Emerging peptide antibiotics with therapeutic potential
Upert, Gregory, Luther, Anatol, Obrecht, Daniel, Ermert, Philipp
Published in Medicine in drug discovery (01.03.2021)
Published in Medicine in drug discovery (01.03.2021)
Get full text
Journal Article
Antibiotic polymyxin arranges lipopolysaccharide into crystalline structures to solidify the bacterial membrane
Manioglu, Selen, Modaresi, Seyed Majed, Ritzmann, Noah, Thoma, Johannes, Overall, Sarah A, Harms, Alexander, Upert, Gregory, Luther, Anatol, Barnes, Alexander B, Obrecht, Daniel, Müller, Daniel J, Hiller, Sebastian
Published in Nature communications (21.10.2022)
Published in Nature communications (21.10.2022)
Get full text
Journal Article
Reply to: Antibiotics and hexagonal order in the bacterial outer membrane
Manioglu, Selen, Modaresi, Seyed Majed, Thoma, Johannes, Overall, Sarah A, Upert, Gregory, Luther, Anatol, Barnes, Alexander B, Obrecht, Daniel, Müller, Daniel J, Hiller, Sebastian
Published in Nature communications (09.08.2023)
Published in Nature communications (09.08.2023)
Get full text
Journal Article
Disulfide Connectivity Analysis of Peptides Bearing Two Intramolecular Disulfide Bonds Using MALDI In-Source Decay
Massonnet, Philippe, Haler, Jean R. N., Upert, Gregory, Smargiasso, Nicolas, Mourier, Gilles, Gilles, Nicolas, Quinton, Loïc, De Pauw, Edwin
Published in Journal of the American Society for Mass Spectrometry (01.10.2018)
Published in Journal of the American Society for Mass Spectrometry (01.10.2018)
Get full text
Journal Article
Web Resource
Ancestral protein resurrection and engineering opportunities of the mamba aminergic toxins
Blanchet, Guillaume, Alili, Doria, Protte, Adèle, Upert, Gregory, Gilles, Nicolas, Tepshi, Livia, Stura, Enrico A, Mourier, Gilles, Servent, Denis
Published in Scientific reports (02.06.2017)
Published in Scientific reports (02.06.2017)
Get full text
Journal Article
Enamine Catalysis with Low Catalyst Loadings - High Efficiency via Kinetic Studies
Wiesner, Markus, Upert, Grégory, Angelici, Gaetano, Wennemers, Helma
Published in Journal of the American Chemical Society (13.01.2010)
Published in Journal of the American Chemical Society (13.01.2010)
Get full text
Journal Article
Chimeric peptidomimetic antibiotics against Gram-negative bacteria
Luther, Anatol, Urfer, Matthias, Zahn, Michael, Müller, Maik, Wang, Shuang-Yan, Mondal, Milon, Vitale, Alessandra, Hartmann, Jean-Baptiste, Sharpe, Timothy, Monte, Fabio Lo, Kocherla, Harsha, Cline, Elizabeth, Pessi, Gabriella, Rath, Parthasarathi, Modaresi, Seyed Majed, Chiquet, Petra, Stiegeler, Sarah, Verbree, Carolin, Remus, Tobias, Schmitt, Michel, Kolopp, Caroline, Westwood, Marie-Anne, Desjonquères, Nicolas, Brabet, Emile, Hell, Sophie, LePoupon, Karen, Vermeulen, Annie, Jaisson, Régis, Rithié, Virginie, Upert, Grégory, Lederer, Alexander, Zbinden, Peter, Wach, Achim, Moehle, Kerstin, Zerbe, Katja, Locher, Hans H, Bernardini, Francesca, Dale, Glenn E, Eberl, Leo, Wollscheid, Bernd, Hiller, Sebastian, Robinson, John A, Obrecht, Daniel
Published in Nature (London) (01.12.2019)
Published in Nature (London) (01.12.2019)
Get full text
Journal Article
From a Cone Snail Toxin to a Competitive MC4R Antagonist
Reynaud, Steve, Laurin, Suli-Anne, Ciolek, Justyna, Barbe, Peggy, Van Baelen, Anne-Cécile, Susset, Michaël, Blondel, Florian, Ghazarian, Marine, Boeri, Julia, Vanden Driessche, Margot, Upert, Grégory, Mourier, Gilles, Kessler, Pascal, Konnert, Laure, Beroud, Rémy, Keck, Mathilde, Servent, Denis, Bouvier, Michel, Gilles, Nicolas
Published in Journal of medicinal chemistry (22.09.2022)
Published in Journal of medicinal chemistry (22.09.2022)
Get full text
Journal Article
A Venomics Approach Coupled to High-Throughput Toxin Production Strategies Identifies the First Venom-Derived Melanocortin Receptor Agonists
