Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors
Chino, Ayaka, Seo, Ryushi, Amano, Yasushi, Namatame, Ichiji, Hamaguchi, Wataru, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki, Masuda, Naoyuki
Published in Chemical & pharmaceutical bulletin (2018)
Published in Chemical & pharmaceutical bulletin (2018)
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Journal Article
In Vitro Activities of a New Lipopeptide Antifungal Agent, FK463, against a Variety of Clinically Important Fungi
TAWARA, S, IKEDA, F, KAWABATA, K, TAKASUGI, H, SAKANE, K, TANAKA, H, MATSUMOTO, F, KUWAHARA, S, MAKI, K, MORISHITA, Y, OTOMO, K, TERATANI, N, GOTO, T, TOMISHIMA, M, OHKI, H, YAMADA, A
Published in Antimicrobial Agents and Chemotherapy (01.01.2000)
Published in Antimicrobial Agents and Chemotherapy (01.01.2000)
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Journal Article
Use of a serum-based antifungal susceptibility assay to predict the in vivo efficacy of novel echinocandin compounds
Maki, Katsuyuki, Matsumoto, Satoru, Watabe, Etsuko, Iguchi, Yumi, Tomishima, Masaki, Ohki, Hidenori, Yamada, Akira, Ikeda, Fumiaki, Tawara, Shuichi, Mutoh, Seitaro
Published in Microbiology and immunology (01.08.2008)
Published in Microbiology and immunology (01.08.2008)
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Determination of antifungal activities in serum samples from mice treated with different antifungal drugs allows detection of an active metabolite of itraconazole
Maki, Katsuyuki, Watabe, Etsuko, Iguchi, Yumi, Nakamura, Hideko, Tomishima, Masaki, Ohki, Hidenori, Yamada, Akira, Matsumoto, Satoru, Ikeda, Fumiaki, Tawara, Shuichi, Mutoh, Seitaro
Published in Microbiology and immunology (2006)
Published in Microbiology and immunology (2006)
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Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability
Chino, Ayaka, Masuda, Naoyuki, Amano, Yasushi, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki
Published in Bioorganic & medicinal chemistry (01.07.2014)
Published in Bioorganic & medicinal chemistry (01.07.2014)
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Journal Article
Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors
Chino, Ayaka, Honda, Shugo, Morita, Masataka, Yonezawa, Koichi, Hamaguchi, Wataru, Amano, Yasushi, Moriguchi, Hiroyuki, Yamazaki, Mayako, Aota, Masaki, Tomishima, Masaki, Masuda, Naoyuki
Published in Bioorganic & medicinal chemistry (15.08.2019)
Published in Bioorganic & medicinal chemistry (15.08.2019)
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Journal Article
Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors
Ayaka Chino, Ryushi Seo, Yasushi Amano, Ichiji Namatame, Wataru Hamaguchi, Kazuya Honbou, Takuma Mihara, Mayako Yamazaki, Masaki Tomishima, Naoyuki Masuda
Published in Chemical and Pharmaceutical Bulletin (01.03.2018)
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Published in Chemical and Pharmaceutical Bulletin (01.03.2018)
Journal Article
Synthesis and antifungal activity of ASP9726, a novel echinocandin with potent Aspergillus hyphal growth inhibition
Morikawa, Hiroshi, Tomishima, Masaki, Kayakiri, Natsuko, Araki, Takanobu, Barrett, David, Akamatsu, Souichirou, Matsumoto, Satoru, Uchida, Satoko, Nakai, Toru, Takeda, Shinobu, Maki, Katsuyuki
Published in Bioorganic & medicinal chemistry letters (15.02.2014)
Published in Bioorganic & medicinal chemistry letters (15.02.2014)
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Journal Article
FR290581, a novel sordarin derivative: Synthesis and antifungal activity
Hanadate, Tadaatsu, Tomishima, Masaki, Shiraishi, Nobuyuki, Tanabe, Daisuke, Morikawa, Hiroshi, Barrett, David, Matsumoto, Satoru, Ohtomo, Kazumi, Maki, Katsuyuki
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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Journal Article
Synthesis and evaluation of nitro 5-deazaflavins as novel bioreductive antitumor agents
Kawamoto, Tetsuji, Ikeuchi, Yoshihiro, Hiraki, Junko, Eikyu, Yoshiteru, Shimizu, Kazue, Tomishima, Masaki, Bessho, Kiyoshi, Yoneda, Fumio, Mikata, Yuji, Nishida, Mamiko, Ikehara, Kenji, Sasaki, Takuma
Published in Bioorganic & medicinal chemistry letters (21.09.1995)
Published in Bioorganic & medicinal chemistry letters (21.09.1995)
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Journal Article
POLYPEPTIDE COMPOUND
TOJO, TAKASHI, ARAKI, TAKANOBU, HARAYAMA, YU, TANABE, DAISUKE, NAGAI, YASUHITO, TOMISHIMA, MASAKI, KAYAKIRI, NATSUKO, MAKINO, TAKUYA
Year of Publication 30.08.2012
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Year of Publication 30.08.2012
Patent
POLYPEPTIDE COMPOUND
TOJO, TAKASHI, ARAKI, TAKANOBU, HARAYAMA, YU, TANABE, DAISUKE, NAGAI, YASUHITO, TOMISHIMA, MASAKI, KAYAKIRI, NATSUKO, MAKINO, TAKUYA
Year of Publication 30.08.2012
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Year of Publication 30.08.2012
Patent
POLYPEPTIDE COMPOUND
MORIKAWA HIROSHI, TOMISHIMA MASAKI, KAYAKIRI NATSUKO, ARAKI TAKANOBU, MAKINO TAKUYA, IMANISHI MASASHI, NAKAGAWA TOSHIYA, ASANO TORU
Year of Publication 05.07.2010
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Year of Publication 05.07.2010
Patent
POLYPEPTIDE COMPOUND
IMANISHI, MASASHI, ARAKI, TAKANOBU, MORIKAWA, HIROSHI, NAKAGAWA, TOSHIYA, ASANO, TORU, TOMISHIMA, MASAKI, MAKINO, TAKUYA, KAYAKIRI, NATSUKO
Year of Publication 07.05.2009
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Year of Publication 07.05.2009
Patent
Atropisomeric Flavoenzyme Models with a Modified Pyrimidine Ring: Syntheses, Physical Properties, and Stereochemistry in the Reactions with NAD(P)H Analogs
Ohno, Atsuyoshi, Kunitomo, Jun, Kawai, Yasushi, Kawamoto, Tetsuji, Tomishima, Masaki, Yoneda, Fumio
Published in Journal of organic chemistry (27.12.1996)
Published in Journal of organic chemistry (27.12.1996)
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Journal Article
NOVEL AMIDE COMPOUNDS
SPEARS, GLEN, W, IMANISHI, MASASHI, ITO, KIYOTAKA, TAKAHASHI, FUMIE, HAYASHIDA, HISASHI, TOMISHIMA, MASAKI, MIYAKE, HIROSHI, YAMADA, AKIRA
Year of Publication 20.09.2001
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Year of Publication 20.09.2001
Patent