Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCβ-selective inhibitors
Tanaka, Masahiro, Sagawa, Shoichi, Hoshi, Jun-ichi, Shimoma, Fumito, Yasue, Katsutaka, Ubukata, Minoru, Ikemoto, Tomoyuki, Hase, Yasunori, Takahashi, Mitsuru, Sasase, Tomohiko, Ueda, Nobuhisa, Matsushita, Mutsuyoshi, Inaba, Takashi
Published in Bioorganic & medicinal chemistry (01.09.2006)
Published in Bioorganic & medicinal chemistry (01.09.2006)
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Journal Article
One-step synthesis of heteroaromatic-fused pyrrolidines via cyclopropane ring-opening reaction: application to the PKCbeta inhibitor JTT-010
Tanaka, Masahiro, Ubukata, Minoru, Matsuo, Takafumi, Yasue, Katsutaka, Matsumoto, Katsuya, Kajimoto, Yasuyuki, Ogo, Takashi, Inaba, Takashi
Published in Organic letters (16.08.2007)
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Published in Organic letters (16.08.2007)
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FIVE-MEMBERED CYCLIC AMIDE COMPOUND AND USE THEREOF
NAKAGAWA, YUICHI, MITANI, IKUO, IIDA, TETSUYA, TANAKA, MASAHIRO, UBUKATA, MINORU
Year of Publication 09.10.2008
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Year of Publication 09.10.2008
Patent
Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCbeta-selective inhibitors
Tanaka, Masahiro, Sagawa, Shoichi, Hoshi, Jun-ichi, Shimoma, Fumito, Yasue, Katsutaka, Ubukata, Minoru, Ikemoto, Tomoyuki, Hase, Yasunori, Takahashi, Mitsuru, Sasase, Tomohiko, Ueda, Nobuhisa, Matsushita, Mutsuyoshi, Inaba, Takashi
Published in Bioorganic & medicinal chemistry (01.09.2006)
Get full text
Published in Bioorganic & medicinal chemistry (01.09.2006)
Journal Article