Comparative neuropharmacology of structurally distinct non-fentanyl opioids that are appearing on recreational drug markets worldwide
Vandeputte, Marthe M., Tsai, Meng-Hua M., Chen, Li, Glatfelter, Grant C., Walther, Donna, Stove, Christophe P., Shi, Lei, Baumann, Michael H.
Published in Drug and alcohol dependence (01.08.2023)
Published in Drug and alcohol dependence (01.08.2023)
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Alkoxy chain length governs the potency of 2-benzylbenzimidazole ‘nitazene’ opioids associated with human overdose
Glatfelter, Grant C., Vandeputte, Marthe M., Chen, Li, Walther, Donna, Tsai, Meng-Hua M., Shi, Lei, Stove, Christophe P., Baumann, Michael H.
Published in Psychopharmacology (01.12.2023)
Published in Psychopharmacology (01.12.2023)
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Binding preference at the μ-opioid receptor underlies distinct pharmacology of cyclopropyl versus valeryl analogs of fentanyl
Xie, Bing, Le Rouzic, Valerie P., Goldberg, Alexander, Tsai, Meng-Hua M., Chen, Li, Zhang, Tiffany, Sinha, Antara, Pan, Ying-Xian, Baumann, Michael H., Shi, Lei
Published in Neuropharmacology (01.04.2023)
Published in Neuropharmacology (01.04.2023)
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In Vitro Functional Profiling of Fentanyl and Nitazene Analogs at the μ‑Opioid Receptor Reveals High Efficacy for Gi Protein Signaling
Tsai, Meng-Hua M., Chen, Li, Baumann, Michael H., Canals, Meritxell, Javitch, Jonathan A., Lane, J. Robert, Shi, Lei
Published in ACS chemical neuroscience (21.02.2024)
Published in ACS chemical neuroscience (21.02.2024)
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The in vitro functional profiles of fentanyl and nitazene analogs at the μ-opioid receptor - high efficacy is dangerous regardless of signaling bias
Tsai, Meng-Hua M, Chen, Li, Baumann, Michael H, Canals, Meritxell, Javitch, Jonathan A, Lane, J Robert, Shi, Lei
Published in bioRxiv : the preprint server for biology (15.11.2023)
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Published in bioRxiv : the preprint server for biology (15.11.2023)
Journal Article
The in vitro functional profiles of fentanyl and nitazene analogs at the μ-opioid receptor - high efficacy is dangerous regardless of signaling bias
Tsai, Meng-Hua M, Chen, Li, Baumann, Michael H, Canals, Meritxell, Javitch, Jonathan A, Lane, J Robert, Shi, Lei
Published in bioRxiv (15.11.2023)
Published in bioRxiv (15.11.2023)
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