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Published in International journal of pharmaceutics (31.03.2009)
Published in International journal of pharmaceutics (31.03.2009)
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Phase I Dose-Escalation Study of the Novel Antiandrogen BMS-641988 in Patients with Castration-Resistant Prostate Cancer
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Metabolism and Disposition of [14C]BMS-690514, an ErbB/Vascular Endothelial Growth Factor Receptor Inhibitor, after Oral Administration to Humans
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Published in Drug metabolism and disposition (01.11.2010)
Published in Drug metabolism and disposition (01.11.2010)
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Phase I Dose-Escalation Study of the Novel Anti-androgen BMS-641988 in Patients with Castration-Resistant Prostate Cancer
Rathkopf, Dana, Liu, Glenn, Carducci, Michael A, Eisenberger, Mario A, Anand, Aseem, Morris, Michael J, Slovin, Susan F, Sasaki, Yasutsuna, Takahashi, Shunji, Ozono, Seiichiro, Fung, Nga Kit Eliza, Cheng, Shinta, Gan, Jinping, Gottardis, Marco, Obermeier, Mary T., Reddy, Jyotsna, Zhang, Steven, Vakkalagadda, Blisse J., Wilding, George, Scher, Howard I.
Published in Clinical cancer research (03.12.2010)
Published in Clinical cancer research (03.12.2010)
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Fremgangsmåte for fremstilling av triazol substituerte azaindoloksoeddikpiperazinderivater
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Year of Publication 28.08.2017
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Year of Publication 28.08.2017
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PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
SIRARD, PIERRE, NATALIE, JR., KENNETH, J, LAI, CHIAJEN, KUANG, SHAN-MING, GAO, QI, DROGHINI, ROBERTO, QIAN, XINHUA, PACK, SHAWN, K, VAKKALAGADDA, BLISSE, J, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL, G, KRONENTHAL, DAVID, R, LAJEUNESSE, JEAN, TANG, ERQING, QIU, YUPING, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, QIAN, FENG, HU, WENHAO
Year of Publication 27.07.2011
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Year of Publication 27.07.2011
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Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein
Soundararajan, Nachimuthu, Qiu, Yuping, Hu, Wenhao, Kronenthal, David R, Sirard, Pierre, Lajeunesse, Jean, Droghini, Robert, Chidambaram, Ramakrishnan, Qian, Xinhua, Natalie, Kenneth J, Pack, Shawn K, Reising, Nathan, Tang, Erqing, Fakes, Michael G, Gao, Qi, Qian, Feng, Vakkalagadda, Blisse J, Lai, Chiajen, Kuang, Shan-Ming
Year of Publication 28.06.2011
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Year of Publication 28.06.2011
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Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein
TANG ERQING, REISING NATHAN, FAKES MICHAEL G, PACK SHAWN K, VAKKALAGADDA BLISSE J, QIAN XINHUA, DROGHINI ROBERT, NATALIE KENNETH J, CHIDAMBARAM RAMAKRISHNAN, KUANG SHAN-MING, SOUNDARARAJAN NACHIMUTHU, SIRARD PIERRE, LAJEUNESSE JEAN, KRONENTHAL DAVID R, LAI CHIAJEN, HU WENHAO, GAO QI, QIU YUPING, QIAN FENG
Year of Publication 28.06.2011
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Year of Publication 28.06.2011
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PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
TANG ERQING, REISING NATHAN, FAKES MICHAEL G, PACK SHAWN K, VAKKALAGADDA BLISSE J, QIAN XINHUA, DROGHINI ROBERT, NATALIE KENNETH J, CHIDAMBARAM RAMAKRISHNAN, KUANG SHAN-MING, SOUNDARARAJAN NACHIMUTHU, SIRARD PIERRE, LAJEUNESSE JEAN, KRONENTHAL DAVID R, LAI CHIAJEN, HU WENHAO, GAO QI, QIU YUPING, QIAN FENG
Year of Publication 25.03.2010
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Year of Publication 25.03.2010
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Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein
TANG ERQING, REISING NATHAN, FAKES MICHAEL G, PACK SHAWN K, VAKKALAGADDA BLISSE J, QIAN XINHUA, DROGHINI ROBERT, NATALIE KENNETH J, CHIDAMBARAM RAMAKRISHNAN, KUANG SHAN-MING, SOUNDARARAJAN NACHIMUTHU, SIRARD PIERRE, LAJEUNESSE JEAN, KRONENTHAL DAVID R, LAI CHIAJEN, HU WENHAO, GAO QI, QIU YUPING, QIAN FENG
Year of Publication 13.10.2009
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Year of Publication 13.10.2009
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Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein
Soundararajan, Nachimuthu, Qiu, Yuping, Hu, Wenhao, Kronenthal, David R, Sirard, Pierre, Lajeunesse, Jean, Droghini, Robert, Chidambaram, Ramakrishnan, Qian, Xinhua, Natalie, Kenneth J, Pack, Shawn K, Reising, Nathan, Tang, Erqing, Fakes, Michael G, Gao, Qi, Qian, Feng, Vakkalagadda, Blisse J, Lai, Chiajen, Kuang, Shan-Ming
Year of Publication 13.10.2009
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Year of Publication 13.10.2009
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PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
