Modulation of plasma protein binding and in vivo liver cell uptake of phosphorothioate oligodeoxynucleotides by cholesterol conjugation
Bijsterbosch, M K, Rump, E T, De Vrueh, R L, Dorland, R, van Veghel, R, Tivel, K L, Biessen, E A, van Berkel, T J, Manoharan, M
Published in Nucleic acids research (15.07.2000)
Published in Nucleic acids research (15.07.2000)
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Base-Sequence Dependence of Emission Lifetimes for D141018-30-6NA Oligomers and Duplexes Covalently Labeled with Pyrene: Relative Electron-Transfer Quenching Efficiencies of A, G, C, and T Nucleosides toward Pyrene
Manoharan, Muthiah, Tivel, Kathleen L, Zhao, Min, Nafisi, Kambiz, Netzel, Thomas L
Published in Journal of physical chemistry (1952) (01.11.1995)
Published in Journal of physical chemistry (1952) (01.11.1995)
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In vivo fate of phosphorothioate antisense oligodeoxynucleotides: predominant uptake by scavenger receptors on endothelial liver cells
Bijsterbosch, Martin K., Manoharan, Muthiah, Rump, Erik T., De Vrueh, Remco L. A., van Veghel, Richard, Tivel, Kathleen L., Biessen, Erik A. L., Bennett, C. Frank, Cook, P. Dan, van Berkel, Theo J. C.
Published in Nucleic acids research (15.08.1997)
Published in Nucleic acids research (15.08.1997)
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Pharmacokinetic properties of several novel oligonucleotide analogs in mice
Crooke, S T, Graham, M J, Zuckerman, J E, Brooks, D, Conklin, B S, Cummins, L L, Greig, M J, Guinosso, C J, Kornbrust, D, Manoharan, M, Sasmor, H M, Schleich, T, Tivel, K L, Griffey, R H
Published in The Journal of pharmacology and experimental therapeutics (01.05.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.1996)
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2′- and 3′- Cholesterol-Conjugated Adenosine and Cytosine Nucleoside Building Blocks: Synthesis of Lipidic Nucleic Acids
Manoharan, Muthiah, Inamati, Gopal, Tivel, Kathleen L., Conklin, Boyd, Ross, Bruce S., Cook, P. Dan
Published in Nucleosides & nucleotides (01.07.1997)
Published in Nucleosides & nucleotides (01.07.1997)
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Cholesterol Conjugated Uniform and Gapmer Phosphorothioate Oligonucleotides Targeted Against PKC-α and C-raf Gene Expression
Manoharan, Muthiah, Tivel, Kathleen L., Inamati, Gopal, Monia, Brett P., Dean, Nick, Cook, P. Dan
Published in Nucleosides & nucleotides (01.07.1997)
Published in Nucleosides & nucleotides (01.07.1997)
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Conjugated Antisense Oligonucleotides
Manoharan, Muthiah, Tivel, Kathleen L., Condon, Thomas P., Andrade, Laura K., Barber-Peoch, Isabelle, Inamati, Gopal, Shah, Shefali, Mohan, Venkatraman, Graham, Mark J., Bennett, C. Frank, Crooke, Stanley T., Cook, P. Dan
Published in Nucleosides & nucleotides (01.07.1997)
Published in Nucleosides & nucleotides (01.07.1997)
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Modification of a Phosphorothioate Oligonucleotide with Cholesterol Induces Association of the Oligonucleotide to Serum Lipoproteins and Affects Its Biological Fate
Bijsterbosch, Martin K., Manoharan, Muthiah, Tivel, Kathleen L., Rump, Erik T., Biessen, Erik A.L., De Vrueh, Remco L.A., Cook, P. Dan, van Berkel, Theo J.C.
Published in Nucleosides & nucleotides (01.07.1997)
Published in Nucleosides & nucleotides (01.07.1997)
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