OPC-41061, a Highly Potent Human Vasopressin V2-Receptor Antagonist: Pharmacological Profile and Aquaretic Effect by Single and Multiple Oral Dosing in Rats
Yamamura, Y, Nakamura, S, Itoh, S, Hirano, T, Onogawa, T, Yamashita, T, Yamada, Y, Tsujimae, K, Aoyama, M, Kotosai, K, Ogawa, H, Yamashita, H, Kondo, K, Tominaga, M, Tsujimoto, G, Mori, T
Published in The Journal of pharmacology and experimental therapeutics (01.12.1998)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.12.1998)
Journal Article
Comparison of kinetic properties of quinidine and dofetilide block of HERG channels
Tsujimae, Kenji, Suzuki, Shingo, Yamada, Mitsuhiko, Kurachi, Yoshihisa
Published in European journal of pharmacology (16.06.2004)
Published in European journal of pharmacology (16.06.2004)
Get full text
Journal Article
Mutational Analysis of Block and Facilitation of HERG Current by A Class III Anti-Arrhythmic Agent, Nifekalant
Hosaka, Yukio, Iwata, Miki, Kamiya, Narutoshi, Yamada, Mitsuhiko, Kinoshita, Kengo, Fukunishi, Yoshifumi, Tsujimae, Kenji, Hibino, Hiroshi, Aizawa, Yoshihusa, Inanobe, Atsushi, Nakamura, Haruki, Kurachi, Yoshihisa
Published in Channels (Austin, Tex.) (01.05.2007)
Published in Channels (Austin, Tex.) (01.05.2007)
Get full text
Journal Article
Antidiuretic Effects of a Nonpeptide Vasopressin V2-Receptor Agonist, OPC-51803, Administered Orally to Rats
Shigeki Nakamura, Takahiro Hirano, Kenji Tsujimae, Masashi Aoyama, Kazumi Kondo, Yoshitaka Yamamura, Toyoki Mori, Michiaki Tominaga
Published in The Journal of pharmacology and experimental therapeutics (01.12.2000)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.12.2000)
Journal Article
Characterization of a novel nonpeptide vasopressin V2‐agonist, OPC‐51803, in cells transfected human vasopressin receptor subtypes
Nakamura, Shigeki, Yamamura, Yoshitaka, Itoh, Shuji, Hirano, Takahiro, Tsujimae, Kenji, Aoyama, Masashi, Kondo, Kazumi, Ogawa, Hidenori, Shinohara, Tomoichi, Kan, Keizo, Tanada, Yoshihisa, Teramoto, Shuji, Sumida, Takumi, Nakayama, Sunao, Sekiguchi, Kazuo, Kambe, Toshimi, Tsujimoto, Gozoh, Mori, Toyoki, Tominaga, Michiaki
Published in British journal of pharmacology (01.04.2000)
Published in British journal of pharmacology (01.04.2000)
Get full text
Journal Article
In silico study on the effects of IKur block kinetics on prolongation of human action potential after atrial fibrillation-induced electrical remodeling
Tsujimae, Kenji, Murakami, Shingo, Kurachi, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (01.02.2008)
Published in American journal of physiology. Heart and circulatory physiology (01.02.2008)
Get full text
Journal Article
In silico study on the effects of I Kur block kinetics on prolongation of human action potential after atrial fibrillation-induced electrical remodeling
Tsujimae, Kenji, Murakami, Shingo, Kurachi, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (01.02.2008)
Published in American journal of physiology. Heart and circulatory physiology (01.02.2008)
Get full text
Journal Article
Frequency-dependent effects of various IKr blockers on cardiac action potential duration in a human atrial model
Tsujimae, Kenji, Suzuki, Shingo, Murakami, Shingo, Kurachi, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (01.07.2007)
Published in American journal of physiology. Heart and circulatory physiology (01.07.2007)
