Activation of TrkB with TAM-163 results in opposite effects on body weight in rodents and non-human primates
Perreault, Mylène, Feng, Guo, Will, Sarah, Gareski, Tiffany, Kubasiak, David, Marquette, Kimberly, Vugmeyster, Yulia, Unger, Thaddeus J, Jones, Juli, Qadri, Ariful, Hahm, Seung, Sun, Ying, Rohde, Cynthia M, Zwijnenberg, Raphael, Paulsen, Janet, Gimeno, Ruth E
Published in PloS one (20.05.2013)
Published in PloS one (20.05.2013)
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First-in-Class, First-in-Human Phase I Study of Selinexor, a Selective Inhibitor of Nuclear Export, in Patients With Advanced Solid Tumors
Abdul Razak, Albiruni R, Mau-Soerensen, Morten, Gabrail, Nashat Y, Gerecitano, John F, Shields, Anthony F, Unger, Thaddeus J, Saint-Martin, Jean R, Carlson, Robert, Landesman, Yosef, McCauley, Dilara, Rashal, Tami, Lassen, Ulrik, Kim, Richard, Stayner, Lee-Anne, Mirza, Mansoor R, Kauffman, Michael, Shacham, Sharon, Mahipal, Amit
Published in Journal of clinical oncology (01.12.2016)
Published in Journal of clinical oncology (01.12.2016)
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Selective inhibition of nuclear export with selinexor in patients with non-Hodgkin lymphoma
Kuruvilla, John, Savona, Michael, Baz, Rachid, Mau-Sorensen, Paul Morten, Gabrail, Nashat, Garzon, Ramiro, Stone, Richard, Wang, Michael, Savoie, Lynn, Martin, Peter, Flinn, Ian, Jacoby, Meagan, Unger, Thaddeus J., Saint-Martin, Jean-Richard, Rashal, Tami, Friedlander, Sharon, Carlson, Robert, Kauffman, Michael, Shacham, Sharon, Gutierrez, Martin
Published in Blood (15.06.2017)
Published in Blood (15.06.2017)
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A phase 1 clinical trial of single-agent selinexor in acute myeloid leukemia
Garzon, Ramiro, Savona, Michael, Baz, Rachid, Andreeff, Michael, Gabrail, Nashat, Gutierrez, Martin, Savoie, Lynn, Mau-Sorensen, Paul Morten, Wagner-Johnston, Nina, Yee, Karen, Unger, Thaddeus J., Saint-Martin, Jean-Richard, Carlson, Robert, Rashal, Tami, Kashyap, Trinayan, Klebanov, Boris, Shacham, Sharon, Kauffman, Michael, Stone, Richard
Published in Blood (15.06.2017)
Published in Blood (15.06.2017)
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Selective Deletion of Bdnf in the Ventromedial and Dorsomedial Hypothalamus of Adult Mice Results in Hyperphagic Behavior and Obesity
Unger, Thaddeus J, Calderon, German A, Bradley, Leila C, Sena-Esteves, Miguel, Rios, Maribel
Published in The Journal of neuroscience (26.12.2007)
Published in The Journal of neuroscience (26.12.2007)
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Phase IB Study of Selinexor, a First-in-Class Inhibitor of Nuclear Export, in Patients With Advanced Refractory Bone or Soft Tissue Sarcoma
Gounder, Mrinal M, Zer, Alona, Tap, William D, Salah, Samer, Dickson, Mark A, Gupta, Abha A, Keohan, Mary Louise, Loong, Herbert H, D'Angelo, Sandra P, Baker, Stephanie, Condy, Mercedes, Nyquist-Schultz, Kjirsten, Tanner, Lanier, Erinjeri, Joseph P, Jasmine, Francis H, Friedlander, Sharon, Carlson, Robert, Unger, Thaddeus J, Saint-Martin, Jean-Richard, Rashal, Tami, Ellis, Joel, Kauffman, Michael, Shacham, Sharon, Schwartz, Gary K, Abdul Razak, Albiruni Ryan
Published in Journal of clinical oncology (10.09.2016)
Published in Journal of clinical oncology (10.09.2016)
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Selinexor‐based regimens for the treatment of myeloma refractory to chimeric antigen receptor T cell therapy
Chari, Ajai, Vogl, Dan T., Jagannath, Sundar, Jasielec, Jagoda, Unger, Thaddeus J., DeCastro, Andrew, Shah, Jatin, Kauffman, Michael, Shacham, Sharon, Jakubowiak, Andrzej
Published in British journal of haematology (01.05.2020)
Published in British journal of haematology (01.05.2020)
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Journal Article
Selinexor synergizes with dexamethasone to repress mTORC1 signaling and induce multiple myeloma cell death
