Deactivatable Bisubstrate Inhibitors of Protein Kinases
Sõrmus, Tanel, Lavogina, Darja, Enkvist, Erki, Uri, Asko, Viht, Kaido
Published in Molecules (Basel, Switzerland) (01.10.2022)
Published in Molecules (Basel, Switzerland) (01.10.2022)
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Conjugates of adenosine mimetics and arginine‐rich peptides serve as inhibitors and fluorescent probes but not as long‐lifetime photoluminescent probes for protein arginine methyltransferases
Lavogina, Darja, Nasirova, Naila, Sõrmus, Tanel, Tähtjärv, Taavo, Enkvist, Erki, Viht, Kaido, Haljasorg, Tõiv, Herodes, Koit, Jaal, Jana, Uri, Asko
Published in Journal of peptide science (01.03.2023)
Published in Journal of peptide science (01.03.2023)
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Journal Article
Competitive ligands facilitate dissociation of the complex of bifunctional inhibitor and protein kinase
Ivan, Taavi, Enkvist, Erki, Sinijarv, Hedi, Uri, Asko
Published in Biophysical chemistry (01.09.2017)
Published in Biophysical chemistry (01.09.2017)
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Almost complete radiationless energy transfer from excited triplet state of a dim phosphor to a covalently linked adjacent fluorescent dye in purely organic tandem luminophores doped into PVA matrix
Jõgela, Joana, Uri, Asko, Pålsson, Lars-Olof, Enkvist, Erki
Published in Journal of materials chemistry. C, Materials for optical and electronic devices (2019)
Published in Journal of materials chemistry. C, Materials for optical and electronic devices (2019)
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Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM Family
Nonga, Olivier E., Lavogina, Darja, Enkvist, Erki, Kestav, Katrin, Chaikuad, Apirat, Dixon-Clarke, Sarah E., Bullock, Alex N., Kopanchuk, Sergei, Ivan, Taavi, Ekambaram, Ramesh, Viht, Kaido, Knapp, Stefan, Uri, Asko
Published in Molecules (Basel, Switzerland) (19.07.2021)
Published in Molecules (Basel, Switzerland) (19.07.2021)
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Acetoxymethyl Ester of Tetrabromobenzimidazole–Peptoid Conjugate for Inhibition of Protein Kinase CK2 in Living Cells
Viht, Kaido, Saaver, Siiri, Vahter, Jürgen, Enkvist, Erki, Lavogina, Darja, Sinijärv, Hedi, Raidaru, Gerda, Guerra, Barbara, Issinger, Olaf-Georg, Uri, Asko
Published in Bioconjugate chemistry (16.12.2015)
Published in Bioconjugate chemistry (16.12.2015)
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Phosphorylation of Notch1 by Pim kinases promotes oncogenic signaling in breast and prostate cancer cells
Santio, Niina M, Landor, Sebastian K-J, Vahtera, Laura, Ylä-Pelto, Jani, Paloniemi, Elina, Imanishi, Susumu Y, Corthals, Garry, Varjosalo, Markku, Manoharan, Ganesh Babu, Uri, Asko, Lendahl, Urban, Sahlgren, Cecilia, Koskinen, Päivi J
Published in Oncotarget (12.07.2016)
Published in Oncotarget (12.07.2016)
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Journal Article
Conjugation of Adenosine and Hexa-(d-arginine) Leads to a Nanomolar Bisubstrate-Analog Inhibitor of Basophilic Protein Kinases
Enkvist, Erki, Lavogina, Darja, Raidaru, Gerda, Vaasa, Angela, Viil, Indrek, Lust, Marje, Viht, Kaido, Uri, Asko
Published in Journal of medicinal chemistry (30.11.2006)
Published in Journal of medicinal chemistry (30.11.2006)
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Thiazole- and selenazole-comprising high-affinity inhibitors possess bright microsecond-scale photoluminescence in complex with protein kinase CK2
Vahter, Jürgen, Viht, Kaido, Uri, Asko, Manoharan, Ganesh babu, Enkvist, Erki
Published in Bioorganic & medicinal chemistry (01.10.2018)
Published in Bioorganic & medicinal chemistry (01.10.2018)
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Journal Article
Discovery of strong inhibitory properties of a monoclonal antibody of PKA and use of the antibody and a competitive photoluminescent orthosteric probe for analysis of the protein kinase
Nonga, Olivier Etebe, Lavogina, Darja, Ivan, Taavi, Viht, Kaido, Enkvist, Erki, Uri, Asko
Published in Biochimica et biophysica acta. Proteins and proteomics (01.08.2020)
Published in Biochimica et biophysica acta. Proteins and proteomics (01.08.2020)
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