KGA-2727, a novel selective inhibitor of a high-affinity sodium glucose cotransporter (SGLT1), exhibits antidiabetic efficacy in rodent models
Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Fushimi, Nobuhiko, Itoh, Fumiaki, Yamada, Mitsuhiko, Isaji, Masayuki
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Published in The Journal of pharmacology and experimental therapeutics (01.08.2012)
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SLC5A9/SGLT4, a new Na +-dependent glucose transporter, is an essential transporter for mannose, 1,5-anhydro-D-glucitol, and fructose
Tazawa, Shigeki, Yamato, Tokuhisa, Fujikura, Hideki, Hiratochi, Masahiro, Itoh, Fumiaki, Tomae, Masaki, Takemura, Yukiko, Maruyama, Hidetoshi, Sugiyama, Tomoyasu, Wakamatsu, Ai, Isogai, Takao, Isaji, Masayuki
Published in Life sciences (1973) (14.01.2005)
Published in Life sciences (1973) (14.01.2005)
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Structure–activity relationship studies of 4-benzyl-1H-pyrazol-3-yl β-d-glucopyranoside derivatives as potent and selective sodium glucose co-transporter 1 (SGLT1) inhibitors with therapeutic activity on postprandial hyperglycemia
Fushimi, Nobuhiko, Fujikura, Hideki, Shiohara, Hiroaki, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Ozawa, Tomonaga, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (15.11.2012)
Published in Bioorganic & medicinal chemistry (15.11.2012)
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Design, synthesis, and structure–activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl β-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)
Fushimi, Nobuhiko, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Yamauchi, Yuji, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.02.2013)
Published in Bioorganic & medicinal chemistry (01.02.2013)
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Design, synthesis, and structure-activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl I2-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)
Fushimi, Nobuhiko, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Yamauchi, Yuji, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.02.2013)
Published in Bioorganic & medicinal chemistry (01.02.2013)
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Design, synthesis, and structure-activity relationships of a series of 4-benzyl-5-isopropyl-1H-pyrazol-3-yl [beta]-d-glycopyranosides substituted with novel hydrophilic groups as highly potent inhibitors of sodium glucose co-transporter 1 (SGLT1)
Fushimi, Nobuhiko, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Yamauchi, Yuji, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.02.2013)
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Published in Bioorganic & medicinal chemistry (01.02.2013)
Journal Article
Structure-activity relationship studies of 4-benzyl-1H-pyrazol-3-yl I2-d-glucopyranoside derivatives as potent and selective sodium glucose co-transporter 1 (SGLT1) inhibitors with therapeutic activity on postprandial hyperglycemia
Fushimi, Nobuhiko, Fujikura, Hideki, Shiohara, Hiroaki, Teranishi, Hirotaka, Shimizu, Kazuo, Yonekubo, Shigeru, Ohno, Kohsuke, Miyagi, Takashi, Itoh, Fumiaki, Shibazaki, Toshihide, Tomae, Masaki, Ishikawa-Takemura, Yukiko, Nakabayashi, Takeshi, Kamada, Noboru, Ozawa, Tomonaga, Kobayashi, Susumu, Isaji, Masayuki
Published in Bioorganic & medicinal chemistry (01.11.2012)
Published in Bioorganic & medicinal chemistry (01.11.2012)
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Corrigendum to “SLC5A9/SGLT4, a new Na+-dependent glucose transporter, is an essential transporter for mannose, 1,5-anhydro- d-glucitol, and fructose” [Life Sciences 76 (2005) 1039–1050]
Tazawa, Shigeki, Yamato, Tokuhisa, Fujikura, Hideki, Hiratochi, Masahiro, Itoh, Fumiaki, Tomae, Masaki, Takemura, Yukiko, Maruyama, Hidetoshi, Sugiyama, Tomoyasu, Wakamatsu, Ai, Isogai, Takao, Isaji, Masayuki
Published in Life sciences (1973) (09.10.2010)
Published in Life sciences (1973) (09.10.2010)
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PREVENTIVE OR REMEDY FOR DISEASES CAUSED BY HYPERGLYCEMIA
TOMAE, MASAKI, FUSHIMI, NOBUHIKO, ITO, FUMIAKI, SHIBAZAKI, TOSHIHIDE, ISAJI, MASAYUKI
Year of Publication 17.06.2004
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Year of Publication 17.06.2004
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