Synthesis, Structure−Activity Relationships, and in Vivo Evaluations of Substituted Di-tert-butylphenols as a Novel Class of Potent, Selective, and Orally Active Cyclooxygenase-2 Inhibitors. 2. 1,3,4- and 1,2,4-Thiadiazole Series
Song, Yuntao, Connor, David T, Sercel, Anthony D, Sorenson, Roderick J, Doubleday, Robert, Unangst, Paul C, Roth, Bruce D, Beylin, Vlad G, Gilbertsen, Richard B, Chan, Kam, Schrier, Denis J, Guglietta, Antonio, Bornemeier, Dirk A, Dyer, Richard D
Published in Journal of medicinal chemistry (08.04.1999)
Published in Journal of medicinal chemistry (08.04.1999)
Get full text
Journal Article
Synthesis and biological evaluation of 5-[[3,5-bis(1,1-dimethylethyl)-4-hydroxyphenyl]methylene]oxazoles, -thiazoles, and -imidazoles: novel dual 5-lipoxygenase and cyclooxygenase inhibitors with antiinflammatory activity
Unangst, Paul C, Connor, David T, Cetenko, Wiaczeslaw A, Sorenson, Roderick J, Kostlan, Catherine R, Sircar, Jagadish C, Wright, Clifford D, Schrier, Denis J, Dyer, Richard D
Published in Journal of medicinal chemistry (01.01.1994)
Published in Journal of medicinal chemistry (01.01.1994)
Get full text
Journal Article
Novel indolecarboxamidotetrazoles as potential antiallergy agents
Unangst, Paul C, Connor, David T, Stabler, S. Russell, Weikert, Robert J, Carethers, Mary E, Kennedy, John A, Thueson, David O, Chestnut, James C, Adolphson, Richard L, Conroy, M. C
Published in Journal of medicinal chemistry (01.06.1989)
Published in Journal of medicinal chemistry (01.06.1989)
Get full text
Journal Article
Synthesis, Structure−Activity Relationships, and in Vivo Evaluations of Substituted Di-tert-butylphenols as a Novel Class of Potent, Selective, and Orally Active Cyclooxygenase-2 Inhibitors. 1. Thiazolone and Oxazolone Series
Song, Yuntao, Connor, David T, Doubleday, Robert, Sorenson, Roderick J, Sercel, Anthony D, Unangst, Paul C, Roth, Bruce D, Gilbertsen, Richard B, Chan, Kam, Schrier, Denis J, Guglietta, Antonio, Bornemeier, Dirk A, Dyer, Richard D
Published in Journal of medicinal chemistry (08.04.1999)
Published in Journal of medicinal chemistry (08.04.1999)
Get full text
Journal Article
2,6-di-tert-butylphenols: a new class of potent and selective PGHS-2 inhibitor
Song, Y, Connor, D T, Sorenson, R J, Doubleday, R, Sercel, A D, Unangst, P C, Gilbertsen, R B, Chan, K, Bornemeier, D A, Dyer, R D
Published in Inflammation research (01.08.1997)
Published in Inflammation research (01.08.1997)
Get full text
Journal Article
Chromeno[3,4-c]pyridin-5-ones: Selective Human Dopamine D4 Receptor Antagonists as Potential Antipsychotic Agents
Unangst, Paul C, Capiris, Thomas, Connor, David T, Heffner, Thomas G, MacKenzie, Robert G, Miller, Steven R, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (15.08.1997)
Published in Journal of medicinal chemistry (15.08.1997)
Get full text
Journal Article
3-(Aminoalkyl)-1,2,3,4-tetrahydro-5H-[1]benzopyrano[3,4-c]pyridin-5-ones as potential anticholinergic bronchodilators
Connor, David T, Unangst, Paul C, Schwender, Charles F, Sorenson, Roderick J, Carethers, Mary E, Puchalski, Chester, Brown, Richard E, Finkel, Martin P
Published in Journal of medicinal chemistry (01.03.1989)
Published in Journal of medicinal chemistry (01.03.1989)
