Pharmacokinetics of Tropifexor, a Potent Farnesoid X Receptor Agonist, in Participants With Varying Degrees of Hepatic Impairment
Chen, Jin, Gu, Jessie, Shah, Bharti, Stringer, Rowan, Reis da Silva Torrao, Leonel, Hackling, Melissa, Nidamarthy, Prasanna Kumar, Prince, William T, Woessner, Ralph
Published in Journal of clinical pharmacology (01.04.2022)
Published in Journal of clinical pharmacology (01.04.2022)
Get more information
Journal Article
Non‐clinical characterization of the disposition of EMA401, a novel small molecule angiotensin II type 2 receptor (AT2R) antagonist
Murgasova, Renata, Carreras, Ester Tor, Suetterlin‐Hachmann, Martina, Silva Torrao, Leonel Reis, Kittelmann, Matthias, Alexandra, Vargas, Fredenhagen, Andreas
Published in Biopharmaceutics & drug disposition (01.04.2020)
Published in Biopharmaceutics & drug disposition (01.04.2020)
Get full text
Journal Article
Synthesis and structure–activity relationships of ionizable 1,3,4-oxadiazol-2(3H)-ones as peripherally selective FAAH inhibitors with improved aqueous solubility
Beliaev, Alexandre, Ferreira, Humberto S., Learmonth, David A., Bonifácio, Maria João, Torrão, Leonel, Pires, Nuno M., Soares-da-Silva, Patrício, Kiss, László E.
Published in Pure and applied chemistry (01.04.2016)
Published in Pure and applied chemistry (01.04.2016)
Get full text
Journal Article
Species differences in pharmacokinetic and pharmacodynamic properties of nebicapone
Bonifácio, Maria João, Loureiro, Ana I., Torrão, Leonel, Fernandes-Lopes, Carlos, Wright, Lyndon, Pinho, Maria João, Soares-da-Silva, Patrício
Published in Biochemical pharmacology (15.10.2009)
Published in Biochemical pharmacology (15.10.2009)
Get full text
Journal Article
Discovery of a Long-Acting, Peripherally Selective Inhibitor of Catechol-O-methyltransferase
Kiss, László E, Ferreira, Humberto S, Torrão, Leonel, Bonifácio, Maria João, Palma, P. Nuno, Soares-da-Silva, Patrício, Learmonth, David A
Published in Journal of medicinal chemistry (22.04.2010)
Published in Journal of medicinal chemistry (22.04.2010)
Get full text
Journal Article
Chronopharmacology of nebicapone, a new catechol-O-methyltransferase inhibitor
Almeida, Luis, Loureiro, Ana I, Vaz-da-Silva, Manuel, Torrão, Leonel, Maia, Joana, Fernandes-Lopes, Carlos, Falcão, Amílcar, Igreja, Bruno, Wright, Lyndon, Soares-da-Silva, Patricio
Published in Current medical research and opinion (01.05.2010)
Published in Current medical research and opinion (01.05.2010)
Get more information
Journal Article
Plasma Protein Binding of Highly Bound Drugs Determined With Equilibrium Gel Filtration of Nonradiolabeled Compounds and LC-MS/MS Detection
Isbell, John, Yuan, Ding, Torrao, Leonel, Gatlik, Ewa, Hoffmann, Laurent, Wipfli, Peter
Published in Journal of pharmaceutical sciences (01.02.2019)
Published in Journal of pharmaceutical sciences (01.02.2019)
Get full text
Journal Article
Pharmacokinetic-Pharmacodynamic Interaction between Nebicapone, a Novel Catechol-O-Methyltransferase Inhibitor, and Controlled-Release Levodopa/Carbidopa 200 mg/50 mg: Randomized, Double-Blind, Placebo-Controlled, Crossover Study in Healthy Subjects
