Design, synthesis and biological evaluation of novel triazole, urea and thiourea derivatives of quinoline against Mycobacterium tuberculosis
Upadhayaya, Ram Shankar, Kulkarni, Girish M., Vasireddy, Nageswara Rao, Vandavasi, Jaya Kishore, Dixit, Shailesh S., Sharma, Vivek, Chattopadhyaya, Jyoti
Published in Bioorganic & medicinal chemistry (01.07.2009)
Published in Bioorganic & medicinal chemistry (01.07.2009)
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Journal Article
Design, synthesis, biological evaluation and molecular modelling studies of novel quinoline derivatives against Mycobacterium tuberculosis
Upadhayaya, Ram Shankar, Vandavasi, Jaya Kishore, Vasireddy, Nageswara Rao, Sharma, Vivek, Dixit, Shailesh S., Chattopadhyaya, Jyoti
Published in Bioorganic & medicinal chemistry (01.04.2009)
Published in Bioorganic & medicinal chemistry (01.04.2009)
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Journal Article
Novel quinoline and naphthalene derivatives as potent antimycobacterial agents
Upadhayaya, Ram Shankar, Vandavasi, Jaya Kishore, Kardile, Ramakant A., Lahore, Santosh V., Dixit, Shailesh S., Deokar, Hemantkumar S., Shinde, Popat D., Sarmah, Manash P., Chattopadhyaya, Jyoti
Published in European journal of medicinal chemistry (01.05.2010)
Published in European journal of medicinal chemistry (01.05.2010)
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Journal Article
Optically active antifungal azoles: synthesis and antifungal activity of (2 R,3 S)-2-(2,4-difluorophenyl)-3-(5-{2-[4-aryl-piperazin-1-yl]-ethyl}-tetrazol-2-yl/1-yl)-1-[1,2,4]-triazol-1-yl-butan-2-ol
Upadhayaya, Ram Shankar, Sinha, Neelima, Jain, Sanjay, Kishore, Nawal, Chandra, Ramesh, Arora, Sudershan K.
Published in Bioorganic & medicinal chemistry (01.05.2004)
Published in Bioorganic & medicinal chemistry (01.05.2004)
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Journal Article
Synthesis of novel substituted tetrazoles having antifungal activity
Upadhayaya, Ram Shankar, Jain, Sanjay, Sinha, Neelima, Kishore, Nawal, Chandra, Ramesh, Arora, Sudershan K
Published in European journal of medicinal chemistry (01.07.2004)
Published in European journal of medicinal chemistry (01.07.2004)
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Journal Article
Conformationally-constrained indeno[2,1-c]quinolines - a new class of anti-mycobacterial agents
Upadhayaya, Ram Shankar, Lahore, Santosh V., Sayyed, Aftab Y., Dixit, Shailesh S., Shinde, Popat D., Chattopadhyaya, Jyoti
Published in Organic & biomolecular chemistry (01.01.2010)
Published in Organic & biomolecular chemistry (01.01.2010)
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Journal Article
Synthesis and antimycobacterial activity of prodrugs of indeno[2,1- c]quinoline derivatives
Upadhayaya, Ram Shankar, Shinde, Popat D., Kadam, Sandip A., Bawane, Amit N., Sayyed, Aftab Y., Kardile, Ramakant A., Gitay, Pallavi N., Lahore, Santosh V., Dixit, Shailesh S., Földesi, András, Chattopadhyaya, Jyoti
Published in European journal of medicinal chemistry (01.04.2011)
Published in European journal of medicinal chemistry (01.04.2011)
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Journal Article
항-감염 복소환식 화합물 및 이의 용도
UPADHAYAYA RAM SHANKAR, KIRSEBOM LEIF, VIRTANEN ANDERS, KETHIRI RAGHAVA REDDY
Year of Publication 25.08.2020
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Year of Publication 25.08.2020
Patent
Synthesis of isonicotinic acid N′-arylidene- N-[2-oxo-2-(4-aryl-piperazin-1-yl)-ethyl]-hydrazides as antituberculosis agents
Sinha, Neelima, Jain, Sanjay, Tilekar, Ajay, Upadhayaya, Ram Shankar, Kishore, Nawal, Jana, Gour Hari, Arora, Sudershan K.
