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Published in Bioorganic & medicinal chemistry letters (01.10.2019)
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Rational Design and Synthesis of 4-((1R,2R)-2-Hydroxycyclohexyl)-2(trifluoromethyl)benzonitrile (PF-998425), a Novel, Nonsteroidal Androgen Receptor Antagonist Devoid of Phototoxicity for Dermatological Indications
Li, Jie Jack, Iula, Donna M, Nguyen, Maria N, Hu, Lain-Yen, Dettling, Danielle, Johnson, Theodore R, Du, Daniel Y, Shanmugasundaram, Veerabahu, Van Camp, Jennifer A, Wang, Zhi, Harter, William G, Yue, Wen-Song, Boys, Mark L, Wade, Kimberly J, Drummond, Elena M, Samas, Brian M, Lefker, Bruce A, Hoge, Garrett S, Lovdahl, Mark J, Asbill, Jeffrey, Carroll, Matthew, Meade, Mary Ann, Ciotti, Susan M, Krieger-Burke, Theresa
Published in Journal of medicinal chemistry (13.11.2008)
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Preparation of 4-aryl-2-trifluoromethylbenzonitrile derivatives as androgen receptor antagonists for topical suppression of sebum production
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Published in Bioorganic & medicinal chemistry letters (15.10.2007)
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Aminopyrrolidineamide inhibitors of site-1 protease
Hay, Bruce A., Abrams, Barbara, Zumbrunn, Allice Y., Valentine, James J., Warren, Laurie C., Petras, Stephen F., Shelly, Lorraine D., Xia, Angela, Varghese, Alison H., Hawkins, Julie L., Van Camp, Jennifer A., Robbins, Michael D., Landschulz, Katherine, Harwood, H. James
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
FRANK KRISTINE E, HOEMANN MICHAEL Z, WILSON NOEL S, OSUMA AUGUSTINE, SHEPPARD GEORGE, BONAFOUX DOMINIQUE, VAN CAMP JENNIFER, VAN EPPS STACY A, HUNTLEY RAYMOND, SOMAL GAGANDEEP K, XU XIANGDONG, WALLACE GRIER A, WANG LU, DAVIS HEATHER M, FRIEDMAN MICHAEL M, VASUDEVAN ANIL, HEROLD J. MARTIN, WANG ZHI
Year of Publication 08.03.2016
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Year of Publication 08.03.2016
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A scalable approach to diaminopyrazoles using flow chemistry
Wilson, Noel S., Osuma, Augustine T., Camp, Jennifer A.Van, Xu, Xiangdong
Published in Tetrahedron letters (22.08.2012)
Published in Tetrahedron letters (22.08.2012)
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ChemInform Abstract: A Scalable Approach to Diaminopyrazoles Using Flow Chemistry
Wilson, Noel S., Osuma, Augustine T., Van Camp, Jennifer A., Xu, Xiangdong
Published in ChemInform (27.11.2012)
Published in ChemInform (27.11.2012)
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
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Year of Publication 08.06.2022
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Year of Publication 08.06.2022
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Primary carboxamides as btk inhibitors
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Year of Publication 25.06.2021
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Year of Publication 25.06.2021
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Primary carboxamides as btk inhibitors
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Year of Publication 25.06.2021
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Year of Publication 25.06.2021
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
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Year of Publication 12.10.2021
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Year of Publication 12.10.2021
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
Frank, Kristine E, Osuma, Augustine, Van Epps, Stacy Anne, Wang, Zhi, Bonafoux, Dominique, Huntley, Raymond, Sheppard, George, Van Camp, Jennifer, Xu, Xiangdong, Friedman, Michael M, Wallace, Grier Allan, Somal, Gagandeep Kaur, Vasudevan, Anil, Hoemann, Michael Z, Davis, Heather Michele, Wilson, Noel S, Wang, Lu, Herold, J. Martin
