Non-covalent inhibitors of rhinovirus 3C protease
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Published in Bioorganic & medicinal chemistry letters (15.01.2011)
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Chan, Bryan K, Estrada, Anthony A, Chen, Huifen, Atherall, John, Baker-Glenn, Charles, Beresford, Alan, Burdick, Daniel J, Chambers, Mark, Dominguez, Sara L, Drummond, Jason, Gill, Andrew, Kleinheinz, Tracy, Le Pichon, Claire E, Medhurst, Andrew D, Liu, Xingrong, Moffat, John G, Nash, Kevin, Scearce-Levie, Kimberly, Sheng, Zejuan, Shore, Daniel G, Van de Poël, Hervé, Zhang, Shuo, Zhu, Haitao, Sweeney, Zachary K
Published in ACS medicinal chemistry letters (10.01.2013)
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Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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Journal Article
Optimization of M3 Antagonist–PDE4 Inhibitor (MAPI) Dual Pharmacology Molecules for the Treatment of COPD
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Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Discovery of M3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
Armani, Elisabetta, Rizzi, Andrea, Capaldi, Carmelida, De Fanti, Renato, Delcanale, Maurizio, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Puccini, Paola, Amadei, Francesco, Pappani, Alice, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles A.G, Van de Poël, Hervé, Blackaby, Wesley P, Nash, Kevin, Amari, Gabriele
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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A Novel, Broad-Spectrum Inhibitor of Enterovirus Replication That Targets Host Cell Factor Phosphatidylinositol 4-Kinase IIIβ
van der Schaar, Hilde M, Leyssen, Pieter, Thibaut, Hendrik J, de Palma, Armando, van der Linden, Lonneke, Lanke, Kjerstin H W, Lacroix, Céline, Verbeken, Erik, Conrath, Katja, Macleod, Angus M, Mitchell, Dale R, Palmer, Nicholas J, van de Poël, Hervé, Andrews, Martin, Neyts, Johan, van Kuppeveld, Frank J M
Published in Antimicrobial Agents and Chemotherapy (01.10.2013)
Published in Antimicrobial Agents and Chemotherapy (01.10.2013)
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Identification of a Series of Compounds with Potent Antiviral Activity for the Treatment of Enterovirus Infections
MacLeod, Angus M, Mitchell, Dale R, Palmer, Nicholas J, Van de Poël, Hervé, Conrath, Katja, Andrews, Martin, Leyssen, Pieter, Neyts, Johan
Published in ACS medicinal chemistry letters (11.07.2013)
Published in ACS medicinal chemistry letters (11.07.2013)
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Journal Article
Optimization of M 3 Antagonist-PDE4 Inhibitor (MAPI) Dual Pharmacology Molecules for the Treatment of COPD
Rizzi, Andrea, Amari, Gabriele, Pivetti, Fausto, Delcanale, Maurizio, Amadei, Francesco, Pappani, Alice, Fornasari, Luca, Villetti, Gino, Marchini, Gessica, Pisano, Anna Rita, Pitozzi, Vanessa, Pittelli, Maria Gloria, Trevisani, Marcello, Salvadori, Michela, Cenacchi, Valentina, Fioni, Alessandro, Puccini, Paola, Civelli, Maurizio, Patacchini, Riccardo, Baker-Glenn, Charles, Van de Poël, Hervé, Blackaby, Wesley, Nash, Kevin, Armani, Elisabetta
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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BAKER-GLENN, Charles, BRUNO, Paolo, FIORELLI, Claudio, VAN DE POËL, Hervè, BIAGETTI, Matteo
Year of Publication 06.06.2024
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Year of Publication 06.06.2024
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PHTHALAZINE DERIVATIVES AS P2X3 INHIBITORS
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Year of Publication 04.01.2024
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Year of Publication 04.01.2024
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(AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS
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Year of Publication 28.12.2023
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Year of Publication 28.12.2023
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PHTHALAZINE DERIVATIVES AS P2X3 INHIBITORS
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Year of Publication 04.10.2023
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Year of Publication 04.10.2023
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(AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS
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Year of Publication 04.10.2023
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BAKER-GLENN, Charles, BRUNO, Paolo, FIORELLI, Claudio, VAN DE POËL, Hervè, BIAGETTI, Matteo
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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(AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS
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Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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AZETIDINE DERIVATIVES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE 1 INHIBITORS
RIZZI, Andrea, GUARIENTO, Sara, ARMANI, Elisabetta, VAN DE POËL, Hervè Pierre Clotaire, VATER, Huw David
Year of Publication 11.01.2024
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Year of Publication 11.01.2024
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Synthesis of 6,7,8,9-tetrahydropyrido[2,3- b ]indolizine and 3,4-dihydro-2 H -pyrido[2′,3′:4,5]pyrrolo[2,1- b ][1,3]oxazine derivatives as new melatonin receptor ligands
Van de Poël, Hervé, Guillaumet, Gérald, Viaud-Massuard, Marie-Claude
Published in Tetrahedron letters (01.02.2002)
Published in Tetrahedron letters (01.02.2002)
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Year of Publication 06.07.2023
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Year of Publication 06.07.2023
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PHTHALAZINE DERIVATIVES AS P2X3 INHIBITORS
BAKER-GLENN, Charles, BRUNO, Paolo, FIORELLI, Claudio, VAN DE POËL, Hervè, BIAGETTI, Matteo
Year of Publication 02.06.2022
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Year of Publication 02.06.2022
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(AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS
BAKER-GLENN, Charles, BRUNO, Paolo, FIORELLI, Claudio, VAN DE POËL, Hervè, BIAGETTI, Matteo
Year of Publication 02.06.2022
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Year of Publication 02.06.2022
Patent