Argueta, Christian, Kashyap, Trinayan, Klebanov, Boris, Unger, Thaddeus J, Guo, Cathy, Harrington, Susie, Baloglu, Erkan, Lee, Margaret, Senapedis, William, Shacham, Sharon, Landesman, Yosef
Published in Oncotarget (22.05.2018)
Published in Oncotarget (22.05.2018)
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Journal Article
A 2:1 randomized, open-label, phase II study of selinexor vs. physician's choice in older patients with relapsed or refractory acute myeloid leukemia
Sweet, Kendra, Bhatnagar, Bhavana, Döhner, Hartmut, Donnellan, Will, Frankfurt, Olga, Heuser, Michael, Kota, Vamsi, Liu, Hongtao, Raffoux, Emmanuel, Roboz, Gail J., Röllig, Christoph, Showel, Margaret M., Strickland, Stephen A., Vives, Susana, Tang, Shijie, Unger, Thaddeus J., Joshi, Anita, Shen, Yao, Alvarez, Mariano J., Califano, Andrea, Crochiere, Marsha, Landesman, Yosef, Kauffman, Michael, Shah, Jatin, Shacham, Sharon, Savona, Michael R., Montesinos, Pau
Published in Leukemia & lymphoma (10.11.2021)
Published in Leukemia & lymphoma (10.11.2021)
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Antiobesity Effect of a Small Molecule Repressor of RORγ
Chang, Mi Ra, He, Yuanjun, Khan, Tanya M, Kuruvilla, Dana S, Garcia-Ordonez, Ruben, Corzo, Cesar A, Unger, Thaddeus J, White, David W, Khan, Susan, Lin, Li, Cameron, Michael D, Kamenecka, Theodore M, Griffin, Patrick R
Published in Molecular pharmacology (01.07.2015)
Published in Molecular pharmacology (01.07.2015)
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Journal Article
Abstract 1998: Selinexor effectively inhibits tumor growth in a triple negative breast cancer brain metastasis mouse model
Chang, Hua, Crochiere, Marsha, Debler, Sophie, Kashyap, Trinayan, Unger, Thaddeus J., Baloglu, Erkan, Senapedis, William, Shacham, Sharon, Landesman, Yosef
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Abstract 3086: SINE compounds demonstrated potent anti-cancer activity in PDX mouse models of chordoma
Chang, Hua, Henegar, Leah, Kashyap, Trinayan, Unger, Thaddeus J., Shacham, Sharon, Sommer, Josh, Cogswell, Patty, Fechner, Stacy, Wick, Michael J., Levy, Joan, Landesman, Yosef
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Bioinformatic analysis of selinexor-induced gene expression in patient-derived-chordomas to reveal mechanisms of action leading to tumor growth inhibition
Walker, Christopher James, Chang, Hua, Henegar, Leah, Kashyap, Trinayan, Unger, Thaddeus J, Shacham, Sharon, Cogswell, Patricia, Fechner, Stacy, Wick, Michael, Levy, Joan, Landesman, Yosef
Published in Journal of clinical oncology (20.05.2020)
Published in Journal of clinical oncology (20.05.2020)
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Journal Article
Abstract 5826: Enhanced anti-tumor effects of selinexor and niraparib in preclinical models of ovarian cancer
Chang, Hua, Kashyap, Trinayan, Debler, Sophie, Unger, Thaddeus J., Wang, Sarah, Mikule, Keith, Wang, Jing, Mirza, Mansoor R., Shacham, Sharon, Landesman, Yosef
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract PR008: MYTHIC: First-in-human (FIH) biomarker-driven phase I trial of PKMYT1 inhibitor lunresertib (lunre) alone and with ATR inhibitor camonsertib (cam) in solid tumors with CCNE1 amplification or deleterious alterations in FBXW7 or PPP2R1A
Yap, Timothy A, Schram, Alison, Lee, Elizabeth K, Simpkins, Fiona, Weiss, Mia C, LoRusso, Patricia, Højgaard, Martin, Carneiro, Benedito A, Moy, Ryan H, Garrido-Laguna, Ignacio, Koehler, Maria, Unger, Thaddeus J, Bacque, Emeline, Aguado-Fraile, Elia, Sethuraman, Sunantha, Dhake, Snehal, Liu, Yajun, Fretland, Adrian J, Sun, Xizi, Xu, Yi, Hawkey, Nathan, Truong, Jen, Lheureux, Stephanie
Published in Molecular cancer therapeutics (01.12.2023)
Published in Molecular cancer therapeutics (01.12.2023)
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