Update on Hsp90 inhibitors in clinical trial
Kim, Y S, Alarcon, S V, Lee, S, Lee, M-J, Giaccone, G, Neckers, L, Trepel, J B
Published in Current topics in medicinal chemistry (01.11.2009)
Published in Current topics in medicinal chemistry (01.11.2009)
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Selumetinib with and without erlotinib in KRAS mutant and KRAS wild-type advanced nonsmall-cell lung cancer
Carter, C.A., Rajan, A., Keen, C., Szabo, E., Khozin, S., Thomas, A., Brzezniak, C., Guha, U., Doyle, L.A., Steinberg, S.M., Xi, L., Raffeld, M., Tomita, Y., Lee, M.J., Lee, S., Trepel, J.B., Reckamp, K.L., Koehler, S., Gitlitz, B., Salgia, R., Gandara, D., Vokes, E., Giaccone, G.
Published in Annals of oncology (01.04.2016)
Published in Annals of oncology (01.04.2016)
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Modulation of tumor eIF4E by antisense inhibition: A phase I/II translational clinical trial of ISIS 183750—an antisense oligonucleotide against eIF4E—in combination with irinotecan in solid tumors and irinotecan‐refractory colorectal cancer
Duffy, A.G., Makarova‐Rusher, O.V., Ulahannan, S.V., Rahma, O.E., Fioravanti, S., Walker, M., Abdullah, S., Raffeld, M., Anderson, V., Abi‐Jaoudeh, N., Levy, E., Wood, B.J., Lee, S., Tomita, Y., Trepel, J.B., Steinberg, S.M., Revenko, A.S., MacLeod, A.R., Peer, C.J., Figg, W.D., Greten, T.F.
Published in International journal of cancer (01.10.2016)
Published in International journal of cancer (01.10.2016)
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A phase II study of durvalumab, a PD-L1 inhibitor and olaparib in recurrent ovarian cancer (OvCa)
Lee, J.-M., Annunziata, C.M., Houston, N., Kohn, E.C., Lipkowitz, S., Minasian, L., Nichols, E., Trepel, J., Trewhitt, K., Zia, F., Zimmer, A.D.S.
Published in Annals of oncology (01.10.2018)
Published in Annals of oncology (01.10.2018)
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A small molecule cell-impermeant Hsp90 antagonist inhibits tumor cell motility and invasion
TSUTSUMI, S, SCROGGINS, B, KOGA, F, LEE, M.-J, TREPEL, J, FELTS, S, CARRERAS, C, NECKERS, L
Published in Oncogene (10.04.2008)
Published in Oncogene (10.04.2008)
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The Hsp90 inhibitor geldanamycin selectively sensitizes Bcr-Abl-expressing leukemia cells to cytotoxic chemotherapy
BLAGOSKLONNY, M. V, FOJO, T, BHALLA, K. N, KIM, J-S, TREPEL, J. B, FIGG, W. D, RIVERA, Y, NECKERS, L. M
Published in Leukemia (01.10.2001)
Published in Leukemia (01.10.2001)
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DNA damage and cell cycle arrest induced by 2-(4-amino-3-methylphenyl)-5-fluorobenzothiazole (5F 203, NSC 703786) is attenuated in aryl hydrocarbon receptor deficient MCF-7 cells
TRAPANI, V, PATEL, V, LEONG, C.-O, CIOLINO, H. P, YEH, G. C, HOSE, C, TREPEL, J. B, STEVENS, M. F. G, SAUSVILLE, E. A, LOAIZA-PEREZ, A. I
Published in British journal of cancer (24.02.2003)
Published in British journal of cancer (24.02.2003)
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Sensitivity of epidermal growth factor receptor and ErbB2 exon 20 insertion mutants to Hsp90 inhibition
XU, W, SOGA, S, BEEBE, K, LEE, M. J, KIM, Y. S, TREPEL, J, NECKERS, L
Published in British journal of cancer (11.09.2007)
Published in British journal of cancer (11.09.2007)
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Tumor-intrinsic and tumor-extrinsic factors impacting hsp90- targeted therapy
Alarcon, S V, Mollapour, M, Lee, M-J, Tsutsumi, S, Lee, S, Kim, Y S, Prince, T, Apolo, A B, Giaccone, G, Xu, W, Neckers, L M, Trepel, J B
Published in Current molecular medicine (01.11.2012)
Published in Current molecular medicine (01.11.2012)
