Search Results - "Umedera, Kohei" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Design of MMP-1 inhibitors via SAR transfer and experimental validation

Design of MMP-1 inhibitors via SAR transfer and experimental validation

by Umedera, Kohei, Yoshimori, Atsushi, Bajorath, Jürgen, Nakamura, Hiroyuki
Published in Scientific reports (03.12.2022)

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Journal Article

Asymmetric construction of densely functionalized three-dimensional aza-tetracyclic scaffolds for drug discovery

Asymmetric construction of densely functionalized three-dimensional aza-tetracyclic scaffolds for drug discovery

by Umedera, Kohei, Morita, Taiki, Nakamura, Hiroyuki
Published in Chemical communications (Cambridge, England) (08.12.2022)

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Journal Article

DeepCubist: Molecular Generator for Designing Peptidomimetics based on Complex three-dimensional scaffolds

DeepCubist: Molecular Generator for Designing Peptidomimetics based on Complex three-dimensional scaffolds

by Umedera, Kohei, Yoshimori, Atsushi, Chen, Hengwei, Kouji, Hiroyuki, Nakamura, Hiroyuki, Bajorath, Jürgen
Published in Journal of computer-aided molecular design (01.02.2023)

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Journal Article

Synthesis of Three‐Dimensional (Di)Azatricyclododecene Scaffold and Its Application to Peptidomimetics

Synthesis of Three‐Dimensional (Di)Azatricyclododecene Scaffold and Its Application to Peptidomimetics

by Umedera, Kohei, Morita, Taiki, Yoshimori, Atsushi, Yamada, Kentaro, Katoh, Akira, Kouji, Hiroyuki, Nakamura, Hiroyuki
Published in Chemistry : a European journal (16.08.2021)

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Journal Article

Discovery of sp3-rich diazatricycloundecanes as lysosomotropic autophagy inhibitors

Discovery of sp3-rich diazatricycloundecanes as lysosomotropic autophagy inhibitors

by Miura, Kazuki, Doi, Tomoya, Umedera, Kohei, Nakamura, Hiroyuki
Published in European journal of medicinal chemistry (15.12.2024)

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Journal Article

Synthesis of the diazatricycloundecane scaffold gold()-catalysed Conia-ene-type 5- cyclization and stepwise substituent assembly for the construction of an sp-rich compound library

Synthesis of the diazatricycloundecane scaffold gold()-catalysed Conia-ene-type 5- cyclization and stepwise substituent assembly for the construction of an sp-rich compound library

by Doi, Tomoya, Umedera, Kohei, Miura, Kazuki, Morita, Taiki, Nakamura, Hiroyuki
Published in Organic & biomolecular chemistry (08.11.2023)

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Journal Article

Synthesis of the diazatricycloundecane scaffold via gold( i )-catalysed Conia-ene-type 5- exo-dig cyclization and stepwise substituent assembly for the construction of an sp 3 -rich compound library

Synthesis of the diazatricycloundecane scaffold via gold( i )-catalysed Conia-ene-type 5- exo-dig cyclization and stepwise substituent assembly for the construction of an sp 3 -rich compound library

by Doi, Tomoya, Umedera, Kohei, Miura, Kazuki, Morita, Taiki, Nakamura, Hiroyuki
Published in Organic & biomolecular chemistry (08.11.2023)

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Journal Article

Synthesis of the diazatricycloundecane scaffold via gold(i)-catalysed Conia-ene-type 5-exo-dig cyclization and stepwise substituent assembly for the construction of an sp3-rich compound library

Synthesis of the diazatricycloundecane scaffold via gold(i)-catalysed Conia-ene-type 5-exo-dig cyclization and stepwise substituent assembly for the construction of an sp3-rich compound library

by Doi, Tomoya, Umedera, Kohei, Miura, Kazuki, Morita, Taiki, Nakamura, Hiroyuki
Published in Organic & biomolecular chemistry (08.11.2023)

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Journal Article

Discovery of sp 3 -rich diazatricycloundecanes as lysosomotropic autophagy inhibitors

Discovery of sp 3 -rich diazatricycloundecanes as lysosomotropic autophagy inhibitors

by Miura, Kazuki, Doi, Tomoya, Umedera, Kohei, Nakamura, Hiroyuki
Published in European journal of medicinal chemistry (05.10.2024)

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Journal Article

NOVEL NITROGEN-CONTAINING TRICYCLIC SKELETON COMPOUND AND USE THEREOF

NOVEL NITROGEN-CONTAINING TRICYCLIC SKELETON COMPOUND AND USE THEREOF

by UMEDERA KOHEI, MORITA DAIKI, NAKAMURA HIROYUKI, YOSHIMORI ATSUSHI, SHOJI HIROYUKI
Year of Publication 21.06.2022

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