Year of Publication 17.06.2021
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Year of Publication 17.06.2021
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Primary carboxamides as BTK inhibitors
FRANK, Kristine E, BONAFOUX, Dominique, OSUMA, Augustine, HUNTLEY, Raymond, VASUDEVAN, Anil, WANG Zhi, DAVIS, Heather M, HEROLD, J. Martin, HOEMANN, Michael Z, VAN CAMP, Jennifer, WILSON, Noel S, FRIEDMAN, Michael M, SHEPPARD, George, VAN EPPS, Stacy A, SOMAL, Gagandeep K, XU, Xiangdong, WALLACE, Grier A, WANG, Lu
Year of Publication 25.03.2021
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Year of Publication 25.03.2021
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
FRANK, Kristine E, BONAFOUX, Dominique, OSUMA, Augustine, HUNTLEY, Raymond, VASUDEVAN, Anil, DAVIS, Heather M, HEROLD, J. Martin, HOEMANN, Michael Z, VAN CAMP, Jennifer, WILSON, Noel S, FRIEDMAN, Michael M, SHEPPARD, George, VAN EPPS, Stacy A, SOMAL, Gagandeep K, XU, Xiangdong, WALLACE, Grier A, WANG, Lu, WANG, Zhi
Year of Publication 27.05.2020
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Year of Publication 27.05.2020
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
HEROLD, J, BONAFOUX, Dominique, OSUMA, Augustine, HOEMANN, Michael, VAN EPPS, Stacy, WILSON, Noel, HUNTLEY, Raymond, VASUDEVAN, Anil, SOMAL, Gagandeep, DAVIS, Heather, VAN CAMP, Jennifer, SHEPPARD, George, WALLACE, Grier, XU, Xiangdong, FRIEDMAN, Michael, FRANK, Kristine, WANG, Lu, WANG, Zhi
Year of Publication 28.03.2019
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Year of Publication 28.03.2019
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
HEROLD, J, BONAFOUX, Dominique, OSUMA, Augustine, HOEMANN, Michael, VAN EPPS, Stacy, WILSON, Noel, HUNTLEY, Raymond, VASUDEVAN, Anil, SOMAL, Gagandeep, DAVIS, Heather, VAN CAMP, Jennifer, SHEPPARD, George, WALLACE, Grier, XU, Xiangdong, FRIEDMAN, Michael, FRANK, Kristine, WANG, Lu, WANG, Zhi
Year of Publication 10.01.2019
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Year of Publication 10.01.2019
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
FRANK, Kristine E, BONAFOUX, Dominique, OSUMA, Augustine, HUNTLEY, Raymond, VASUDEVAN, Anil, DAVIS, Heather M, HEROLD, J. Martin, HOEMANN, Michael Z, VAN CAMP, Jennifer, WILSON, Noel S, FRIEDMAN, Michael M, SHEPPARD, George, VAN EPPS, Stacy A, SOMAL, Gagandeep K, XU, Xiangdong, WALLACE, Grier A, WANG, Lu, WANG, Zhi
Year of Publication 20.10.2019
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Year of Publication 20.10.2019
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
Frank, Kristine E, Osuma, Augustine, Van Epps, Stacy Anne, Wang, Zhi, Bonafoux, Dominique, Huntley, Raymond, Sheppard, George, Van Camp, Jennifer, Xu, Xiangdong, Friedman, Michael M, Wallace, Grier Allan, Somal, Gagandeep Kaur, Vasudevan, Anil, Hoemann, Michael Z, Davis, Heather Michele, Wilson, Noel S, Wang, Lu, Herold, J. Martin
Year of Publication 19.09.2019
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Year of Publication 19.09.2019
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PRIMARY CARBOXAMIDES AS BTK INHIBITORS
VAN EPPS, STACY A, HUNTLEY, RAYMOND, WALLACE, GRIER A, DAVIS, HEATHER M, SOMAL, GAGANDEEP K, WANG, ZHI, SHEPPARD, GEORGE, VAN CAMP, JENNIFER, WANG, LU, OSUMA, AUGUSTINE, FRIEDMAN, MICHAEL M, VASUDEVAN, ANIL, FRANK, KRISTINE E, BONAFOUX, DOMINIQUE, XU, XIANGDONG, HEROLD, J. MARTIN, WILSON, NOEL S, HOEMANN, MICHAEL Z
Year of Publication 28.06.2019
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Year of Publication 28.06.2019
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