Interaction of SSR161421, a novel specific adenosine A(3) receptor antagonist with adenosine A(3) receptor agonists both in vitro and in vivo
Mikus, Endre G, Boér, Kinga, Timári, Géza, Urbán-Szabó, Katalin, Kapui, Zoltán, Szeredi, Judit, Gerber, Katalin, Szabó, Tibor, Bátori, Sándor, Finet, Michel, Arányi, Péter, Galzin, Anne-Marie
Published in European journal of pharmacology (15.01.2013)
Published in European journal of pharmacology (15.01.2013)
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A novel orally active inhibitor of HLE
Varga, Márton, Kapui, Zoltán, Bátori, Sándor, Nagy, Lajos T., Vasvári-Debreczy, Lelle, Mikus, Endre, Urbán-Szabó, Katalin, Arányi, Péter
Published in European journal of medicinal chemistry (01.04.2003)
Published in European journal of medicinal chemistry (01.04.2003)
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Biochemical and Pharmacological Characterization of 2-(9-(2-Piperidinoethoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yloxymethyl)-4-(1-methylethyl)-6-methoxy-1,2-benzisothiazol-3(2H)-one-1,1-dioxide (SSR69071), a Novel, Orally Active Elastase Inhibitor
Kapui, Zoltan, Varga, Marton, Urban-Szabo, Katalin, Mikus, Endre, Szabo, Tibor, Szeredi, Judit, Batori, Sandor, Finance, Olivier, Aranyi, Peter
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
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Journal Article
Interaction of SSR161421, a novel specific adenosine A3 receptor antagonist with adenosine A3 receptor agonists both in vitro and in vivo
Mikus, Endre G., Boér, Kinga, Timári, Géza, Urbán-Szabó, Katalin, Kapui, Zoltán, Szeredi, Judit, Gerber, Katalin, Szabó, Tibor, Bátori, Sándor, Finet, Michel, Arányi, Péter, Galzin, Anne-Marie
Published in European journal of pharmacology (15.01.2013)
Published in European journal of pharmacology (15.01.2013)
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Journal Article
SSR240612 [(2R)-2-[((3R)-3-(1,3-Benzodioxol-5-yl)-3-{[(6-methoxy-2-naphthyl)sulfonyl]amino}propanoyl)amino]-3-(4-{[2R,6S)-2,6-dimethylpiperidinyl]methyl}phenyl)-N-isopropyl-N-methylpropanamide Hydrochloride], a New Nonpeptide Antagonist of the Bradykinin B1 Receptor: Biochemical and Pharmacological Characterization
Gougat, Jean, Ferrari, Bernard, Sarran, Lionel, Planchenault, Claudine, Poncelet, Martine, Maruani, Jeanne, Alonso, Richard, Cudennec, Annie, Croci, Tiziano, Guagnini, Fabio, Urban-Szabo, Katalin, Martinolle, Jean-Pierre, Soubrié, Philippe, Finance, Olivier, Le Fur, Gérard
Published in The Journal of pharmacology and experimental therapeutics (01.05.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2004)
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Hydantoine derivatives as CD38 inhibitors
BALOGH, MÁRIA, BUZDER-LANTOS, PÉTER, VASAS, ATTILA, BÁTORI, SÁNDOR, KAPUI, ZOLTÁN, FERENCZY, GYÖRGY, SZABÓ, TIBOR, URBÁN-SZABÓ, KATALIN
Year of Publication 12.11.2014
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Year of Publication 12.11.2014
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TRIAZOLO [1, 5-A] QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
SZABÓ, Tibor, KAPUI, Zoltán, SZLÁVIK, Zoltán, FINET, Michel, BOÉR, Kinga, MIKUS, Endre, SUSÁN, Edit, VARGÁNÉ SZEREDI, Judit, URBÁN SZABÓ, Katalin, BÁTORI, Sándor, TÍMÁRI, Géza
Year of Publication 20.06.2012
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Year of Publication 20.06.2012
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Biochemical and Pharmacological Characterization of 2-(9-(2-Piperidinoethoxy)-4-oxo-4 H -pyrido[1,2- a ]pyrimidin-2-yloxymethyl)-4-(1-methylethyl)-6-methoxy-1,2-benzisothiazol-3(2 H )-one-1,1-dioxide (SSR69071), a Novel, Orally Active Elastase Inhibitor
Kapui, Zoltán, Varga, Márton, Urban-Szabó, Katalin, Mikus, Endre, Szabó, Tibor, Szeredi, Judit, Bátori, Sándor, Finance, Olivier, Arányi, Péter
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
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Journal Article
TRIAZOLO [1, 5-A]QUINOLINES AS ADENOSINE A3 RECEPTOR LIGANDS
KAPUI, Zoltán, SZLÁVIK, Zoltán, SZABÓ, Tibor, FINET, Michel, BOÉR, Kinga, TIMÁRI, Géza, MIKUS, Endre, SUSÁN, Edit, VARGÁNÉ SZEREDI, Judit, BÁTORI, Sándor, URBÁN SZABÓ, Katalin
Year of Publication 31.08.2011
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Year of Publication 31.08.2011
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Compounds