Get full text
Journal Article
(Aryloxy)alkylamines as Selective Human Dopamine D4 Receptor Antagonists: Potential Antipsychotic Agents
Unangst, Paul C, Capiris, Thomas, Connor, David T, Doubleday, Robert, Heffner, Thomas G, MacKenzie, Robert G, Miller, Steven R, Pugsley, Thomas A, Wise, Lawrence D
Published in Journal of medicinal chemistry (05.12.1997)
Published in Journal of medicinal chemistry (05.12.1997)
Get full text
Journal Article
Synthesis of novel 3-and 5-substituted indole-2-carboxamides
Bratton, LD, Roth, BD, Trivedi, BK, Unangst, PC
Published in Journal of heterocyclic chemistry (01.09.2000)
Published in Journal of heterocyclic chemistry (01.09.2000)
Get more information
Journal Article
Addition reactions of allyl stannanes to an indolo[2 ',3 ': 3,4]pyrido[1,2-b]isoquinoline imminium salt
Unangst, PC, Bratton, LD, Connor, DT, Roth, BD, Rubin, Trivedi, BK
Published in Journal of heterocyclic chemistry (01.09.2000)
Published in Journal of heterocyclic chemistry (01.09.2000)
Get more information
Journal Article
Acidic furo[3,2-b]indoles. A new series of potent antiallergy agents
Unangst, P C, Carethers, M E, Webster, K, Janik, G M, Robichaud, L J
Published in Journal of medicinal chemistry (01.12.1984)
Published in Journal of medicinal chemistry (01.12.1984)
Get full text
Journal Article
Synthesis and antiallergy activity of 4-oxopyrano[3,2-b]indoles
Unangst, Paul C, Brown, Richard E, Herzig, David J
Published in Journal of medicinal chemistry (01.11.1980)
Published in Journal of medicinal chemistry (01.11.1980)
Get full text
Journal Article
Novel benzothiophene-, benzofuran-, and naphthalenecarboxamidotetrazoles as potential antiallergy agents
Connor, David T, Cetenko, Wiaczeslaw A, Mullican, Michael D, Sorenson, Roderick J, Unangst, Paul C, Weikert, Robert J, Adolphson, Richard L, Kennedy, John A, Thueson, David O
Published in Journal of medicinal chemistry (01.03.1992)
Published in Journal of medicinal chemistry (01.03.1992)
Get full text
Journal Article
Synthesis, structure-activity relationships, and in vivo evaluations of substituted di-tert-butylphenols as a novel class of potent, selective, and orally active cyclooxygenase-2 inhibitors. 1. Thiazolone and oxazolone series1
YUNTAO SONG, CONNOR, D. T, GUGLIETTA, A, BORNEMEIER, D. A, DYER, R. D, DOUBLEDAY, R, SORENSON, R. J, SERCEL, A. D, UNANGST, P. C, ROTH, B. D, GILBERTSEN, R. B, KAM CHAN, SCHRIER, D. J
Published in Journal of medicinal chemistry (1999)
Get full text
Published in Journal of medicinal chemistry (1999)
Journal Article
Preparation of 6-, 7-, and 9-substituted derivatives of 2-oxa-1,3,4,10-tetraazacyclopenta[b]fluoren-9-one
Bratton, LD, Unangst, PC, Rubin, Trivedi, BK
Published in Journal of heterocyclic chemistry (01.09.2001)
Published in Journal of heterocyclic chemistry (01.09.2001)
Get more information
Journal Article
Oxazole, thiazole, and imidazole derivatives of 2,6-di-tert-butylphenol as udal 5-lipoxygenase and cyclooxygenase inhibitors
UNANGST, P. C, CONNOR, D. T, CETENKO, W. A, SORENSON, R. J, SIRCAR, J. C, WRIGHT, C. D, SCHRIER, D. J, DYER, R. D
Published in Bioorganic & medicinal chemistry letters (1993)
Get full text
Published in Bioorganic & medicinal chemistry letters (1993)
Journal Article