Get full text
Journal Article
Frequency-dependent effects of various I Kr blockers on cardiac action potential duration in a human atrial model
Tsujimae, Kenji, Suzuki, Shingo, Murakami, Shingo, Kurachi, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (01.07.2007)
Published in American journal of physiology. Heart and circulatory physiology (01.07.2007)
Get full text
Journal Article
In silico study on the effects of I^sub Kur^ block kinetics on prolongation of human action potential after atrial fibrillation-induced electrical remodeling
Tsujimae, Kenji, Murakami, Shingo, Kurachi, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (01.02.2008)
Get full text
Published in American journal of physiology. Heart and circulatory physiology (01.02.2008)
Journal Article
In silico study on the effects of IKUr block kinetics on prolongation of human action potential after atrial fibrillation-induced electrical remodeling
TSUJIMAE, Kenji, MURAKAMI, Shingo, KURACHI, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (2008)
Get full text
Published in American journal of physiology. Heart and circulatory physiology (2008)
Journal Article
Characterization of a novel nonpeptide vasopressin V 2 ‐agonist, OPC‐51803, in cells transfected human vasopressin receptor subtypes
Nakamura, Shigeki, Yamamura, Yoshitaka, Itoh, Shuji, Hirano, Takahiro, Tsujimae, Kenji, Aoyama, Masashi, Kondo, Kazumi, Ogawa, Hidenori, Shinohara, Tomoichi, Kan, Keizo, Tanada, Yoshihisa, Teramoto, Shuji, Sumida, Takumi, Nakayama, Sunao, Sekiguchi, Kazuo, Kambe, Toshimi, Tsujimoto, Gozoh, Mori, Toyoki, Tominaga, Michiaki
Published in British journal of pharmacology (30.01.2009)
Published in British journal of pharmacology (30.01.2009)
Get full text
Journal Article
Frequency-dependent effects of various I^sub Kr^ blockers on cardiac action potential duration in a human atrial model
Tsujimae, Kenji, Suzuki, Shingo, Murakami, Shingo, Kurachi, Yoshihisa
Published in American journal of physiology. Heart and circulatory physiology (01.07.2007)
Get full text
Published in American journal of physiology. Heart and circulatory physiology (01.07.2007)
Journal Article
In silico risk assessment for drug-induction of cardiac arrhythmia
Suzuki, Shingo, Murakami, Shingo, Tsujimae, Kenji, Findlay, Ian, Kurachi, Yoshihisa
Published in Progress in biophysics and molecular biology (01.09.2008)
Published in Progress in biophysics and molecular biology (01.09.2008)
Get full text
Journal Article
NITROGEN-CONTAINING COMPOUND AND PHARMACEUTICAL COMPOSITION
KOGA YASUO, MENJO YASUHIRO, UEDA MASATAKA, ONOGAWA TOSHIYUKI, OSHIMA KUNIO, TAKEMURA KENSHO, TAIRA SHINICHI, ISONO NAOHIRO, NAKAYAMA SUNAO, YAMABE HOKUTO, OSHIYAMA TAKASHI, MATSUMURA SHUJI, ITOTANI MOTOHIRO, TSUJIMAE KENJI, NAGASE TAKESHI, TAI KUNINORI
Year of Publication 12.11.2015
Get full text
Year of Publication 12.11.2015
Patent
NITROGEN-CONTAINING COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF ATRIAL FIBRILLATION
KOGA YASUO, MENJO YASUHIRO, UEDA MASATAKA, ONOGAWA TOSHIYUKI, OSHIMA KUNIO, MATSUMURA SHUUJI, TAIRA SHINICHI, ISONO NAOHIRO, TAKEMURA NORIAKI, NAKAYAMA SUNAO, YAMABE HOKUTO, OSHIYAMA TAKASHI, ITOTANI MOTOHIRO, TSUJIMAE KENJI, TAI KUNINORI, NAGASE TSUYOSHI
Year of Publication 20.07.2012
Get full text
Year of Publication 20.07.2012
Patent