Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors
Mollica, Adriano, Pelliccia, Sveva, Famiglini, Valeria, Stefanucci, Azzurra, Macedonio, Giorgia, Chiavaroli, Annalisa, Orlando, Giustino, Brunetti, Luigi, Ferrante, Claudio, Pieretti, Stefano, Novellino, Ettore, Benyhe, Sandor, Zador, Ferenc, Erdei, Anna, Szucs, Edina, Samavati, Reza, Dvorácskó, Szabolcs, Tomboly, Csaba, Ragno, Rino, Patsilinakos, Alexandros, Silvestri, Romano
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
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Endomorphins interact with the substance P (SP) aminoterminal SP1-7 binding in the ventral tegmental area of the rat brain
BOBOS, Milad, JOHANSSON, Tobias, QIN ZHOU, LINDEBERG, Gunnar, TOMBOLY, Csaba, TOTH, Géza, LE GREVES, Pierre, NYBERG, Fred, HALLBERG, Mathias
Published in Peptides (New York, N.Y. : 1980) (01.10.2008)
Published in Peptides (New York, N.Y. : 1980) (01.10.2008)
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Pro-Inflammatory Cytokines: Potential Links between the Endocannabinoid System and the Kynurenine Pathway in Depression
Zádor, Ferenc, Joca, Sâmia, Nagy-Grócz, Gábor, Dvorácskó, Szabolcs, Szűcs, Edina, Tömböly, Csaba, Benyhe, Sándor, Vécsei, László
Published in International journal of molecular sciences (31.05.2021)
Published in International journal of molecular sciences (31.05.2021)
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Journal Article
Rimonabant-Based Compounds Bearing Hydrophobic Amino Acid Derivatives as Cannabinoid Receptor Subtype 1 Ligands
Dvorácskó, Szabolcs, Dimmito, Marilisa Pia, Sebastiani, Jessica, La Regina, Giuseppe, Silvestri, Romano, Pieretti, Stefano, Stefanucci, Azzurra, Tömböly, Csaba, Mollica, Adriano
Published in ACS medicinal chemistry letters (13.04.2023)
Published in ACS medicinal chemistry letters (13.04.2023)
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Journal Article
Novel Fubinaca/Rimonabant hybrids as endocannabinoid system modulators
Stefanucci, Azzurra, Macedonio, Giorgia, Dvorácskó, Szabolcs, Tömböly, Csaba, Mollica, Adriano
Published in Amino acids (01.11.2018)
Published in Amino acids (01.11.2018)
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Journal Article
Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors
Dvorácskó, Szabolcs, Keresztes, Attila, Mollica, Adriano, Stefanucci, Azzurra, Macedonio, Giorgia, Pieretti, Stefano, Zádor, Ferenc, Walter, Fruzsina R., Deli, Mária A., Kékesi, Gabriella, Bánki, László, Tuboly, Gábor, Horváth, Gyöngyi, Tömböly, Csaba
Published in European journal of medicinal chemistry (15.09.2019)
Published in European journal of medicinal chemistry (15.09.2019)
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Journal Article
Kynurenines and the Endocannabinoid System in Schizophrenia: Common Points and Potential Interactions
Zádor, Ferenc, Nagy-Grócz, Gábor, Kekesi, Gabriella, Dvorácskó, Szabolcs, Szűcs, Edina, Tömböly, Csaba, Horvath, Gyongyi, Benyhe, Sándor, Vécsei, László
Published in Molecules (Basel, Switzerland) (15.10.2019)
Published in Molecules (Basel, Switzerland) (15.10.2019)
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Journal Article
Novel High Affinity Sigma-1 Receptor Ligands from Minimal Ensemble Docking-Based Virtual Screening
Dvorácskó, Szabolcs, Lázár, László, Fülöp, Ferenc, Palkó, Márta, Zalán, Zita, Penke, Botond, Fülöp, Lívia, Tömböly, Csaba, Bogár, Ferenc
Published in International journal of molecular sciences (29.07.2021)
Published in International journal of molecular sciences (29.07.2021)
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Journal Article
Lessons on the Sigma-1 Receptor in TNBS-Induced Rat Colitis: Modulation of the UCHL-1, IL-6 Pathway
Almási, Nikoletta, Török, Szilvia, Dvorácskó, Szabolcs, Tömböly, Csaba, Csonka, Ákos, Baráth, Zoltán, Murlasits, Zsolt, Valkusz, Zsuzsanna, Pósa, Anikó, Varga, Csaba, Kupai, Krisztina
Published in International journal of molecular sciences (05.06.2020)
Published in International journal of molecular sciences (05.06.2020)
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Journal Article
Selective antiproliferative effect of C-2 halogenated 13α-estrones on cells expressing Organic anion-transporting polypeptide 2B1 (OATP2B1)
Laczkó-Rigó, Réka, Bakos, Éva, Jójárt, Rebeka, Tömböly, Csaba, Mernyák, Erzsébet, Özvegy-Laczka, Csilla
Published in Toxicology and applied pharmacology (15.10.2021)
Published in Toxicology and applied pharmacology (15.10.2021)
