Desymmetrization of meso-Glycerol Derivatives Induced by L-Histidine-Derived Acylation Catalysts
Sakakura, Akira, Umemura, Shuhei, Ishihara, Kazuaki
Published in Advanced synthesis & catalysis (01.08.2011)
Published in Advanced synthesis & catalysis (01.08.2011)
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Journal Article
Dehydrative cyclization of serine, threonine, and cysteine residues catalyzed by molybdenum(VI) oxo compounds
Sakakura, Akira, Kondo, Rei, Umemura, Shuhei, Ishihara, Kazuaki
Published in Tetrahedron (07.03.2009)
Published in Tetrahedron (07.03.2009)
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Journal Article
GCL INHIBITOR
UMEMURA, Shuhei, INUKAI, Takayuki, KASANO, Miki, OKADA, Takuya, KAWAMATA, Takahiro
Year of Publication 19.05.2023
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Year of Publication 19.05.2023
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PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH KDM5 INHIBITORY EFFECT
ANATOLY LUBINSKI, TAKAHASHI SHUSUKE, KAKUUCHI AKITO, IYAMA DAIGO, GORAN KURILOFF, MATZ SVENSSON, ASADA MASAKI, KYLE CONZE, UMEMURA SHUHEI, YAN CHAN
Year of Publication 18.05.2023
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Year of Publication 18.05.2023
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KDM5 억제 활성을 갖는 화합물 및 이의 약학적 용도
KRILOV GORAN, INOYAMA DAIGO, KAKUUCHI AKITO, ZHANG YAN, RUVINSKY ANATOLY, SVENSSON MATS, KONZE KYLE, TAKAHASHI HIDENORI, ASADA MASAKI, UMEMURA SHUHEI
Year of Publication 12.01.2023
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Year of Publication 12.01.2023
Patent
Preparation of Stereodefined Homoallylic Amines from the Reductive Cross-Coupling of Allylic Alcohols with Imines
Chen, Ming Z, McLaughlin, Martin, Takahashi, Masayuki, Tarselli, Michael A, Yang, Dexi, Umemura, Shuhei, Micalizio, Glenn C
Published in Journal of organic chemistry (03.12.2010)
Published in Journal of organic chemistry (03.12.2010)
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Journal Article
Dehydrative Cyclization Catalyzed by the Combination of Molybdenum(VI) Oxides and Benzoic Acids: First Synthesis of the Antitumour Substance BE-70016
Sakakura, Akira, Umemura, Shuhei, Kondo, Rei, Ishihara, Kazuaki
Published in Advanced synthesis & catalysis (05.03.2007)
Published in Advanced synthesis & catalysis (05.03.2007)
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Journal Article
COMPOUND HAVING KDM5 INHIBITORY ACTIVITY AND PHARMACEUTICAL USE THEREOF
UMEMURA, Shuhei, KRILOV, Goran, KAKUUCHI, Akito, RUVINSKY, Anatoly, ASADA, Masaki, ZHANG, Yan, TAKAHASHI, Hidenori, SVENSSON, Mats, INOYAMA, Daigo, KONZE, Kyle
Year of Publication 31.08.2023
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Year of Publication 31.08.2023
Patent
Compound having KDM5 inhibitory activity and pharmaceutical use thereof
Takahashi, Hidenori, Kakuuchi, Akito, Asada, Masaki, Krilov, Goran, Konze, Kyle, Ruvinsky, Anatoly, Umemura, Shuhei, Svensson, Mats, Zhang, Yan, Inoyama, Daigo
Year of Publication 04.07.2023
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Year of Publication 04.07.2023
Patent
COMPOUND HAVING KDM5 INHIBITORY ACTIVITY AND PHARMACEUTICAL USE THEREOF
UMEMURA, Shuhei, KRILOV, Goran, KAKUUCHI, Akito, RUVINSKY, Anatoly, ASADA, Masaki, ZHANG, Yan, TAKAHASHI, Hidenori, SVENSSON, Mats, INOYAMA, Daigo, KONZE, Kyle
Year of Publication 06.04.2023
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Year of Publication 06.04.2023
Patent