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Distinct immune characteristics in women with deleterious germline BRCA1/2 mutations (gBRCAm)-associated high-grade serous ovarian cancer (HGSOC)
Tomita, Y, Chiou, V, Lee, S, Yu, M, Houston, N, Lee, M.J, Kohn, E.C, Trepel, J
Published in Gynecologic oncology (01.04.2015)
Published in Gynecologic oncology (01.04.2015)
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FLT3 regulates β-catenin tyrosine phosphorylation, nuclear localization, and transcriptional activity in acute myeloid leukemia cells
KAJIGUCHI, T, CHUNG, E. J, LEE, S, STINE, A, KIYOI, H, NAOE, T, LEVIS, M. J, NECKERS, L, TREPEL, J. B
Published in Leukemia (01.12.2007)
Published in Leukemia (01.12.2007)
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A phase II study of TRC105 in patients with hepatocellular carcinoma who have progressed on sorafenib
Duffy, AG, Ulahannan, SV, Cao, L, Rahma, OE, Makarova-Rusher, OV, Kleiner, DE, Fioravanti, S, Walker, M, Carey, S, Yu, Y, Venkatesan, AM, Turkbey, B, Choyke, P, Trepel, J, Bollen, KC, Steinberg, SM, Figg, WD, Greten, TF
Published in United European gastroenterology journal (01.10.2015)
Published in United European gastroenterology journal (01.10.2015)
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Five-lipoxygenase inhibitors can mediate apoptosis in human breast cancer cell lines through complex eicosanoid interactions
Avis, I, Hong, S H, Martinez, A, Moody, T, Choi, Y H, Trepel, J, Das, R, Jett, M, Mulshine, J L
Published in The FASEB journal (01.09.2001)
Published in The FASEB journal (01.09.2001)
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Phase I study of lovastatin, an inhibitor of the mevalonate pathway, in patients with cancer
THIBAULT, A, DVORIT SAMID, REED, E, MYERS, C. E, TOMPKINS, A. C, FIGG, W. D, COOPER, M. R, HOHL, R. J, TREPEL, J, LIANG, B, PATRONAS, N, VENZON, D. J
Published in Clinical cancer research (01.03.1996)
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Published in Clinical cancer research (01.03.1996)
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Destabilization of Raf-1 by geldanamycin leads to disruption of the Raf-1-MEK-mitogen-activated protein kinase signalling pathway
Schulte, Theodor W., Blagosklonny, Mikhail V., Romanova, Larissa, Mushinski, J. Frederic, Monia, Brett P., Johnston, Joseph F., Nguyen, Phuongmai, Trepel, Jane, Neckers, Leonard M.
Published in Molecular and Cellular Biology (01.10.1996)
Published in Molecular and Cellular Biology (01.10.1996)
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Terminal Neuroendocrine Differentiation of Human Prostate Carcinoma Cells in Response to Increased Intracellular Cyclic AMP
Y.-J. Bang, Pirnia, F., W.-G. Fang, Kang, W. K., Sartor, O., Whitesell, L., Ha, M. J., Tsokos, M., Sheahan, M. D., Nguyen, P., Niklinski, W. T., Myers, C. E., Trepel, J. B.
Published in Proceedings of the National Academy of Sciences - PNAS (07.06.1994)
Published in Proceedings of the National Academy of Sciences - PNAS (07.06.1994)
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Regulation of BRCA1 by protein degradation
BLAGOSKLONNY, M. V, AN, W. G, MELILLO, G, NGUYEN, P, TREPEL, J. B, NECKERS, L. M
Published in Oncogene (11.11.1999)
Published in Oncogene (11.11.1999)
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Drug-induced apoptosis is not necessarily dependent on macromolecular synthesis or proliferation in the p53-negative human prostate cancer cell line PC-3
BORNER, M. M, MYERS, C. E, SARTOR, O, SEI, Y, TOKO, T, TREPEL, J. B, SCHNEIDER, E
Published in Cancer research (Chicago, Ill.) (15.05.1995)
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Published in Cancer research (Chicago, Ill.) (15.05.1995)
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