The Small Molecule GMX1778 Is a Potent Inhibitor of NAD+ Biosynthesis: Strategy for Enhanced Therapy in Nicotinic Acid Phosphoribosyltransferase 1-Deficient Tumors
Watson, Mark, Roulston, Anne, Bélec, Laurent, Billot, Xavier, Marcellus, Richard, Bédard, Dominique, Bernier, Cynthia, Branchaud, Stéphane, Chan, Helen, Dairi, Kenza, Gilbert, Karine, Goulet, Daniel, Gratton, Michel-Olivier, Isakau, Henady, Jang, Anne, Khadir, Abdelkrim, Koch, Elizabeth, Lavoie, Manon, Lawless, Michael, Nguyen, Mai, Paquette, Denis, Turcotte, Émilie, Berger, Alvin, Mitchell, Matthew, Shore, Gordon C., Beauparlant, Pierre
Published in Molecular and Cellular Biology (01.11.2009)
Published in Molecular and Cellular Biology (01.11.2009)
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Preclinical development of the nicotinamide phosphoribosyl transferase inhibitor prodrug GMX1777
Beauparlant, Pierre, Bédard, Dominique, Bernier, Cynthia, Chan, Helen, Gilbert, Karine, Goulet, Daniel, Gratton, Michel-Olivier, Lavoie, Manon, Roulston, Anne, Turcotte, Emilie, Watson, Mark
Published in Anti-cancer drugs (01.06.2009)
Published in Anti-cancer drugs (01.06.2009)
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Abstract LB-33: Pre-clinical evaluation of AB-16B5, a monoclonal antibody specific for tumor-associated sCLU, demonstrates therapeutic potential as an inhibitor of EMT in prostate, pancreatic and lung cancer
Tremblay, Gilles B., Viau, Elisabeth, Malouin, Mireille, Turcotte, Émilie, Fortin, Annie, Filion, Mario
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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