SIRARD, PIERRE, NATALIE, JR., KENNETH, J, LAI, CHIAJEN, QUIAN, FENG, KUANG, SHAN-MING, GAO, QI, DROGHINI, ROBERTO, QIAN, XINHUA, PACK, SHAWN, K, VAKKALAGADDA, BLISSE, J, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL, G, KRONENTHAL, DAVID, R, LAJEUNESSE, JEAN, TANG, ERQING, QIU, YUPING, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, HU, WENHAO
Year of Publication 09.04.2008
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Year of Publication 09.04.2008
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PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
SIRARD, PIERRE, NATALIE, JR., KENNETH, J, LAI, CHIAJEN, KUANG, SHAN-MING, GAO, QI, DROGHINI, ROBERTO, QIAN, XINHUA, PACK, SHAWN, K, VAKKALAGADDA, BLISSE, J, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL, G, KRONENTHAL, DAVID, R, LAJEUNESSE, JEAN, TANG, ERQING, QIU, YUPING, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, QIAN, FENG, HU, WENHAO
Year of Publication 12.07.2007
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Year of Publication 12.07.2007
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PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
SIRARD, PIERRE, NATALIE, JR., KENNETH, J, LAI, CHIAJEN, KUANG, SHAN-MING, GAO, QI, DROGHINI, ROBERTO, QIAN, XINHUA, PACK, SHAWN, K, VAKKALAGADDA, BLISSE, J, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL, G, KRONENTHAL, DAVID, R, LAJEUNESSE, JEAN, TANG, ERQING, QIU, YUPING, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, QIAN, FENG, HU, WENHAO
Year of Publication 01.03.2007
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Year of Publication 01.03.2007
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PROCESS FOR PREPARING TRIAZOLE SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES AND NOVEL SALT FORMS PRODUCED THEREIN
SIRARD, PIERRE, NATALIE, JR., KENNETH, J, LAI, CHIAJEN, KUANG, SHAN-MING, GAO, QI, DROGHINI, ROBERTO, QIAN, XINHUA, PACK, SHAWN, K, VAKKALAGADDA, BLISSE, J, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL, G, KRONENTHAL, DAVID, R, LAJEUNESSE, JEAN, TANG, ERQING, QIU, YUPING, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, QIAN, FENG, HU, WENHAO
Year of Publication 04.01.2007
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Year of Publication 04.01.2007
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Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein
TANG ERQING, REISING NATHAN, FAKES MICHAEL G, PACK SHAWN K, VAKKALAGADDA BLISSE J, QIAN XINHUA, DROGHINI ROBERT, NATALIE KENNETH J, CHIDAMBARAM RAMAKRISHNAN, KUANG SHAN-MING, SOUNDARARAJAN NACHIMUTHU, SIRARD PIERRE, LAJEUNESSE JEAN, KRONENTHAL DAVID R, LAI CHIAJEN, HU WENHAO, GAO QI, QIU YUPING, QIAN FENG
Year of Publication 28.12.2006
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Year of Publication 28.12.2006
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Fremgangsmåte for fremstilling av triazol substituerte azaindoloksoeddikpiperazinderivater og nye saltformer derved fremstilt
TANG ERQING, REISING NATHAN, FAKES MICHAEL G, PACK SHAWN K, VAKKALAGADDA BLISSE J, QIAN XINHUA, DROGHINI ROBERTO, NATHALIE KENNETH J, CHIDAMBARAM RAMAKRISHNAN, KUANG SHAN-MING, SOUNDARARAJAN NACHIMUTHU, SIRARD PIERRE, LAJEUNESSE JEAN, KRONENTHAL DAVID R, LAI CHIAJEN, GAO QI, HU WENHAO, QIU YUPING, QIAN FENG
Year of Publication 18.03.2008
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Year of Publication 18.03.2008
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Process for preparing triazole substituted azaindoleoxoacetic piperazine derivatives and novel salt forms produced therein
SIRARD, PIERRE, LAI, CHIAJEN, PACK, SHAWN K, KUANG, SHAN-MING, GAO, QI, VAKKALAGADDA, BLISSE J, DROGHINI, ROBERTO, QIU, YU-PING, HU, WEN-HAO, QIAN, XINHUA, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL G, LAJEUNESSE, JEAN, TANG, ERQING, KRONENTHAL, DAVID R, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, QIAN, FENG, NATALIE, KENNETH J. JR
Year of Publication 01.11.2007
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Year of Publication 01.11.2007
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DERIVADOS DE PIPERAZINA AZAINDOLOXOACETICA SUSTITUIDA, FORMA CRISTALINA DEL DERIVADO 1,2,3-TRIAZOL, PROCESOS DE PREPARACION DE LOS MISMOS Y COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN
SIRARD, PIERRE, LAI, CHIAJEN, PACK, SHAWN K, KUANG, SHAN-MING, GAO, QI, VAKKALAGADDA, BLISSE J, DROGHINI, ROBERTO, QIAN, XINHUA, CHIDAMBARAM, RAMAKRISHNAN, FAKES, MICHAEL G, LAJEUNESSE, JEAN, TANG, ERQING, QIU, YUPING, KRONENTHAL, DAVID R, SOUNDARARAJAN, NACHIMUTHU, REISING, NATHAN, QIAN, FENG, HU, WENHAO, NATALIE, KENNETH J. JR
Year of Publication 05.09.2007
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Year of Publication 05.09.2007
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PROCESO PARA PREPARAR DERIVADOS DE PIPERAZINA AZINDOLOXOACETICA SUSTITUIDA CON TRIAZOL Y NUEVAS FORMAS DE SAL PRODUCIDAS DE LOS MISMOS
NATALIE, FAKES MICHAEL G, PACK SHAWN K, VAKKALAGADDA BLISSE J, QIAN XINHUA, DROGHINI ROBERTO, TANG ERQUING, KUANG SHAN-MING, CHIDAMBARAM RAMAKRISHNAN, SOUNDARARAJAN NACHIMUTHU, SIRARD PIERRE, LAJEUNESSE JEAN, KRONENTHAL DAVID R, LAI CHIAJEN, HU WENHAO, GAO QI, QIU YUPING, QIAN FENG
Year of Publication 11.03.2007
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Year of Publication 11.03.2007
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