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Therapeutic Targeting of the Soluble Guanylate Cyclase
Makrynitsa, Garyfallia I, Zompra, Aikaterini A, Argyriou, Aikaterini I, Spyroulias, Georgios A, Topouzis, Stavros
Published in Current medicinal chemistry (01.01.2019)
Published in Current medicinal chemistry (01.01.2019)
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Thioglycine and l-thiovaline: Biologically active H2S-donors
Zhou, Zongmin, von Wantoch Rekowski, Margarete, Coletta, Ciro, Szabo, Csaba, Bucci, Mariarosaria, Cirino, Giuseppe, Topouzis, Stavros, Papapetropoulos, Andreas, Giannis, Athanassios
Published in Bioorganic & medicinal chemistry (15.04.2012)
Published in Bioorganic & medicinal chemistry (15.04.2012)
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Design, synthesis and biological evaluation of new 3,4-dihydroquinoxalin-2(1H)-one derivatives as soluble guanylyl cyclase (sGC) activators
Kintos, Dionysios-Panagiotis, Salagiannis, Konstantinos, Vazoura, Vasiliki, Wittrien, Theresa, Papakyriakou, Athanasios, Nikolaropoulos, Sotiris S., Behrends, Soenke, Topouzis, Stavros, Fousteris, Manolis A.
Published in Heliyon (01.11.2022)
Published in Heliyon (01.11.2022)
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Mapping of the sGC Stimulator BAY 41-2272 Binding Site on H-NOX Domain and Its Regulation by the Redox State of the Heme
Makrynitsa, Garyfallia I., Argyriou, Aikaterini I., Zompra, Aikaterini A., Salagiannis, Konstantinos, Vazoura, Vassiliki, Papapetropoulos, Andreas, Topouzis, Stavros, Spyroulias, Georgios A.
Published in Frontiers in cell and developmental biology (17.06.2022)
Published in Frontiers in cell and developmental biology (17.06.2022)
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Replacement of heme by soluble guanylate cyclase (sGC) activators abolishes heme-nitric oxide/oxygen (H-NOX) domain structural plasticity
Argyriou, Aikaterini I., Makrynitsa, Garyfallia I., Dalkas, Georgios, Georgopoulou, Dimitra A., Salagiannis, Konstantinos, Vazoura, Vassiliki, Papapetropoulos, Andreas, Topouzis, Stavros, Spyroulias, Georgios A.
Published in Current research in structural biology (01.01.2021)
Published in Current research in structural biology (01.01.2021)
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PDGF-DD, a novel mediator of smooth muscle cell phenotypic modulation, is upregulated in endothelial cells exposed to atherosclerosis-prone flow patterns
Thomas, James A, Deaton, Rebecca A, Hastings, Nicole E, Shang, Yueting, Moehle, Christopher W, Eriksson, Ulf, Topouzis, Stavros, Wamhoff, Brian R, Blackman, Brett R, Owens, Gary K
Published in American journal of physiology. Heart and circulatory physiology (01.02.2009)
Published in American journal of physiology. Heart and circulatory physiology (01.02.2009)
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Ascertainment and critical assessment of the views of the general public and healthcare professionals on nutrigenomics in Greece
Pavlidis, Cristiana, Karamitri, Angeliki, Barakou, Aglaia, Cooper, David N, Poulas, Konstantinos, Topouzis, Stavros, Patrinos, George P
Published in Personalized medicine (01.03.2012)
Published in Personalized medicine (01.03.2012)
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Comparison of the effects of e-cigarette vapor with cigarette smoke on lung function and inflammation in mice
Glynos, Constantinos, Bibli, Sofia-Iris, Katsaounou, Paraskevi, Pavlidou, Athanasia, Magkou, Christina, Karavana, Vassiliki, Topouzis, Stavros, Kalomenidis, Ioannis, Zakynthinos, Spyros, Papapetropoulos, Andreas
Published in American journal of physiology. Lung cellular and molecular physiology (01.11.2018)
Published in American journal of physiology. Lung cellular and molecular physiology (01.11.2018)
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Platelet-derived growth factor-D expression in developing and mature human kidneys
Changsirikulchai, Siribha, Hudkins, Kelly L., Goodpaster, Tracy A., Volpone, John, Topouzis, Stavros, Gilbertson, Debra G., Alpers, Charles E.
