Abstract P141: Preclinical characterization of LOX-24350, a highly potent and isoform-selective FGFR3 inhibitor
Ballard, Joshua A., Kercher, Timothy, Abraham, David, Brecht, Ryan, Brooks, Nathan A., Buckles, Thomas, Bume, Desta, Busha, David, Cedervall, Ernst Peder, Condroski, Kevin, Ebata, Kevin, Gharbi, Severine Isabelle, Hazlitt, Robert, Morales, Tony, Patel, Nisha, Podoll, Jessica, Urkalan, Kaveri, Villalain, Sandra Gomez, Walls, Shane, Watson, Faith, Yang, Peiyi, Brandhuber, Barbara J., Andrews, Steven W.
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Journal Article
Abstract 1302: Targeting hormone receptor-dependent cancers with potent, selective and orally-available small molecule inhibitors of eIF4E
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Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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FGFR3 억제제 화합물
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Year of Publication 11.09.2023
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Year of Publication 11.09.2023
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NILEWSKI CHRISTIAN, PACKARD GARRICK KENNETH, MICHELS THEO, SPRENGELER PAUL A, MUKAIYAMA TAKASUKE, URKALAN KAVERI, ERNST JUSTIN T, XIANG ALAN X, SHAGHAFI MIKE, SPERRY SAMUEL, GRUBBS ALAN, REICH SIEGFRIED H, TRAN CHINH VIET
Year of Publication 13.05.2022
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Year of Publication 13.05.2022
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SMALL MOLECULE INHIBITORS OF FIBROSIS
BOLLONG MICHAEL, YANG BAIYUAN, CHATTERJEE ARNAB K, KUMAR PUNEET, SCHULTZ PETER G, LAIRSON LUKE, URKALAN KAVERI
Year of Publication 14.03.2016
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Year of Publication 14.03.2016
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ITRACONAZOLE ANALOGS AS INHIBITORS OF FIBROSIS
URKALAN, Kaveri, SCHULTZ, Peter, G, CHATTERJEE, Arnab, K, YANG, Baiyuan, BOLLONG, Michael, KUMAR, Puneet, LAIRSON, Luke
Year of Publication 07.08.2024
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Year of Publication 07.08.2024
Patent