Vaz-da-Silva, Manuel, Loureiro, Ana I., Nunes, Teresa, Lopes, Carlos, Rocha, José, Machado, Rita, Costa, Raquel, Torrão, Leonel, Falcão, Amílcar, Wright, Lyndon, Almeida, Luis, Soares-da-Silva, Patrício
Published in Drugs in R&D (01.01.2008)
Published in Drugs in R&D (01.01.2008)
Get full text
Journal Article
Pharmacokinetic—pharmacodynamic interaction between nebicapone and controlled-release levodopa/benserazide: A single-center, phase I, double-blind, randomized, placebo-controlled, four-way crossover study in healthy subjects
Nunes, Teresa, MD, Machado, Rita, MSc, Rocha, José F., BSc, Fernandes-Lopes, Carlos, BSc, Costa, Raquel, PharmD, Torrão, Leonel, MSc, Loureiro, Ana I., MSc, Falcão, Amílcar, PharmD, PhD, Vaz-da-Silva, Manuel, MD, PhD, Wright, Lyndon, PhD, Almeida, Luis, MD, PhD, Soares-da-Silva, Patricio, MD, PhD
Published in Clinical therapeutics (01.10.2009)
Published in Clinical therapeutics (01.10.2009)
Get full text
Journal Article
Pharmacokinetic-pharmacodynamic interaction between BIA 3-202, a novel COMT inhibitor, and levodopa/benserazide
SILVEIRA, Pedro, VAZ-DA-SILVA, Manuel, ALMEIDA, Luis, MAIA, Joana, FALCAO, Amilcar, LOUREIRO, Ana, TORRAO, Leonel, MACHADO, Rita, WRIGHT, Lyndon, SOARES-DA-SILVA, Patricio
Published in European journal of clinical pharmacology (01.11.2003)
Published in European journal of clinical pharmacology (01.11.2003)
Get full text
Journal Article
Programmed cell death induces male sterility in Actinidia deliciosa female flowers
Coimbra, Sílvia, Torrão, Leonel, Abreu, Ilda
Published in Plant physiology and biochemistry (01.06.2004)
Published in Plant physiology and biochemistry (01.06.2004)
Get full text
Journal Article
Pharmacokinetic--pharmacodynamic interaction between nebicapone and controlled-release levodopa/benserazide: A single-center, phase I, double-blind, randomized, placebo-controlled, four-way crossover study in healthy subjects: Original research
Nunes, Teresa, Machado, Rita, Rocha, José F, Fernandes-Lopes, Carlos, Costa, Raquel, Torrão, Leonel, Loureiro, Ana I, Falcão, Amílcar, Vaz-da-Silva, Manuel, Wright, Lyndon, Almeida, Luis, Soares-da-Silva, Patricio
Published in Clinical therapeutics (01.10.2009)
Published in Clinical therapeutics (01.10.2009)
Get full text
Journal Article
Poster Abstract #7: Pharmacokinetic-Pharmacodynamic Interaction Between Nebicapone (BIA 3-202) and Controlled-release Levodopa/Benserazide (Madopar HBS 125)
Almeida, Luis, Rocha, Jose Francisco, Lopes, Carlos, Nunes, Teresa, Machado, Rita, Costa, Raquel, Torrão, Leonel, Loureiro, Ana-Isabel, Vaz-da-Silva, Manuel, Wright, Lyndon, Soares-da-Silva, Patricio, Falcão, Amilcar
Published in Neurotherapeutics (01.07.2008)
Published in Neurotherapeutics (01.07.2008)
Get full text
Journal Article
Pharmacokinetic-pharmacodynamic interaction between BIA 3-202, a novel COMT inhibitor, and levodopa/carbidopa
Almeida, Luis, Vaz-da-Silva, Manuel, Silveira, Pedro, Falcão, Amilcar, Maia, Joana, Loureiro, Ana, Torrão, Leonel, Machado, Rita, Wright, Lyndon, Soares-da-Silva, Patrício
Published in Clinical neuropharmacology (01.01.2004)
Published in Clinical neuropharmacology (01.01.2004)
Get more information
Journal Article