In Vivo Mutagenicity Testing of Arylboronic Acids and Esters
Masuda‐Herrera, Melisa J., Dobo, Krista L., Kenyon, Michelle O., Kenny, Julia D., Galloway, Sheila M., Escobar, Patricia A., Reddy, M. Vijayaraj, Jolly, Robert A., Trejo‐Martin, Alejandra, Brown, Caren, Mckeon, Marie, Young, Megan, Bruce, Shannon, Pant, Kamala, Dutta, Aparajita, Kulkarni, Rohan, Bercu, Joel P.
Published in Environmental and molecular mutagenesis (01.12.2019)
Published in Environmental and molecular mutagenesis (01.12.2019)
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An Evaluation of the Occupational Health Hazards of Peptide Couplers
Graham, Jessica C., Trejo-Martin, Alejandra, Chilton, Martyn L., Kostal, Jakub, Bercu, Joel, Beutner, Gregory L., Bruen, Uma S., Dolan, David G., Gomez, Stephen, Hillegass, Jedd, Nicolette, John, Schmitz, Matthew
Published in Chemical research in toxicology (20.06.2022)
Published in Chemical research in toxicology (20.06.2022)
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The utility of hERG channel inhibition data in the derivation of occupational exposure limits
Parker, Jillian A., Fung, Ernest S., Trejo-Martin, Alejandra, Liang, Lisa, Gibbs, Katherine, Bandara, Suren, Chen, Stephanie, Sandhu, Reena, Bercu, Joel, Maier, Andrew
Published in Regulatory toxicology and pharmacology (01.10.2022)
Published in Regulatory toxicology and pharmacology (01.10.2022)
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Discovery of velpatasvir (GS-5816): A potent pan-genotypic HCV NS5A inhibitor in the single-tablet regimens Vosevi® and Epclusa
Link, John O., Taylor, James G., Trejo-Martin, Alejandra, Kato, Darryl, Katana, Ashley A., Krygowski, Evan S., Yang, Zheng-Yu, Zipfel, Sheila, Cottell, Jeromy J., Bacon, Elizabeth M., Tran, Chinh V., Yang, Cheng Y., Wang, Yujin, Wang, Kelly W., Zhao, Guangyu, Cheng, Guofeng, Tian, Yang, Gong, Ruoyu, Lee, Yu-Jen, Yu, Mei, Gorman, Eric, Mogalian, Erik, Perry, Jason K.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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SYNTHESIS OF HETEROARYL-FUSED PYRAZOLES AS P38 KINASE INHIBITORS
Abbot, Sarah C., Billedeau, Roland J., Dewdney, Nolan J., Gabriel, Tobias, Goldstein, David M., McCaleb, Kristen L., Soth, Michael, Trejo-Martin, Teresa Alejandra, Zecic, Hasim
Published in Heterocycles (01.11.2009)
Published in Heterocycles (01.11.2009)
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Journal Article
Quantum-Mechanics Calculations Elucidate Skin-Sensitizing Pharmaceutical Compounds
Kostal, Jakub, Voutchkova-Kostal, Adelina, Bercu, Joel P., Graham, Jessica C., Hillegass, Jedd, Masuda-Herrera, Melisa, Trejo-Martin, Alejandra, Gould, Janet
Published in Chemical research in toxicology (19.08.2024)
Published in Chemical research in toxicology (19.08.2024)
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In silico toxicology protocols
