Enzymatic Characterization of c-Met Receptor Tyrosine Kinase Oncogenic Mutants and Kinetic Studies with Aminopyridine and Triazolopyrazine Inhibitors
Timofeevski, Sergei L, McTigue, Michele A, Ryan, Kevin, Cui, Jean, Zou, Helen Y, Zhu, Jeff X, Chau, Fannie, Alton, Gordon, Karlicek, Shannon, Christensen, James G, Murray, Brion W
Published in Biochemistry (Easton) (16.06.2009)
Published in Biochemistry (Easton) (16.06.2009)
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Synthesis and SAR of 4-substituted-2-aminopyrimidines as novel c-Jun N-terminal kinase (JNK) inhibitors
Humphries, Paul S., Lafontaine, Jennifer A., Agree, Charles S., Alexander, David, Chen, Ping, Do, Quyen-Quyen T., Li, Lilian Y., Lunney, Elizabeth A., Rajapakse, Ranjan J., Siegel, Karen, Timofeevski, Sergei L., Wang, Tianlun, Wilhite, David M.
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
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Isoform-Selective Interaction of Cyclooxygenase-2 with Indomethacin Amides Studied by Real-Time Fluorescence, Inhibition Kinetics, and Site-Directed Mutagenesis
Timofeevski, Sergei L, Prusakiewicz, Jeffery J, Rouzer, Carol A, Marnett, Lawrence J
Published in Biochemistry (Easton) (30.07.2002)
Published in Biochemistry (Easton) (30.07.2002)
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Abstract 5903: MASTL small-molecule inhibition to target mitosis for cancer therapy
Toledo, Chad M., Eisele, Koleen J., Kim, Dong Hyun, Mu, Xinmeng, Brun, Sonja, Davis, Carl, Greenwald, Eric C., Hui, Fion, He, Meilan, Yang, Yanling, Flores-Bojorquez, Ana, Li, Yuxin, Khamphavong, Penney L., Lee, Joseph H., Li, Jian, Ramms, Dana J., Jones, Greg, Auth, Marin, Painter, Cory L., Nager, Andrew, Oyer, Jon, Timofeevski, Sergei L., Pierceall, William E., Murtaza, Anwar, Heyen, Jonathan R., Gallego, Rebecca, Quinlan, Casey, McAlpine, Indrawan, VanArsdale, Todd L.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract 2327: Structural and kinetic characterization of crizotinib with wild-type and mutant anaplastic lymphoma kinase
McTigue, Michele A., Timofeevski, Sergei L., Liu, Wei, Deng, Ya-Li, Marrone, Tami, Cui, Jean, Brooun, Alexei
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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