Published in Kidney international (01.12.2002)
Published in Kidney international (01.12.2002)
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Extending the translational potential of targeting NO/cGMP‐regulated pathways in the CVS
Papapetropoulos, Andreas, Hobbs, Adrian J, Topouzis, Stavros
Published in British journal of pharmacology (01.03.2015)
Published in British journal of pharmacology (01.03.2015)
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Identification of new multi-substituted 1H-pyrazolo3,4-cpyridin-7(6H)-ones as soluble guanylyl cyclase (sGC) stimulators with vasoprotective and anti-inflammatory activities
Kintos, Dionysios-Panagiotis, Salagiannis, Konstantinos, Sgouros, Antonis, Nikolaropoulos, Sotiris S, Topouzis, Stavros, Fousteris, Manolis A
Published in Bioorganic chemistry (01.03.2024)
Published in Bioorganic chemistry (01.03.2024)
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BRF110, an Orally Active Nurr1-RXRα-Selective Rexinoid, Enhances BDNF Expression without Elevating Triglycerides
Asvos, Xenophon, El Mubarak, Mohamed A., Karampelas, Theodoros, Rampias, Theodoros, Tamvakopoulos, Constantin, Sivolapenko, Gregory B., Papakyriakou, Athanasios, Topouzis, Stavros, Vassilatis, Demetrios K., Fokas, Demosthenes
Published in Journal of medicinal chemistry (27.02.2025)
Published in Journal of medicinal chemistry (27.02.2025)
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Novel drugs approved by the EMA, the FDA and the MHRA in 2024: A year in review
Topouzis, Stavros, Papapetropoulos, Andreas, Alexander, Steve P. H., Cortese‐Krott, Miriam, Kendall, Dave A., Martemyanov, Kirill, Mauro, Claudio, Nagercoil, Nithyanandan, Panettieri, Reynold A., Patel, Hemal H., Schulz, Rainer, Stefanska, Barbara, Stephens, Gary J., Teixeira, Mauro M., Vergnolle, Nathalie, Wang, Xin, Ferdinandy, Péter
Published in British journal of pharmacology (01.04.2025)
Published in British journal of pharmacology (01.04.2025)
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Nurr1: RXRα heterodimer activation as monotherapy for Parkinson’s disease
Spathis, Athanasios D., Asvos, Xenophon, Ziavra, Despina, Karampelas, Theodoros, Topouzis, Stavros, Cournia, Zoe, Qing, Xiaobing, Alexakos, Pavlos, Smits, Lisa M., Dalla, Christina, Rideout, Hardy J., Schwamborn, Jens Christian, Tamvakopoulos, Constantin, Fokas, Demosthenes, Vassilatis, Demetrios K.
Published in Proceedings of the National Academy of Sciences - PNAS (11.04.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (11.04.2017)
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Novel drugs approved by the EMA, the FDA, and the MHRA in 2023: A year in review
Papapetropoulos, Andreas, Topouzis, Stavros, Alexander, Steve P. H., Cortese‐Krott, Miriam, Kendall, Dave A., Martemyanov, Kirill A., Mauro, Claudio, Nagercoil, Nithyanandan, Panettieri, Reynold A., Patel, Hemal H., Schulz, Rainer, Stefanska, Barbara, Stephens, Gary J., Teixeira, Mauro M., Vergnolle, Nathalie, Wang, Xin, Ferdinandy, Péter
Published in British journal of pharmacology (01.06.2024)
Published in British journal of pharmacology (01.06.2024)
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Identification of new multi-substituted 1H-pyrazolo[3,4-c]pyridin-7(6H)-ones as soluble guanylyl cyclase (sGC) stimulators with vasoprotective and anti-inflammatory activities
Kintos, Dionysios-Panagiotis, Salagiannis, Konstantinos, Sgouros, Antonis, Nikolaropoulos, Sotiris S., Topouzis, Stavros, Fousteris, Manolis A.
Published in Bioorganic chemistry (01.03.2024)
Published in Bioorganic chemistry (01.03.2024)
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Role of cGMP in hydrogen sulfide signaling
Bibli, Sofia-Iris, Yang, Guangdong, Zhou, Zongmin, Wang, Rui, Topouzis, Stavros, Papapetropoulos, Andreas
Published in Nitric oxide (30.04.2015)
Published in Nitric oxide (30.04.2015)
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