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
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Journal Article
항-감염 헤테로사이클릭 화합물 및 이의 용도
UPADHAYAYA RAM SHANKAR, KIRSEBOM LEIF, VIRTANEN ANDERS, KETHIRI RAGHAVA REDDY
Year of Publication 12.03.2019
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Year of Publication 12.03.2019
Patent
BRD4 및 JAK2 이중 억제제로서의 융합된 피리미딘 및 이의 사용 방법
UPADHAYAYA RAM SHANKAR, MADAN SACHIN, RAJAIAH SANTOSH KUMAR KOTTURI, KETHIRI RAGHAVA
Year of Publication 06.12.2019
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Year of Publication 06.12.2019
Patent
Synthesis and anti-cancer activity of disubstituted- and deoxytrisubstituted-α-D-allofuranoses
Kishore, Nawal, Jain, Sanjay, Sinha, Neelima, Upadhayaya, Ram Shankar, Chandra, Ramesh, Arora, Sudershan K.
Published in ARKIVOC (01.01.2005)
Published in ARKIVOC (01.01.2005)
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Web Resource
New antiprotozoal agents: Their synthesis and biological evaluations
Upadhayaya, Ram Shankar, Dixit, Shailesh S., Földesi, Andras, Chattopadhyaya, Jyoti
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
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Journal Article
JAK-STAT inhibitor as a potential therapeutic opportunity in AML patients resistant to cytarabine and epigenetic therapy
Babu, Govind, Chaudhuri, Padmaparna, Rajappa, Manoj, Biswas, Manjusha, Sansar, Bipinesh, Rajegowda, Chethan, Radhakrishnan, Aneesha, Advani, Jayshree, Tewary, Biplab, Radhakrishnan, Padhma, Thiyagarajan, Saravanan, Chatterjee, Aditi, Upadhayaya, Ram Shankar, Majumder, Pradip K
Published in Cancer biology & therapy (02.01.2021)
Published in Cancer biology & therapy (02.01.2021)
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Journal Article
Synthesis of disubstituted- and deoxydisubstituted- derivatives of α-D-xylofuranose as anticancer agents
Kishore, Nawal, Sinha, Neelima, Jain, Sanjay, Upadhayaya, Ram Shankar, Chandra, Ramesh, Arora, Sudershan K.
Published in ARKIVOC (04.01.2005)
Published in ARKIVOC (04.01.2005)
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Carbocyclic C-C Bond Formation: Intramolecular Radical Ring Closure to Yield Diastereomerically Pure (7'S-Me- or 7'R-Me-) Carba-LNA Nucleotide Analogs
Plashkevych, Oleksandr, Upadhayaya, Ram Shankar, Chattopadhyaya, Jyoti
Published in Current protocols in nucleic acid chemistry (01.06.2017)
Published in Current protocols in nucleic acid chemistry (01.06.2017)
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Journal Article
New parasite inhibitors encompassing novel conformationally-locked 5-acyl sulfamoyl adenosinesThis article is part of the Organic & Biomolecular Chemistry 10th Anniversary issue.Electronic supplementary information available: Spectral data (1H, 13C NMR, DEPT, HSQC, LCMS, Mass and HPLC) for all new compounds are included. See DOI: 10.1039/c2ob25879j
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Journal Article
Synthesis and structure of azole-fused indeno[2,1-c]quinolines and their anti-mycobacterial properties
Upadhayaya, Ram Shankar, Shinde, Popat D., Sayyed, Aftab Y., Kadam, Sandip A., Bawane, Amit N., Poddar, Avijit, Plashkevych, Oleksandr, Foldesi, Andras, Chattopadhyaya, Jyoti
Published in Organic & biomolecular chemistry (01.01.2010)
Published in Organic & biomolecular chemistry (01.01.2010)
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Journal Article
Synthesis and structure of azole-fused indeno[2,1-c]quinolines and their anti-mycobacterial propertiesElectronic supplementary information (ESI) available: Spectral data (1D-NMR, 2D-NMR, LCMS, Mass, HPLC and IR) for all new compounds is included. See DOI: 10.1039/c0ob00445f
Upadhayaya, Ram Shankar, Shinde, Popat D, Sayyed, Aftab Y, Kadam, Sandip A, Bawane, Amit N, Poddar, Avijit, Plashkevych, Oleksandr, Földesi, Andras, Chattopadhyaya, Jyoti
Year of Publication 15.12.2010
Year of Publication 15.12.2010
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