Arányi, Péter, Balázs, László, Bata, Imre, Bátori, Sándor, Boronkay, Éva, Kapui, Zoltán, Susán, Edit, Szabó, Tibor, Nagy, Lajos T, Urbán-Szabó, Katalin, Varga, Márton
Year of Publication 24.08.2010
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Year of Publication 24.08.2010
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PYRROLIDINYL-ALKYL-AMIDE DERIVATIVES THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION AS CCR3 RECEPTOR LIGANDS
BARTÁNÉ BODOR, VERONIKA, PAPPNÉ BEHR, ÁGNES, BÁTORI, SÁNDOR, BATA, IMRE, KAPUI, ZOLTÁN, MIKUS, ENDRE, SZLÁVIK, ZOLTÁN, URBÁN-SZABÓ, KATALIN
Year of Publication 10.10.2014
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Year of Publication 10.10.2014
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ΤΡΙΑΖΟΛΟ [1,5-Α] ΚΙΝΟΛΙΝΕΣ ΩΣ ΣΥΝΔΕΤΕΣ ΤΟΥ ΥΠΟΔΟΧΕΑ A3 ΤΗΣ ΑΔΕΝΟΣΙΝΗΣ
SUSÁN EDIT, KAPUI ZOLTÁN, BÁTORI SÁNDOR, URBÁN SZABÓ KATALIN, SZABÓ TIBOR, BOÉR KINGA, VARGÁNÉ SZEREDI JUDIT, TIMÁRI GÉZA, FINET MICHEL, SZLÁVIK ZOLTÁN, MIKUS ENDRE
Year of Publication 07.10.2015
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Year of Publication 07.10.2015
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SSR240612 [(2 R )-2-[((3 R )-3-(1,3-Benzodioxol-5-yl)-3-{[(6-methoxy-2-naphthyl)sulfonyl]amino}propanoyl)amino]-3-(4-{[2 R ,6 S )-2,6-dimethylpiperidinyl]methyl}phenyl)- N -isopropyl- N -methylpropanamide Hydrochloride], a New Nonpeptide Antagonist of the Bradykinin B 1 Receptor: Biochemical and Pharmacological Characterization
Gougat, Jean, Ferrari, Bernard, Sarran, Lionel, Planchenault, Claudine, Poncelet, Martine, Maruani, Jeanne, Alonso, Richard, Cudennec, Annie, Croci, Tiziano, Guagnini, Fabio, Urban-Szabo, Katalin, Martinolle, Jean-Pierre, Soubrié, Philippe, Finance, Olivier, Le Fur, Gérard
Published in The Journal of pharmacology and experimental therapeutics (01.05.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2004)
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NEW COMPOUNDS - DDP - IV difluor
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Year of Publication 12.03.2007
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Year of Publication 12.03.2007
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Imidazoquinoline derivatives and their use as adenosine A3 ligands
Arányi, Péter, Balázs, László, Balogh, Mária, Bátori, Sándor, Boér, Kinga, Gerber, Katalin, Kapui, Zoltán, Mikus, Endre, Tímári, Geza, Lajos, T. Nagy, Urbán-Szabó, Katalin, Szeredi, Judit Vargáné
Year of Publication 13.02.2007
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Year of Publication 13.02.2007
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Aminoquinoline and aminopyridine derivatives and their use as adenosine a3 ligands
Arányi, Peter, Balázs, László, Balogh, Mária, Bata, Imre, Bátori, Sándor, Nagy, Lajos T, Tímári, Geza, Boér, Kinga, Finance, Olivier, Kapui, Zoltán, Mikus, Endre, Szamosvölgyi, Zsuzsanna, Szeleczky, Gábor, Urbán-Szabó, Katalin
Year of Publication 29.11.2005
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Year of Publication 29.11.2005
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QUINOLEINAS DE TRIAZOLO [1, 5-A] COMO LIGANDOS RECEPTORES DE ADENOSINA A3
JUDIT VARGÁNÉ SZEREDI, KINGA BOÉR, SÁNDOR BÁTORI, ZOLTÁN KAPUI, GÉZA TÍMÁRI, TIBOR SZABÓ, EDIT SUSÁN, ENDRE MIKUS, ZOLTÁN SZLÁVIK, MICHEL FINET, KATALIN SZABÓ URBÁN
Year of Publication 15.07.2010
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Year of Publication 15.07.2010
Patent
A Novel Orally Active Inhibitor of HLE
Varga, Marton, Kapui, Zoltan, Batori, Sandor, Nagy, Lajos T., Vasvari-Debreczy, Lelle, Mikus, Endre, Urban-Szabo, Katalin, Aranyi, Peter
Published in ChemInform (16.09.2003)
Published in ChemInform (16.09.2003)
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HYDANTOINE DERIVATIVES AS CD38 INHIBITORS
BALOGH, MÁRIA, BUZDER-LANTOS, PÉTER, URBÁN-SZÁBÓ, KATALIN, VASAS, ATTILA, BÁTORI, SÁNDOR, KAPUI, ZOLTÁN, FERENCZY, GYÖRGY, SZABÓ, TIBOR
Year of Publication 13.11.2014
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Year of Publication 13.11.2014
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Adamantane and azabicyclo-octane and nonane derivatives, process of their preparation and their use as DPP-IV inhibitors
ARANYI PETER,BATA IMRE,BATORI SANDOR,BORONKAY EVA,BOVY PHILIPPE,KAPUI ZOLTAN,SUSAN EDIT,SZABO TIBOR,URBAN-SZABO KATALIN,VARGA MARTON
Year of Publication 11.10.2006
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Year of Publication 11.10.2006
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