FKBPL and its peptide derivatives inhibit endocrine therapy resistant cancer stem cells and breast cancer metastasis by downregulating DLL4 and Notch4
McClements, Lana, Annett, Stephanie, Yakkundi, Anita, O'Rourke, Martin, Valentine, Andrea, Moustafa, Nermeen, Alqudah, Abdelrahim, Simões, Bruno M, Furlong, Fiona, Short, Amy, McIntosh, Stuart A, McCarthy, Helen O, Clarke, Robert B, Robson, Tracy
Published in BMC cancer (11.04.2019)
Published in BMC cancer (11.04.2019)
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Identification and Characterization of Dual Inhibitors of the USP25/28 Deubiquitinating Enzyme Subfamily
Wrigley, Jonathan D, Gavory, Gerald, Simpson, Iain, Preston, Marian, Plant, Helen, Bradley, Jenna, Goeppert, Anne U, Rozycka, Ewelina, Davies, Gareth, Walsh, Jarrod, Valentine, Andrea, McClelland, Keeva, Odrzywol, Krzysztofa Ewa, Renshaw, Jonathan, Boros, Joanna, Tart, Jonathan, Leach, Lindsey, Nowak, Thorsten, Ward, Richard A, Harrison, Timothy, Andrews, David M
Published in ACS chemical biology (15.12.2017)
Published in ACS chemical biology (15.12.2017)
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Biogenic Amines and Aflatoxins in Some Imported Meat Products: Incidence, Occurrence, and Public Health Impacts
Elabbasy, Mohamed Tharwat, Adeboye, Adeniyi, Abouelkheir, Essam Said, Hussein, Mohamed A., Morshdy, Alaa Eldin, Algahtani, Fahad Dhafer, Valentine, Andrea
Published in Journal of food quality (2020)
Published in Journal of food quality (2020)
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Water challenges and Urban Sustainable Development in Changing Climate: Economic Growth Agenda for Global South
Raza, Tabassam, C. Rentoy, Frederika, Ahmed, Nisar, Thess Khas S. Raza, Andrea Valentine L. Andres, E. Marasigan, Karl Michael, M. Espinosa, Ramon Iñigo
Published in European journal of sustainable development (01.10.2019)
Published in European journal of sustainable development (01.10.2019)
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Extreme weather disasters challenges for sustainable development: Innovating a science and policy framework for disaster-resilient and sustainable Quezon City, Philippines
Raza, Tabassam, Liwag, Carmelita R.E.U., Andres, Andrea Valentine L., Castro, Jun T., Cuña, Aldrin C., Vinarao, Vincent G., Raza, Thess Khaz S., Marasigan, Karl Michael E., Espinosa, Ramon Iñigo M., Rentoy, Frederika C., Perez, Bianca D., Ahmed, Nisar
Published in Progress in disaster science (01.01.2020)
Published in Progress in disaster science (01.01.2020)
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Evaluation of the Antiangiogenic Potential of AQ4N
O'ROURKE, Martin, WARD, Claire, WORTHINGTON, Jenny, MCKENNA, Julie, VALENTINE, Andrea, ROBSON, Tracy, HIRST, David G, MCKEOWN, Stephanie R
Published in Clinical cancer research (01.03.2008)
Published in Clinical cancer research (01.03.2008)
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Discovery of a Novel Class of D-Amino Acid Oxidase Inhibitors Usingthe Schro?dinger Computational Platform
Tang, Haifeng, Jensen, Kristian, Houang, Evelyne, McRobb, Fiona M., Bhat, Sathesh, Svensson, Mats, Bochevarov, Art, Day, Tyler, Dahlgren, Markus K., Bell, Jeffery A., Frye, Leah, Skene, Robert J., Lewis, James H., Osborne, James D., Tierney, Jason P., Gordon, James A., Palomero, Maria A., Gallati, Caroline, Chapman, Robert S. L., Jones, Daniel R., Hirst, Kim L., Sephton, Mark, Chauhan, Alka, Sharpe, Andrew, Tardia, Piero, Dechaux, Elsa A., Taylor, Andrea, Waddell, Ross D., Valentine, Andrea, Janssens, Holden B., Aziz, Omar, Bloomfield, Dawn E., Ladha, Sandeep, Fraser, Ian J., Ellard, John M.
