Potent MCH-1 receptor antagonists from cis-1,4-diaminocyclohexane-derived indane analogs
Qian, Yimin, Conde-Knape, Karin, Erickson, Shawn D., Falcioni, Fiorenza, Gillespie, Paul, Hakimi, Irina, Mennona, Francis, Ren, Yonglin, Salari, Hamid, So, Sung-Sau, Tilley, Jefferson W.
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
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Novel glucokinase activators: a patent review (2008 - 2010)
Sarabu, Ramakanth, Berthel, Steven J, Kester, Robert F, Tilley, Jefferson W
Published in Expert opinion on therapeutic patents (01.01.2011)
Published in Expert opinion on therapeutic patents (01.01.2011)
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Identification of N-acyl 4-(5-pyrimidine-2,4-dionyl)phenylalanine derivatives and their orally active prodrug esters as dual-acting alpha4–beta1 and alpha4–beta7 receptor antagonists
Sidduri, Achyutharao, Tilley, Jefferson W., Lou, Jianping, Tare, Nadine, Cavallo, Gary, Frank, Karl, Pamidimukkala, Anjula, Choi, Duk Soon, Gerber, Louise, Railkar, Aruna, Renzetti, Louis
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
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Identification of N-acyl 4-(3-pyridonyl)phenylalanine derivatives and their orally active prodrug esters as dual acting α4β1 and α4β7 receptor antagonists
Tilley, Jefferson W., Sidduri, Achyutharao, Lou, Jianping, Kaplan, Gerry, Tare, Nadine, Cavallo, Gary, Frank, Karl, Pamidimukkala, Anjula, Choi, Duk Soon, Gerber, Louise, Railkar, Aruna, Renzetti, Louis
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
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Discovery of camphor-derived pyrazolones as 11β-hydroxysteroid dehydrogenase type 1 inhibitors
Gillespie, Paul, Pietranico-Cole, Sherrie, Myers, Michael, Bilotta, Joseph A., Conde-Knape, Karin, Fotouhi, Nader, Goodnow, Robert A., Guertin, Kevin R., Hamilton, Matthew M., Haynes, Nancy-Ellen, Liu, Baolian, Qi, Lida, Ren, Yonglin, Scott, Nathan R., So, Sung-Sau, Spence, Cheryl, Taub, Rebecca, Thakkar, Kshitij, Tilley, Jefferson W., Zwingelstein, Catherine
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
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The discovery of VLA-4 antagonists
Tilley, Jefferson W, Chen, Li, Sidduri, Achyutharao, Fotouhi, Nader
Published in Current topics in medicinal chemistry (01.01.2004)
Published in Current topics in medicinal chemistry (01.01.2004)
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Potent, selective MCH-1 receptor antagonists
Erickson, Shawn D., Banner, Bruce, Berthel, Steven, Conde-Knape, Karin, Falcioni, Fiorenza, Hakimi, Irina, Hennessy, Bernard, Kester, Robert F., Kim, Kyungjin, Ma, Chun, McComas, Warren, Mennona, Francis, Mischke, Steven, Orzechowski, Lucy, Qian, Yimin, Salari, Hamid, Tengi, John, Thakkar, Kshitij, Taub, Rebecca, Tilley, Jefferson W., Wang, Hong
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
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Metabolic/endocrine system
Sarabu, Ramakanth, Tilley, Jefferson W
Published in Drug discovery today. Therapeutic strategies (01.06.2007)
Published in Drug discovery today. Therapeutic strategies (01.06.2007)
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Identification of a Small Molecule Inhibitor of the IL-2/IL-2Rα Receptor Interaction Which Binds to IL-2
Tilley, Jefferson W, Chen, Li, Fry, David C, Emerson, S. Donald, Powers, Gordon D, Biondi, Denise, Varnell, Tracey, Trilles, Richard, Guthrie, Robert, Mennona, Francis, Kaplan, Gerry, LeMahieu, Ronald A, Carson, Mathew, Han, Ru-Jen, Liu, C.-M, Palermo, Robert, Ju, Grace
Published in Journal of the American Chemical Society (13.08.1997)
Published in Journal of the American Chemical Society (13.08.1997)
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Focused library approach for identification of new N-acylphenylalanines as VCAM/VLA-4 antagonists
Chen, Li, Trilles, Richard, Miklowski, Dorota, Huang, Tai-Nan, Fry, David, Campbell, Robert, Rowan, Karen, Schwinge, Virginia, Tilley, Jefferson W.