Reynaud, Steve, Ciolek, Justyna, Degueldre, Michel, Saez, Natalie J, Sequeira, Ana Filipa, Duhoo, Yoan, Brás, Joana L. A, Meudal, Hervé, Cabo Díez, Miguel, Fernández Pedrosa, Victoria, Verdenaud, Marion, Boeri, Julia, Pereira Ramos, Oscar, Ducancel, Frédéric, Vanden Driessche, Margot, Fourmy, Rudy, Violette, Aude, Upert, Grégory, Mourier, Gilles, Beck-Sickinger, Annette G, Mörl, Karin, Landon, Céline, Fontes, Carlos M. G. A, Miñambres Herráiz, Rebeca, Rodríguez de la Vega, Ricardo C, Peigneur, Steve, Tytgat, Jan, Quinton, Loïc, De Pauw, Edwin, Vincentelli, Renaud, Servent, Denis, Gilles, Nicolas
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
Get full text
Journal Article
Web Resource
RgIA4 potently blocks mouse $\alpha$9$\alpha$10 nAChRs and provides long lasting protection against oxaliplatin-induced cold allodynia
Christensen, Sean, Hone, Arik, Roux, Isabelle, Kniazeff, Julie, Pin, Jean-Philippe, Upert, Grégory, Servent, Denis, Glowatzki, Elisabeth, Mcintosh, J Michael, Mcintosh, J. Michael
Published in Frontiers in cellular neuroscience (21.07.2017)
Published in Frontiers in cellular neuroscience (21.07.2017)
Get full text
Journal Article
RgIA4 Potently Blocks Mouse α9α10 nAChRs and Provides Long Lasting Protection against Oxaliplatin-Induced Cold Allodynia
Christensen, Sean B, Hone, Arik J, Roux, Isabelle, Kniazeff, Julie, Pin, Jean-Philippe, Upert, Grégory, Servent, Denis, Glowatzki, Elisabeth, McIntosh, J Michael
Published in Frontiers in cellular neuroscience (21.07.2017)
Published in Frontiers in cellular neuroscience (21.07.2017)
Get full text
Journal Article
Acidosis increases MHC class II-restricted presentation of a protein endowed with a pH-dependent heparan sulfate-binding ability
Knittel, Delphine, Savatier, Alexandra, Upert, Grégory, Lortat-Jacob, Hugues, Léonetti, Michel
Published in The Journal of immunology (1950) (15.04.2015)
Published in The Journal of immunology (1950) (15.04.2015)
Get full text
Journal Article
High-throughput production of two disulphide-bridge toxins
Upert, Grégory, Mourier, Gilles, Pastor, Alexandra, Verdenaud, Marion, Alili, Doria, Servent, Denis, Gilles, Nicolas
Published in Chemical communications (Cambridge, England) (07.08.2014)
Published in Chemical communications (Cambridge, England) (07.08.2014)
Get full text
Journal Article
Silver Nanoparticle Formation in Different Sizes Induced by Peptides Identified within Split-and-Mix Libraries
Belser, Kirsten, Vig Slenters, Tünde, Pfumbidzai, Conelious, Upert, Grégory, Mirolo, Laurent, Fromm, Katharina M, Wennemers, Helma
Published in Angewandte Chemie (International ed.) (01.01.2009)
Published in Angewandte Chemie (International ed.) (01.01.2009)
Get full text
Journal Article
Peptidomimetic antibiotics disrupt the lipopolysaccharide transport bridge of drug-resistant Enterobacteriaceae
Schuster, Matthias, Brabet, Emile, Oi, Kathryn K, Desjonquères, Nicolas, Moehle, Kerstin, Le Poupon, Karen, Hell, Sophie, Gable, Stéphane, Rithié, Virginie, Dillinger, Séverine, Zbinden, Peter, Luther, Anatol, Li, Claudia, Stiegeler, Sarah, D'Arco, Carolin, Locher, Hans, Remus, Tobias, DiMaio, Selena, Motta, Paola, Wach, Achim, Jung, Françoise, Upert, Grégory, Obrecht, Daniel, Benghezal, Mohammed, Zerbe, Oliver
Published in Science advances (26.05.2023)
Published in Science advances (26.05.2023)
Get full text
Journal Article
Zinc-selective inhibition of the promiscuous bacterial amide-hydrolase DapE: implications of metal heterogeneity for evolution and antibiotic drug design
Uda, Narasimha Rao, Upert, Grégory, Angelici, Gaetano, Nicolet, Stefan, Schmidt, Tobias, Schwede, Torsten, Creus, Marc
Published in Metallomics (01.01.2014)
Published in Metallomics (01.01.2014)
Get more information
Journal Article
Combined Use of Ion Mobility and Collision-Induced Dissociation To Investigate the Opening of Disulfide Bridges by Electron-Transfer Dissociation in Peptides Bearing Two Disulfide Bonds
Massonnet, Philippe, Upert, Gregory, Smargiasso, Nicolas, Gilles, Nicolas, Quinton, Loïc, De Pauw, Edwin
Published in Analytical chemistry (Washington) (19.05.2015)
Published in Analytical chemistry (Washington) (19.05.2015)
Get full text
Journal Article
Web Resource