Oxidative alpha,omega-diyne coupling as an approach towards novel peptidic macrocycles
Verlinden, S., Geudens, N., Martins, J. C., Tourwe, D., Ballet, S., Verniest, G.
Published in Organic & biomolecular chemistry (28.09.2015)
Published in Organic & biomolecular chemistry (28.09.2015)
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Journal Article
Rapid construction of substituted 3-amino-1,5-benzothiazepin-4(5H)-one dipeptide scaffolds through an Ugi-4CR-Ullmann cross-coupling sequence
Van der Poorten, O., Van den Hauwe, R., Hollanders, K., Maes, B. U. W., Tourwe, D., Jida, M., Ballet, S.
Published in Organic & biomolecular chemistry (2018)
Published in Organic & biomolecular chemistry (2018)
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Journal Article
DFT-based ranking of zinc-binding groups in histone deacetylase inhibitors
Vanommeslaeghe, K., Loverix, S., Geerlings, P., Tourwé, D.
Published in Bioorganic & medicinal chemistry (01.11.2005)
Published in Bioorganic & medicinal chemistry (01.11.2005)
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Journal Article
Influence of Stacking on the Hydrogen Bond Donating Potential of Nucleic Bases
Vanommeslaeghe, K, Mignon, P, Loverix, S, Tourwé, D, Geerlings, P
Published in Journal of chemical theory and computation (01.09.2006)
Published in Journal of chemical theory and computation (01.09.2006)
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Journal Article
New [99mTc]bombesin analogues with improved biodistribution for targeting gastrin releasing-peptide receptor-positive tumors
García Garayoa, E, Schweinsberg, C, Maes, V, Rüegg, D, Blanc, A, Bläuenstein, P, Tourwé, D A, Beck-Sickinger, A G, Schubiger, P A
Published in The quarterly journal of nuclear medicine and molecular imaging (01.03.2007)
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Published in The quarterly journal of nuclear medicine and molecular imaging (01.03.2007)
Journal Article
A Metabolic Screening Study of Trichostatin A (TSA) and TSA-Like Histone Deacetylase Inhibitors in Rat and Human Primary Hepatocyte Cultures
Elaut, G, Laus, G, Alexandre, E, Richert, L, Bachellier, P, Tourwé, D, Rogiers, V, Vanhaecke, T
Published in The Journal of pharmacology and experimental therapeutics (01.04.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2007)
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Journal Article
Effect of temperature on retention of enantiomers of β-methyl amino acids on a teicoplanin chiral stationary phase
Péter, Antal, Török, Gabriella, Armstrong, Daniel W, Tóth, Géza, Tourwé, Dirk
Published in Journal of Chromatography A (18.12.1998)
Published in Journal of Chromatography A (18.12.1998)
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Journal Article
Conference Proceeding
Amide analogues of TSA: synthesis, binding mode analysis and HDAC inhibition
Van Ommeslaeghe, K, Elaut, G, Brecx, V, Papeleu, P, Iterbeke, K, Geerlings, P, Tourwé, D, Rogiers, V
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
Published in Bioorganic & medicinal chemistry letters (02.06.2003)
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Journal Article
Bradykinin analogs containing the 4-amino-2-benzazepin-3-one scaffold at the C-terminus
Ballet, S., De Wachter, R., Van Rompaey, K., Tömböly, Cs, Feytens, D., Töth, G., Quartara, L., Cucchi, P., Meini, S., Tourwé, D.
Published in Journal of peptide science (01.03.2007)
Published in Journal of peptide science (01.03.2007)
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Journal Article
New endomorphin analogs with mu-agonist and delta-antagonist properties
Tóth, G., Keresztes, A., Tömböly, Cs, Péter, A., Fülöp, F., Tourwé, D., Navratilova, E., Varga, É., Roeske, W. R., Yamamura, H. I., Szucs, M., Borsodi, A.
Published in Pure and applied chemistry (01.01.2004)
Published in Pure and applied chemistry (01.01.2004)
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Journal Article
LC enantioseparation of tryptophan analogs on α-cyclodextrin stationary phase
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Conference Proceeding
Journal Article
In vitro and in vivo evaluation of new radiolabeled neurotensin(8–13) analogues with high affinity for NT1 receptors
García-Garayoa, Elisa, Allemann-Tannahill, Lesley, Bläuenstein, Peter, Willmann, Martine, Carrel-Rémy, Nathalie, Tourwé, Dirk, Iterbeke, Koen, Conrath, Peter, Schubiger, P.August
Published in Nuclear medicine and biology (01.01.2001)
Published in Nuclear medicine and biology (01.01.2001)
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Journal Article
Synthesis and biological evaluation of constrained analogues of the opioid peptide H-Tyr-d-Ala-Phe-Gly-NH2 using the 4-amino-2-benzazepin-3-one scaffold
Ballet, S., Frycia, A., Piron, J., Chung, N.N., Schiller, P.W., Kosson, P., Lipkowski, A.W., Tourwé, D.
Published in The journal of peptide research (01.11.2005)
Published in The journal of peptide research (01.11.2005)
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Journal Article
High-performance liquid chromatographic separation of the enantiomers of unusual α-amino acid analogues
Péter, Antal, Olajos, Edit, Casimir, Richard, Tourwé, Dirk, Broxterman, Quirinus B, Kaptein, Bernard, Armstrong, Daniel W
Published in Journal of Chromatography A (25.02.2000)
Published in Journal of Chromatography A (25.02.2000)
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Journal Article
Conference Proceeding
Unprecedented Sigmatropic Rearrangements Leading to 2,3-Dihydro-1H-2-benzazepine-3-carboxylic Acid
Martins, José C, Van Rompaey, Karolien, Wittmann, Guyla, Tömböly, Csaba, Tóth, Géza, De Kimpe, Norbert, Tourwé, Dirk
Published in Journal of organic chemistry (20.04.2001)
Published in Journal of organic chemistry (20.04.2001)
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Journal Article