Myatt, Glenn J, Ahlberg, Ernst, Akahori, Yumi, Allen, David, Amberg, Alexander, Anger, Lennart T, Aptula, Aynur, Auerbach, Scott, Beilke, Lisa, Bellion, Phillip, Benigni, Romualdo, Bercu, Joel, Booth, Ewan D, Bower, Dave, Brigo, Alessandro, Burden, Natalie, Cammerer, Zoryana, Cronin, Mark T D, Cross, Kevin P, Custer, Laura, Dettwiler, Magdalena, Dobo, Krista, Ford, Kevin A, Fortin, Marie C, Gad-McDonald, Samantha E, Gellatly, Nichola, Gervais, Véronique, Glover, Kyle P, Glowienke, Susanne, Van Gompel, Jacky, Gutsell, Steve, Hardy, Barry, Harvey, James S, Hillegass, Jedd, Honma, Masamitsu, Hsieh, Jui-Hua, Hsu, Chia-Wen, Hughes, Kathy, Johnson, Candice, Jolly, Robert, Jones, David, Kemper, Ray, Kenyon, Michelle O, Kim, Marlene T, Kruhlak, Naomi L, Kulkarni, Sunil A, Kümmerer, Klaus, Leavitt, Penny, Majer, Bernhard, Masten, Scott, Miller, Scott, Moser, Janet, Mumtaz, Moiz, Muster, Wolfgang, Neilson, Louise, Oprea, Tudor I, Patlewicz, Grace, Paulino, Alexandre, Lo Piparo, Elena, Powley, Mark, Quigley, Donald P, Reddy, M Vijayaraj, Richarz, Andrea-Nicole, Ruiz, Patricia, Schilter, Benoit, Serafimova, Rositsa, Simpson, Wendy, Stavitskaya, Lidiya, Stidl, Reinhard, Suarez-Rodriguez, Diana, Szabo, David T, Teasdale, Andrew, Trejo-Martin, Alejandra, Valentin, Jean-Pierre, Vuorinen, Anna, Wall, Brian A, Watts, Pete, White, Angela T, Wichard, Joerg, Witt, Kristine L, Woolley, Adam, Woolley, David, Zwickl, Craig, Hasselgren, Catrin
Published in Regulatory toxicology and pharmacology (01.07.2018)
Published in Regulatory toxicology and pharmacology (01.07.2018)
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Journal Article
Mechanisms of Nitrosamine Mutagenicity and Their Relationship to Rodent Carcinogenic Potency
Snodin, David J., Trejo-Martin, Alejandra, Ponting, David J., Smith, Graham F., Czich, Andreas, Cross, Kevin, Custer, Laura, Elloway, Joanne, Greene, Nigel, Kalgutkar, Amit S., Stalford, Susanne A., Tennant, Rachael E., Vock, Esther, Zalewski, Adam, Ziegler, Verena, Dobo, Krista L.
Published in Chemical research in toxicology (19.02.2024)
Published in Chemical research in toxicology (19.02.2024)
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Journal Article
Acceptable intakes (AIs) for 11 small molecule N-nitrosamines (NAs)
Bercu, Joel P., Masuda-Herrera, Melisa, Trejo-Martin, Alejandra, Sura, Priyanka, Jolly, Robert, Kenyon, Michelle, Thomas, Rob, Ponting, David J., Snodin, David, Tuschl, Gregor, Simon, Stephanie, De Vlieger, Kathleen, Hutchinson, Richard, Czich, Andreas, Glowienke, Susanne, Reddy, M. Vijayaraj, Johanssen, Sandra, Vock, Esther, Claude, Nancy, Weaver, Richard J.
Published in Regulatory toxicology and pharmacology (01.08.2023)
Published in Regulatory toxicology and pharmacology (01.08.2023)
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Journal Article
Use of the bacterial reverse mutation assay to predict carcinogenicity of N-nitrosamines
Trejo-Martin, Alejandra, Bercu, Joel P., Thresher, Andrew, Tennant, Rachael E., Thomas, Robert F., Cross, Kevin, Czich, Andreas, Waese, Kerstin, Nicolette, John J., Murray, Joel, Sonders, Paul, Kondratiuk, Alison, Cheung, Jennifer R., Thomas, Dean, Lynch, Anthony, Harvey, James, Glowienke, Susanne, Custer, Laura, Escobar, Patricia A.
