Tyrosine Kinase 2-mediated Signal Transduction in T Lymphocytes Is Blocked by Pharmacological Stabilization of Its Pseudokinase Domain
Tokarski, John S., Zupa-Fernandez, Adriana, Tredup, Jeffrey A., Pike, Kristen, Chang, ChiehYing, Xie, Dianlin, Cheng, Lihong, Pedicord, Donna, Muckelbauer, Jodi, Johnson, Stephen R., Wu, Sophie, Edavettal, Suzanne C., Hong, Yang, Witmer, Mark R., Elkin, Lisa L., Blat, Yuval, Pitts, William J., Weinstein, David S., Burke, James R.
Published in The Journal of biological chemistry (24.04.2015)
Published in The Journal of biological chemistry (24.04.2015)
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Synthesis and SAR of new pyrrolo[2,1- f][1,2,4]triazines as potent p38α MAP kinase inhibitors
Wrobleski, Stephen T., Lin, Shuqun, Hynes, John, Wu, Hong, Pitt, Sidney, Shen, Ding Ren, Zhang, Rosemary, Gillooly, Kathleen M., Shuster, David J., McIntyre, Kim W., Doweyko, Arthur M., Kish, Kevin F., Tredup, Jeffrey A., Duke, Gerald J., Sack, John S., McKinnon, Murray, Dodd, John, Barrish, Joel C., Schieven, Gary L., Leftheris, Katerina
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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Decrypting the Biochemical Function of an Essential Gene from Streptococcus pneumoniae Using ThermoFluor® Technology
Carver, Theodore E., Bordeau, Brian, Cummings, Maxwell D., Petrella, Eugene C., Pucci, Michael J., Zawadzke, Laura E., Dougherty, Brian A., Tredup, Jeffrey A., Bryson, James W., Yanchunas, Joseph, Doyle, Michael L., Witmer, Mark R., Nelen, Marina I., DesJarlais, Renee L., Jaeger, Edward P., Devine, Heather, Asel, Eric D., Springer, Barry A., Bone, Roger, Salemme, F. Raymond, Todd, Matthew J.
Published in The Journal of biological chemistry (25.03.2005)
Published in The Journal of biological chemistry (25.03.2005)
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Discovery of N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4- morpholineacetamide as a Novel and Potent Inhibitor of Inosine Monophosphate Dehydrogenase with Excellent in Vivo Activity
Dhar, T. G. Murali, Shen, Zhongqi, Guo, Junqing, Liu, Chunjian, Watterson, Scott H, Gu, Henry H, Pitts, William J, Fleener, Catherine A, Rouleau, Katherine A, Sherbina, N. Z, McIntyre, Kim W, Witmer, Mark R, Tredup, Jeffrey A, Chen, Bang-Chi, Zhao, Rulin, Bednarz, Mark S, Cheney, Daniel L, MacMaster, John F, Miller, Laura M, Berry, Karen K, Harper, Timothy W, Barrish, Joel C, Hollenbaugh, Diane L, Iwanowicz, Edwin J
Published in Journal of medicinal chemistry (23.05.2002)
Published in Journal of medicinal chemistry (23.05.2002)
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BMS-229724 Is a Tight-Binding Inhibitor of Cytosolic Phospholipase A2 That Acts at the Lipid/Water Interface and Possesses Anti-Inflammatory Activity in Skin Inflammation Models
Burke, J R, Davern, L B, Stanley, P L, Gregor, K R, Banville, J, Remillard, R, Russell, J W, Brassil, P J, Witmer, M R, Johnson, G, Tredup, J A, Tramposch, K M
Published in The Journal of pharmacology and experimental therapeutics (01.07.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.2001)
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Structural basis for the high-affinity binding of pyrrolotriazine inhibitors of p38 MAP kinase
Sack, John S., Kish, Kevin F., Pokross, Matthew, Xie, Dianlin, Duke, Gerald J., Tredup, Jeffrey A., Kiefer, Susan E., Newitt, John A.
Published in Acta crystallographica. Section D, Biological crystallography. (01.07.2008)
Published in Acta crystallographica. Section D, Biological crystallography. (01.07.2008)
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Discovery of N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4-morpholineacetamide as a Novel and Potent Inhibitor of Inosine Monophosphate Dehydrogenase (IMPDH) with Excellent in Vivo Activity
Murali Dhar, T. G, Shen, Zhongqi, Guo, Junqing, Liu, Chunjian, Watterson, Scott H, Gu, Henry H, Pitts, William J, Fleener, Catherine A, Rouleau, Katherine A, Sherbina, N. Z, McIntyre, Kim W, Shuster, David J, Witmer, Mark R, Tredup, Jeffrey A, Chen, Bang-Chi, Zhao, Rulin, Bednarz, Mark S, Cheney, Daniel L, MacMaster, John F, Miller, Laura M, Berry, Karen K, Harper, Timothy W, Barrish, Joel C, Hollenbaugh, Diane L, Iwanowicz, Edwin J
Published in Journal of medicinal chemistry (07.11.2002)
Published in Journal of medicinal chemistry (07.11.2002)
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Competitive, Reversible Inhibition of Cytosolic Phospholipase A2 at the Lipid-Water Interface by Choline Derivatives That Partially Partition into the Phospholipid Bilayer
Burke, J R, Witmer, M R, Zusi, F C, Gregor, K R, Davern, L B, Padmanabha, R, Swann, R T, Smith, D, Tredup, J A, Micanovic, R, Manly, S P, Villafranca, J J, Tramposch, K M
Published in The Journal of biological chemistry (02.07.1999)
Published in The Journal of biological chemistry (02.07.1999)
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Journal Article
Decrypting the Biochemical Function of an Essential Gene from Streptococcus pneumoniae Using ThermoFluor® Technology
Theodore E. Carver, Brian Bordeau, Maxwell D. Cummings, Eugene C. Petrella, Michael J. Pucci, Laura E. Zawadzke, Brian A. Dougherty, Jeffrey A. Tredup, James W. Bryson, Joseph Yanchunas, Jr, Michael L. Doyle, Mark R. Witmer, Marina I. Nelen, Renee L. DesJarlais, Edward P. Jaeger, Heather Devine, Eric D. Asel, Barry A. Springer, Roger Bone, F. Raymond Salemme, Matthew J. Todd
Published in The Journal of biological chemistry (25.03.2005)
Published in The Journal of biological chemistry (25.03.2005)
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Journal Article
Presence of Glycerol Masks the Effects of Phosphorylation on the Catalytic Efficiency of Cytosolic Phospholipase A2
Burke, James R., Guenther, Matthew G., Witmer, Mark R., Tredup, Jeffrey A., Hail, Mark E., Micanovic, Radmila, Villafranca, Joseph J.
Published in Archives of biochemistry and biophysics (01.05.1997)
Published in Archives of biochemistry and biophysics (01.05.1997)
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