Published in Journal of medicinal chemistry (12.05.2022)
Published in Journal of medicinal chemistry (12.05.2022)
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Journal Article
Discovery of a Novel Class of d‑Amino Acid Oxidase Inhibitors Using the Schrödinger Computational Platform
Tang, Haifeng, Jensen, Kristian, Houang, Evelyne, McRobb, Fiona M., Bhat, Sathesh, Svensson, Mats, Bochevarov, Art, Day, Tyler, Dahlgren, Markus K., Bell, Jeffery A., Frye, Leah, Skene, Robert J., Lewis, James H., Osborne, James D., Tierney, Jason P., Gordon, James A., Palomero, Maria A., Gallati, Caroline, Chapman, Robert S. L., Jones, Daniel R., Hirst, Kim L., Sephton, Mark, Chauhan, Alka, Sharpe, Andrew, Tardia, Piero, Dechaux, Elsa A., Taylor, Andrea, Waddell, Ross D., Valentine, Andrea, Janssens, Holden B., Aziz, Omar, Bloomfield, Dawn E., Ladha, Sandeep, Fraser, Ian J., Ellard, John M.
Published in Journal of medicinal chemistry (12.05.2022)
Published in Journal of medicinal chemistry (12.05.2022)
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Journal Article
Discovery of a Novel Class of d-Amino Acid Oxidase Inhibitors Using the Schrödinger Computational Platform
Tang, Haifeng, Jensen, Kristian, Houang, Evelyne, McRobb, Fiona M, Bhat, Sathesh, Svensson, Mats, Bochevarov, Art, Day, Tyler, Dahlgren, Markus K, Bell, Jeffery A, Frye, Leah, Skene, Robert J, Lewis, James H, Osborne, James D, Tierney, Jason P, Gordon, James A, Palomero, Maria A, Gallati, Caroline, Chapman, Robert S L, Jones, Daniel R, Hirst, Kim L, Sephton, Mark, Chauhan, Alka, Sharpe, Andrew, Tardia, Piero, Dechaux, Elsa A, Taylor, Andrea, Waddell, Ross D, Valentine, Andrea, Janssens, Holden B, Aziz, Omar, Bloomfield, Dawn E, Ladha, Sandeep, Fraser, Ian J, Ellard, John M
Published in Journal of medicinal chemistry (12.05.2022)
Published in Journal of medicinal chemistry (12.05.2022)
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Journal Article
FKBPL and Peptide Derivatives: Novel Biological Agents that Inhibit Angiogenesis by a CD44-Dependent Mechanism
VALENTINE, Andrea, O'ROURKE, Martin, MCKEEN, Hayley, WAUGH, David J. J, ROBERTS, Jennifer, MCGREGOR, Joanne, COTTON, Graham, JAMES, Lain, HARRISON, Timothy, HIRST, David G, ROBSON, Tracy, YAKKUNDI, Anita, WORTHINGTON, Jenny, HOOKHAM, Michelle, BICKNELL, Roy, MCCARTHY, Helen O, MCCLELLAND, Keeva, MCCALLUM, Lynn, DYER, Hayder
Published in Clinical cancer research (01.03.2011)
Published in Clinical cancer research (01.03.2011)
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Journal Article
FKBPL Regulates Estrogen Receptor Signaling and Determines Response to Endocrine Therapy
MCKEEN, Hayley D, BYRNE, Christopher, ROBSON, Tracy, JITHESH, Puthen V, DONLEY, Christopher, VALENTINE, Andrea, YAKKUNDI, Anita, O'ROURKE, Martin, SWANTON, Charles, MCCARTHY, Helen O, HIRST, David G
Published in Cancer research (Chicago, Ill.) (01.02.2010)
Published in Cancer research (Chicago, Ill.) (01.02.2010)
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Journal Article
A Novel FK506-Like Binding Protein Interacts with the Glucocorticoid Receptor and Regulates Steroid Receptor Signaling
McKeen, Hayley D, McAlpine, Kerry, Valentine, Andrea, Quinn, Derek J, McClelland, Keeva, Byrne, Christopher, O'Rourke, Martin, Young, Sheila, Scott, Christopher J, McCarthy, Helen O, Hirst, David G, Robson, Tracy
Published in Endocrinology (Philadelphia) (01.11.2008)
Published in Endocrinology (Philadelphia) (01.11.2008)
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Journal Article
Abstract 3288: The anti-tumour efficacy of the novel peptide inhibitor of angiogenesis ALM-201
O'Rourke, Martin, Valentine, Andrea, McLean, Estelle, Page, Natalie, Cotton, Graham, Robson, Tracy, Hirst, David, Harrison, Timothy, James, Iain
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Journal Article
FKBP-L polypeptides and uses in angiogenesis-mediated disorders
Robson, Tracy, O'Rourke, Martin Gerard, Valentine, Andrea, Hirst, David
Year of Publication 03.03.2020
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Year of Publication 03.03.2020
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