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Journal Article
N,N-Dimethyltryptamine attenuates spreading depolarization and restrains neurodegeneration by sigma-1 receptor activation in the ischemic rat brain
Szabó, Írisz, Varga, Viktória É., Dvorácskó, Szabolcs, Farkas, Attila E., Körmöczi, Tímea, Berkecz, Róbert, Kecskés, Szilvia, Menyhárt, Ákos, Frank, Rita, Hantosi, Dóra, Cozzi, Nicholas V., Frecska, Ede, Tömböly, Csaba, Krizbai, István A., Bari, Ferenc, Farkas, Eszter
Published in Neuropharmacology (01.07.2021)
Published in Neuropharmacology (01.07.2021)
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Journal Article
Focusing on the 5F-MDMB-PICA, 4F-MDMB-BICA synthetic cannabinoids and their primary metabolites in analytical and pharmacological aspects
Dvorácskó, Szabolcs, Körmöczi, Tímea, Sija, Éva, Bende, Balázs, Weiczner, Roland, Varga, Tibor, Ilisz, István, Institóris, László, Kereszty, Éva M., Tömböly, Csaba, Berkecz, Róbert
Published in Toxicology and applied pharmacology (01.07.2023)
Published in Toxicology and applied pharmacology (01.07.2023)
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Journal Article
Decreased CB receptor binding and cannabinoid signaling in three brain regions of a rat model of schizophrenia
Szűcs, Edina, Dvorácskó, Szabolcs, Tömböly, Csaba, Büki, Alexandra, Kékesi, Gabriella, Horváth, Gyöngyi, Benyhe, Sándor
Published in Neuroscience letters (28.10.2016)
Published in Neuroscience letters (28.10.2016)
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Journal Article
Interactions between the Kynurenine and the Endocannabinoid System with Special Emphasis on Migraine
Nagy-Grócz, Gábor, Zádor, Ferenc, Dvorácskó, Szabolcs, Bohár, Zsuzsanna, Benyhe, Sándor, Tömböly, Csaba, Párdutz, Árpád, Vécsei, László
Published in International journal of molecular sciences (30.07.2017)
Published in International journal of molecular sciences (30.07.2017)
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Journal Article
Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity
Dimmito, Marilisa P, Stefanucci, Azzurra, Pieretti, Stefano, Minosi, Paola, Dvorácskó, Szabolcs, Tömböly, Csaba, Zengin, Gokhan, Mollica, Adriano
Published in Biomolecules (Basel, Switzerland) (16.09.2019)
Published in Biomolecules (Basel, Switzerland) (16.09.2019)
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Journal Article
Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration
Perlikowska, Renata, Piekielna, Justyna, Gentilucci, Luca, De Marco, Rossella, Cerlesi, Maria Camilla, Calo, Girolamo, Artali, Roberto, Tömböly, Csaba, Kluczyk, Alicja, Janecka, Anna
Published in European journal of medicinal chemistry (15.02.2016)
Published in European journal of medicinal chemistry (15.02.2016)
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Journal Article
Synthesis and in Vitro Evaluation of Stabilized and Selective Neuromedin U‑1 Receptor Agonists
De Prins, An, Martin, Charlotte, Van Wanseele, Yannick, Tömböly, Csaba, Tourwé, Dirk, Caveliers, Vicky, Holst, Birgitte, Van Eeckhaut, Ann, Rosenkilde, Mette M, Smolders, Ilse, Ballet, Steven
Published in ACS medicinal chemistry letters (10.05.2018)
Published in ACS medicinal chemistry letters (10.05.2018)
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Journal Article
Investigation of receptor binding and functional characteristics of hemopressin(1–7)
Dvorácskó, Szabolcs, Tömböly, Csaba, Berkecz, Róbert, Keresztes, Attila
Published in Neuropeptides (Edinburgh) (01.08.2016)
Published in Neuropeptides (Edinburgh) (01.08.2016)
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Journal Article
Synthesis and structure-activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis
Bacsa, Ildikó, Herman, Bianka Edina, Jójárt, Rebeka, Herman, Kevin Stefán, Wölfling, János, Schneider, Gyula, Varga, Mónika, Tömböly, Csaba, Rižner, Tea Lanišnik, Szécsi, Mihály, Mernyák, Erzsébet
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
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Journal Article
Effects of RVD-hemopressin (α) on feeding and body weight after standard or cafeteria diet in rats
Leone, Sheila, Ferrante, Claudio, Recinella, Lucia, Chiavaroli, Annalisa, Mollica, Adriano, Tömböly, Csaba, Stefanucci, Azzurra, Dimmito, Marilisa Pia, Dvorácskó, Szabolcs, Verratti, Vittore, De Petrocellis, Luciano, Orlando, Giustino, Brunetti, Luigi
Published in Neuropeptides (Edinburgh) (01.12.2018)
Published in Neuropeptides (Edinburgh) (01.12.2018)
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