Published in Regulatory toxicology and pharmacology (01.11.2022)
Published in Regulatory toxicology and pharmacology (01.11.2022)
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Genetic toxicology in silico protocol
Hasselgren, Catrin, Ahlberg, Ernst, Akahori, Yumi, Amberg, Alexander, Anger, Lennart T, Atienzar, Franck, Auerbach, Scott, Beilke, Lisa, Bellion, Phillip, Benigni, Romualdo, Bercu, Joel, Booth, Ewan D, Bower, Dave, Brigo, Alessandro, Cammerer, Zoryana, Cronin, Mark T D, Crooks, Ian, Cross, Kevin P, Custer, Laura, Dobo, Krista, Doktorova, Tatyana, Faulkner, David, Ford, Kevin A, Fortin, Marie C, Frericks, Markus, Gad-McDonald, Samantha E, Gellatly, Nichola, Gerets, Helga, Gervais, Véronique, Glowienke, Susanne, Van Gompel, Jacky, Harvey, James S, Hillegass, Jedd, Honma, Masamitsu, Hsieh, Jui-Hua, Hsu, Chia-Wen, Barton-Maclaren, Tara S, Johnson, Candice, Jolly, Robert, Jones, David, Kemper, Ray, Kenyon, Michelle O, Kruhlak, Naomi L, Kulkarni, Sunil A, Kümmerer, Klaus, Leavitt, Penny, Masten, Scott, Miller, Scott, Moudgal, Chandrika, Muster, Wolfgang, Paulino, Alexandre, Lo Piparo, Elena, Powley, Mark, Quigley, Donald P, Reddy, M Vijayaray, Richarz, Andrea-Nicole, Schilter, Benoit, Snyder, Ronald D, Stavitskaya, Lidiya, Stidl, Reinhard, Szabo, David T, Teasdale, Andrew, Tice, Raymond R, Trejo-Martin, Alejandra, Vuorinen, Anna, Wall, Brian A, Watts, Pete, White, Angela T, Wichard, Joerg, Witt, Kristine L, Woolley, Adam, Woolley, David, Zwickl, Craig, Myatt, Glenn J
Published in Regulatory toxicology and pharmacology (01.10.2019)
Published in Regulatory toxicology and pharmacology (01.10.2019)
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Journal Article
A cross-industry collaboration to assess if acute oral toxicity (Q)SAR models are fit-for-purpose for GHS classification and labelling
Bercu, Joel, Masuda‐Herrera, Melisa J., Trejo-Martin, Alejandra, Hasselgren, Catrin, Lord, Jean, Graham, Jessica, Schmitz, Matthew, Milchak, Lawrence, Owens, Colin, Lal, Surya Hari, Robinson, Richard Marchese, Whalley, Sarah, Bellion, Phillip, Vuorinen, Anna, Gromek, Kamila, Hawkins, William A., van de Gevel, Iris, Vriens, Kathleen, Kemper, Raymond, Naven, Russell, Ferrer, Pierre, Myatt, Glenn J.
Published in Regulatory toxicology and pharmacology (01.03.2021)
Published in Regulatory toxicology and pharmacology (01.03.2021)
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Journal Article
Calculating qualified non-mutagenic impurity levels: Harmonization of approaches
Graham, Jessica C., Powley, Mark W., Udovic, Erika, Glowienke, Susanne, Nicolette, John, Parris, Patricia, Kenyon, Michelle, White, Angela, Maisey, Ailis, Harvey, James, Martin, Elizabeth A., Dowdy, Eric, Masuda-Herrera, Melisa, Trejo-Martin, Alejandra, Bercu, Joel
Published in Regulatory toxicology and pharmacology (01.11.2021)
Published in Regulatory toxicology and pharmacology (01.11.2021)
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Journal Article
Corrigendum to a cross-industry collaboration to assess if acute toxicity (Q)SAR models are fit-for-purpose for GHS classification and labelling. Regulatory toxicology and pharmacology (2021) 104843
Bercu, Joel, Masuda Herrera, Melisa J., Trejo-Martin, Alejandra, Hasselgren, Catrin, Lord, Jean, Graham, Jessica, Schmitz, Matthew, Milchak, Lawrence, Owens, Colin, Lal, Surya Hari, Robinson, Richard Marchese, Whalley, Sarah, Bellion, Phillip, Vuorinen, Anna, Gromek, Kamila, Hawkins, William A., Van de Gevel, Iris, Vriens, Kathleen, Kemper, Raymond, Naven, Russell, Ferrer, Pierre, Myatt, Glenn J.
Published in Regulatory toxicology and pharmacology (01.06.2022)
Published in Regulatory toxicology and pharmacology (01.06.2022)
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Journal Article
Extending (Q)SARs to incorporate proprietary knowledge for regulatory purposes: is aromatic N-oxide a structural alert for predicting DNA-reactive mutagenicity?
