Nonclassical Phenyl Bioisosteres as Effective Replacements in a Series of Novel Open-Source Antimalarials
Tse, Edwin G, Houston, Sevan D, Williams, Craig M, Savage, G. Paul, Rendina, Louis M, Hallyburton, Irene, Anderson, Mark, Sharma, Raman, Walker, Gregory S, Obach, R. Scott, Todd, Matthew H
Published in Journal of medicinal chemistry (22.10.2020)
Published in Journal of medicinal chemistry (22.10.2020)
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Journal Article
Experimentally Validated Pharmacoinformatics Approach to Predict hERG Inhibition Potential of New Chemical Entities
Munawar, Saba, Windley, Monique J, Tse, Edwin G, Todd, Matthew H, Hill, Adam P, Vandenberg, Jamie I, Jabeen, Ishrat
Published in Frontiers in pharmacology (19.09.2018)
Published in Frontiers in pharmacology (19.09.2018)
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Journal Article
The Metallodrug BOLD-100 Is a Potent Inhibitor of SARS-CoV-2 Replication and Has Broad-Acting Antiviral Activity
Labach, Daniel S, Kohio, Hinissan P, Tse, Edwin A, Paparisto, Ermela, Friesen, Nicole J, Pankovich, Jim, Bazett, Mark, Barr, Stephen D
Published in Biomolecules (Basel, Switzerland) (01.07.2023)
Published in Biomolecules (Basel, Switzerland) (01.07.2023)
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Journal Article
An Open Drug Discovery Competition: Experimental Validation of Predictive Models in a Series of Novel Antimalarials
Tse, Edwin G, Aithani, Laksh, Anderson, Mark, Cardoso-Silva, Jonathan, Cincilla, Giovanni, Conduit, Gareth J, Galushka, Mykola, Guan, Davy, Hallyburton, Irene, Irwin, Benedict W. J, Kirk, Kiaran, Lehane, Adele M, Lindblom, Julia C. R, Lui, Raymond, Matthews, Slade, McCulloch, James, Motion, Alice, Ng, Ho Leung, Öeren, Mario, Robertson, Murray N, Spadavecchio, Vito, Tatsis, Vasileios A, van Hoorn, Willem P, Wade, Alexander D, Whitehead, Thomas M, Willis, Paul, Todd, Matthew H
Published in Journal of medicinal chemistry (25.11.2021)
Published in Journal of medicinal chemistry (25.11.2021)
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Journal Article
Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus
Klug, Dana M, Tse, Edwin G, Silva, Daniel G, Cao, Yafeng, Charman, Susan A, Chauhan, Jyoti, Crighton, Elly, Dichiara, Maria, Drake, Chris, Drewry, David, da Silva Emery, Flavio, Ferrins, Lori, Graves, Lee, Hopkins, Emily, Kresina, Thomas A C, Lorente-Macías, Álvaro, Perry, Benjamin, Phipps, Richard, Quiroga, Bruno, Quotadamo, Antonio, Sabatino, Giada N, Sama, Anthony, Schätzlein, Andreas, Simpson, Quillon J, Steele, Jonathan, Shanu-Wilson, Julia, Sjö, Peter, Stapleton, Paul, Swain, Christopher J, Vaideanu, Alexandra, Xie, Huanxu, Zuercher, William, Todd, Matthew H
Published in ACS infectious diseases (08.12.2023)
Published in ACS infectious diseases (08.12.2023)
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Journal Article
Structure–Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis
Dichiara, Maria, Simpson, Quillon J., Quotadamo, Antonio, Jalani, Hitesh B., Huang, Anson X., Millard, Caroline C., Klug, Dana M., Tse, Edwin G., Todd, Matthew H., Silva, Daniel Gedder, da Silva Emery, Flavio, Carlson, J. Eric, Zheng, Shao-Liang, Vleminckx, Margot, Matheeussen, An, Caljon, Guy, Pollastri, Michael P., Sjö, Peter, Perry, Benjamin, Ferrins, Lori
Published in ACS infectious diseases (11.08.2023)
Published in ACS infectious diseases (11.08.2023)
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Journal Article
Comparison of knowledge, attitudes and practice of dental safety from eight countries at the turn of the century
Puttaiah, Raghunath, Miller, Kierste, Bedi, Daniela Raman, Shetty, Sadashiva, Almas, Khalid, Tse, Edwin, Kim, Byoung Ock, Youngblood, Dennis, Minquan, Du
Published in The journal of contemporary dental practice (2011)
Published in The journal of contemporary dental practice (2011)
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Journal Article
Open Source Code Contributions to Global Health: The Case of Antimalarial Drug Discovery
Turon, Gemma, Tse, Edwin, Qiu, Xin, Todd, Matthew, Duran-Frigola, Miquel
Published in ACS medicinal chemistry letters (12.09.2024)
Published in ACS medicinal chemistry letters (12.09.2024)
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