H., Leenders, R.G.G., Scheeren, J.W., Pinedo, H.M., Haisma, H.J.
Published in International journal of cancer (15.02.2001)
Published in International journal of cancer (15.02.2001)
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Cloning and characterization of human liver cytosolic beta-glycosidase
de Graaf, M, van Veen, I C, van der Meulen-Muileman, I H, Gerritsen, W R, Pinedo, H M, Haisma, H J
Published in Biochemical journal (15.06.2001)
Published in Biochemical journal (15.06.2001)
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Distribution and pharmacokinetics of the prodrug daunorubicin-GA3 in nude mice bearing human ovarian cancer xenografts
Houba, Pieter H.J, Boven, Epie, van der Meulen-Muileman, Ida H, Leenders, Ruben G.G, Scheeren, Johannes W, Pinedo, Herbert M, Haisma, Hidde J
Published in Biochemical pharmacology (15.03.1999)
Published in Biochemical pharmacology (15.03.1999)
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Adenoviral vector-mediated expression of a gene encoding secreted, EpCAM-targeted carboxylesterase-2 sensitises colon cancer spheroids to CPT- II
OOSTERHOFF, D, OVERMEER, R. M, DE GRAAF, M, VAN DER MEULEN, I. H, GIACCONE, G, VAN BEUSECHEM, V. W, HAISMA, H. J, PINEDO, H. M, GERRITSEN, W. R
Published in British journal of cancer (2005)
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Published in British journal of cancer (2005)
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Pronounced antitumor efficacy by extracellular activation of a doxorubicin-glucuronide prodrug after adenoviral vector-mediated expression of a human antibody-enzyme fusion protein
de Graaf, Michelle, Pinedo, Herbert M, Oosterhoff, Dinja, van der Meulen-Muileman, Ida H, Gerritsen, Winald R, Haisma, Hidde J, Boven, Epie
Published in Human gene therapy (01.03.2004)
Published in Human gene therapy (01.03.2004)
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