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Published in Nature communications (15.01.2024)
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Published in mBio (30.09.2014)
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Published in mBio (2012)
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Published in Synlett (01.01.2010)
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Published in Bioorganic & medicinal chemistry (01.12.2007)
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Late-stage oxidative C(sp 3 )-H methylation
Feng, Kaibo, Quevedo, Raundi E, Kohrt, Jeffrey T, Oderinde, Martins S, Reilly, Usa, White, M Christina
Published in Nature (London) (30.04.2020)
Published in Nature (London) (30.04.2020)
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Published in Organic & biomolecular chemistry (04.10.2017)
Published in Organic & biomolecular chemistry (04.10.2017)
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Late-Stage Lead Diversification Coupled with Quantitative Nuclear Magnetic Resonance Spectroscopy to Identify New Structure-Activity Relationship Vectors at Nanomole-Scale Synthesis: Application to Loratadine, a Human Histamine H-1 Receptor Inverse Agonist
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Published in Journal of medicinal chemistry (09.07.2020)
Published in Journal of medicinal chemistry (09.07.2020)
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Incorporation of [2H1]-(1R,2R)- and [2H1]-(1S,2R)-glycerols into the antibiotic nucleocidin in Streptomyces calvusElectronic supplementary information (ESI) available. See DOI: 10.1039/c7ob02163a
Feng, Xuan, Al Maharik, Nawaf, Bartholomé, Axel, Janso, Jeffrey E, Reilly, Usa, O'Hagan, David
Year of Publication 04.10.2017
Year of Publication 04.10.2017
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Journal Article
Late-Stage Lead Diversification Coupled with Quantitative Nuclear Magnetic Resonance Spectroscopy to Identify New Structure–Activity Relationship Vectors at Nanomole-Scale Synthesis: Application to Loratadine, a Human Histamine H1 Receptor Inverse Agonist
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Published in Journal of medicinal chemistry (09.07.2020)
Published in Journal of medicinal chemistry (09.07.2020)
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Novel 3-fluoro-6-methoxyquinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV
Mitton-Fry, Mark J., Brickner, Steven J., Hamel, Judith C., Barham, Rose, Brennan, Lori, Casavant, Jeffrey M., Ding, Xiaoyuan, Finegan, Steven, Hardink, Joel, Hoang, Thuy, Huband, Michael D., Maloney, Meghan, Marfat, Anthony, McCurdy, Sandra P., McLeod, Dale, Subramanyam, Chakrapani, Plotkin, Michael, Reilly, Usa, Schafer, John, Stone, Gregory G., Uccello, Daniel P., Wisialowski, Todd, Yoon, Kwansik, Zaniewski, Richard, Zook, Christopher
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
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Pyridone Methylsulfone Hydroxamate LpxC Inhibitors for the Treatment of Serious Gram-Negative Infections
Montgomery, Justin I, Brown, Matthew F, Reilly, Usa, Price, Loren M, Abramite, Joseph A, Arcari, Joel, Barham, Rose, Che, Ye, Chen, Jinshan Michael, Chung, Seung Won, Collantes, Elizabeth M, Desbonnet, Charlene, Doroski, Matthew, Doty, Jonathan, Engtrakul, Juntyma J, Harris, Thomas M, Huband, Michael, Knafels, John D, Leach, Karen L, Liu, Shenping, Marfat, Anthony, McAllister, Laura, McElroy, Eric, Menard, Carol A, Mitton-Fry, Mark, Mullins, Lisa, Noe, Mark C, O’Donnell, John, Oliver, Robert, Penzien, Joseph, Plummer, Mark, Shanmugasundaram, Veerabahu, Thoma, Christy, Tomaras, Andrew P, Uccello, Daniel P, Vaz, Alfin, Wishka, Donn G
Published in Journal of medicinal chemistry (23.02.2012)
Published in Journal of medicinal chemistry (23.02.2012)
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Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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Novel quinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV
Mitton-Fry, Mark J., Brickner, Steven J., Hamel, Judith C., Brennan, Lori, Casavant, Jeffrey M., Chen, Michael, Chen, Tao, Ding, Xiaoyuan, Driscoll, James, Hardink, Joel, Hoang, Thuy, Hua, Erbing, Huband, Michael D., Maloney, Meghan, Marfat, Anthony, McCurdy, Sandra P., McLeod, Dale, Plotkin, Michael, Reilly, Usa, Robinson, Shaughn, Schafer, John, Shepard, Richard M., Smith, James F., Stone, Gregory G., Subramanyam, Chakrapani, Yoon, Kwansik, Yuan, Wei, Zaniewski, Richard P., Zook, Christopher
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Published in Bioorganic & medicinal chemistry letters (15.05.2013)
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Farley, Kathleen A., Reilly, Usa, Anderson, Dennis P., Boscoe, Brian P., Bundesmann, Mark W., Foley, David A., Lall, Manjinder S., Li, Chao, Reese, Matthew R., Yan, Jiangli
Published in Magnetic resonance in chemistry (01.04.2017)
Published in Magnetic resonance in chemistry (01.04.2017)
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Published in Bioorganic & medicinal chemistry letters (15.11.2012)
Published in Bioorganic & medicinal chemistry letters (15.11.2012)
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Late Stage Lead Diversification (LSLD) Coupled with Quantitative NMR Spectroscopy to Identify New SAR Vectors at Nanomole Scale Synthesis: Application to Loratadine a Human Histamine H 1 Receptor Inverse Agonist
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Published in Journal of medicinal chemistry (28.05.2020)
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Published in Journal of medicinal chemistry (28.05.2020)
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Discovery of Azetidinyl Ketolides for the Treatment of Susceptible and Multidrug Resistant Community-Acquired Respiratory Tract Infections
Magee, Thomas V, Ripp, Sharon L, Li, Bryan, Buzon, Richard A, Chupak, Lou, Dougherty, Thomas J, Finegan, Steven M, Girard, Dennis, Hagen, Anne E, Falcone, Michael J, Farley, Kathleen A, Granskog, Karl, Hardink, Joel R, Huband, Michael D, Kamicker, Barbara J, Kaneko, Takushi, Knickerbocker, Michael J, Liras, Jennifer L, Marra, Andrea, Medina, Ivy, Nguyen, Thuy-Trinh, Noe, Mark C, Obach, R. Scott, O’Donnell, John P, Penzien, Joseph B, Reilly, Usa Datta, Schafer, John R, Shen, Yue, Stone, Gregory G, Strelevitz, Timothy J, Sun, Jianmin, Tait-Kamradt, Amelia, Vaz, Alfin D. N, Whipple, David A, Widlicka, Daniel W, Wishka, Donn G, Wolkowski, Joanna P, Flanagan, Mark E
Published in Journal of medicinal chemistry (10.12.2009)
Published in Journal of medicinal chemistry (10.12.2009)
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