Published in Bioorganic & medicinal chemistry letters (17.06.2002)
Published in Bioorganic & medicinal chemistry letters (17.06.2002)
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N-Aroyl- l-Phenylalanine Derivatives as VCAM/VLA-4 Antagonists
Sidduri, Achyutharao, Tilley, Jefferson W., Lou, Jian Ping, Chen, Li, Kaplan, Gerry, Mennona, Frank, Campbell, Robert, Guthrie, Robert, Huang, Tai-Nan, Rowan, Karen, Schwinge, Virginia, Renzetti, Louis M.
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
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The design and synthesis of potent cyclic peptide VCAM-VLA-4 antagonists incorporating an achiral Asp-Pro mimetic
FOTOUHI, N, JOSHI, P, FRY, D, COOK, C, TILLEY, J. W, KAPLAN, G, HANGLOW, A, ROWAN, K, SCHWINGE, V, WOLITZKY, B
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
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N-Benzylpyroglutamyl-L-phenylalanine derivatives as VCAM/VLA-4 antagonists
LI CHEN, TILLEY, J. W, WOLITZKY, B, ROWAN, K, GUTHRIE, R. W, MENNONA, F, HUANG, T.-N, KAPLAN, G, TRILLES, R, MIKLOWSKI, D, HUBY, N, SCHWINGE, V
Published in Bioorganic & medicinal chemistry letters (17.04.2000)
Published in Bioorganic & medicinal chemistry letters (17.04.2000)
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Synthesis of constrained L-phenylalanine derivatives incorporating a benzazepinone or an azepinone ring as VCAM/VLA-4 antagonists
Sidduri, A, Lou, JP, Campbell, R, Rowan, K, Tilley, JW
Published in Tetrahedron letters (10.12.2001)
Published in Tetrahedron letters (10.12.2001)
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Discovery of 2‑[3,5-Dichloro-4-(5-isopropyl-6-oxo-1,6-dihydropyridazin-3-yloxy)phenyl]-3,5-dioxo-2,3,4,5-tetrahydro[1,2,4]triazine-6-carbonitrile (MGL-3196), a Highly Selective Thyroid Hormone Receptor β Agonist in Clinical Trials for the Treatment of Dyslipidemia
Kelly, Martha J, Pietranico-Cole, Sherrie, Larigan, J. Douglas, Haynes, Nancy-Ellen, Reynolds, Charles H, Scott, Nathan, Vermeulen, John, Dvorozniak, Mark, Conde-Knape, Karin, Huang, Kuo-Sen, So, Sung-Sau, Thakkar, Kshitij, Qian, Yimin, Banner, Bruce, Mennona, Frank, Danzi, Sara, Klein, Irwin, Taub, Rebecca, Tilley, Jefferson
Published in Journal of medicinal chemistry (22.05.2014)
Published in Journal of medicinal chemistry (22.05.2014)
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N-Cycloalkanoyl- l-Phenylalanine Derivatives as VCAM/VLA-4 Antagonists
Sidduri, Achyutharao, Tilley, Jefferson W, Hull, Kenneth, Ping Lou, Jian, Kaplan, Gerry, Sheffron, Allen, Chen, Li, Campbell, Robert, Guthrie, Robert, Huang, Tai-Nan, Huby, Nicholas, Rowan, Karen, Schwinge, Virginia, Renzetti, Louis M
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
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N-Acyl phenylalanine analogues as potent small molecule VLA-4 antagonists
LI CHEN, TILLEY, J. W, WOLITZKY, B, HUANG, T.-N, MIKLOWSKI, D, TRILLES, R, GUTHRIE, R. W, KIN LUK, HANGLOW, A, ROWAN, K, SCHWINGE, V
Published in Bioorganic & medicinal chemistry letters (17.04.2000)
Published in Bioorganic & medicinal chemistry letters (17.04.2000)
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