Amberg, Alexander, Anger, Lennart T, Bercu, Joel, Bower, David, Cross, Kevin P, Custer, Laura, Harvey, James S, Hasselgren, Catrin, Honma, Masamitsu, Johnson, Candice, Jolly, Robert, Kenyon, Michelle O, Kruhlak, Naomi L, Leavitt, Penny, Quigley, Donald P, Miller, Scott, Snodin, David, Stavitskaya, Lidiya, Teasdale, Andrew, Trejo-Martin, Alejandra, White, Angela T, Wichard, Joerg, Myatt, Glenn J
Published in Mutagenesis (06.03.2019)
Published in Mutagenesis (06.03.2019)
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Journal Article
Principles and procedures for handling out-of-domain and indeterminate results as part of ICH M7 recommended (Q)SAR analyses
Amberg, Alexander, Andaya, Roxanne V., Anger, Lennart T., Barber, Chris, Beilke, Lisa, Bercu, Joel, Bower, Dave, Brigo, Alessandro, Cammerer, Zoryanna, Cross, Kevin P., Custer, Laura, Dobo, Krista, Gerets, Helga, Gervais, Véronique, Glowienke, Susanne, Gomez, Stephen, Van Gompel, Jacky, Harvey, James, Hasselgren, Catrin, Honma, Masamitsu, Johnson, Candice, Jolly, Robert, Kemper, Raymond, Kenyon, Michelle, Kruhlak, Naomi, Leavitt, Penny, Miller, Scott, Muster, Wolfgang, Naven, Russell, Nicolette, John, Parenty, Alexis, Powley, Mark, Quigley, Donald P., Reddy, M. Vijayaraj, Sasaki, Jennifer C., Stavitskaya, Lidiya, Teasdale, Andrew, Trejo-Martin, Alejandra, Weiner, Sandy, Welch, Dennie S., White, Angela, Wichard, Joerg, Woolley, David, Myatt, Glenn J.
Published in Regulatory toxicology and pharmacology (01.03.2019)
Published in Regulatory toxicology and pharmacology (01.03.2019)
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Journal Article
In silico approaches in carcinogenicity hazard assessment: Current status and future needs
Tice, Raymond R., Bassan, Arianna, Amberg, Alexander, Anger, Lennart T., Beal, Marc A., Bellion, Phillip, Benigni, Romualdo, Birmingham, Jeffrey, Brigo, Alessandro, Bringezu, Frank, Ceriani, Lidia, Crooks, Ian, Cross, Kevin, Elespuru, Rosalie, Faulkner, David M., Fortin, Marie C., Fowler, Paul, Frericks, Markus, Gerets, Helga H.J., Jahnke, Gloria D., Jones, David R., Kruhlak, Naomi L., Piparo, Elena Lo, Lopez-Belmonte, Juan, Luniwal, Amarjit, Luu, Alice, Madia, Federica, Manganelli, Serena, Manickam, Balasubramanian, Mestres, Jordi, Mihalchik-Burhans, Amy L., Neilson, Louise, Pandiri, Arun, Pavan, Manuela, Rider, Cynthia V., Rooney, John P., Trejo-Martin, Alejandra, Watanabe-Sailor, Karen H., White, Angela T., Woolley, David, Myatt, Glenn J.
Published in Computational toxicology (01.11.2021)
Published in Computational toxicology (01.11.2021)
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Spiropiperidine CCR5 antagonists
Rotstein, David M., Gabriel, Stephen D., Makra, Ferenc, Filonova, Lubov, Gleason, Shelley, Brotherton-Pleiss, Christine, Setti, Lina Q., Trejo-Martin, Alejandra, Lee, Eun Kyung, Sankuratri, Surya, Ji, Changhua, deRosier, Andre, Dioszegi, Marianna, Heilek, Gabrielle, Jekle, Andreas, Berry, Pamela, Weller, Paul, Mau, Cheng-I.
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Journal Article
ChemInform Abstract: Synthesis of Heteroaryl-Fused Pyrazoles as P38 Kinase Inhibitors
Abbot, Sarah C., Billedeau, Roland J., Dewdney, Nolan J., Gabriel, Tobias, Goldstein, David M., McCaleb, Kristen L., Soth, Michael, Trejo-Martin, Teresa Alejandra, Zecic, Hasim
Published in ChemInform (30.03.2010)
Published in ChemInform (30.03.2010)
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