Discovery and Preclinical Validation of [11C]AZ13153556, a Novel Probe for the Histamine Type 3 Receptor
Schou, Magnus, Varnäs, Katarina, Jureus, Anders, Ahlgren, Charlotte, Malmquist, Jonas, Häggkvist, Jenny, Tari, Lenke, Wesolowski, Steven S, Throner, Scott R, Brown, Dean G, Nilsson, Maria, Johnström, Peter, Finnema, Sjoerd J, Nakao, Ryuji, Amini, Nahid, Takano, Akihiro, Farde, Lars
Published in ACS chemical neuroscience (17.02.2016)
Published in ACS chemical neuroscience (17.02.2016)
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Discovery of Spirofused Piperazine and Diazepane Amides as Selective Histamine‑3 Antagonists with in Vivo Efficacy in a Mouse Model of Cognition
Brown, Dean G, Bernstein, Peter R, Griffin, Andrew, Wesolowski, Steve, Labrecque, Denis, Tremblay, Maxime C, Sylvester, Mark, Mauger, Russell, Edwards, Phillip D, Throner, Scott R, Folmer, James J, Cacciola, Joseph, Scott, Clay, Lazor, Lois A, Pourashraf, Mehrnaz, Santhakumar, Vijayaratnam, Potts, William M, Sydserff, Simon, Giguère, Pascall, Lévesque, Carine, Dasser, Mohammed, Groblewski, Thierry
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Discovery of novel positive allosteric modulators of the metabotropic glutamate receptor 5 (mGlu 5)
Varnes, Jeffrey G., Marcus, Andrew P., Mauger, Russell C., Throner, Scott R., Hoesch, Valerie, King, Megan M., Wang, Xia, Sygowski, Linda A., Spear, Nathan, Gadient, Reto, Brown, Dean G., Campbell, James B.
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
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SAR development of a series of 8-azabicyclo[3.2.1]octan-3-yloxy-benzamides as kappa opioid receptor antagonists. Part 2
Brugel, Todd A., Smith, Reed W., Balestra, Michael, Becker, Christopher, Daniels, Thalia, Koether, Gerard M., Throner, Scott R., Panko, Laura M., Brown, Dean G., Liu, Ruifeng, Gordon, John, Peters, Matthew F.
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
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Discovery of 8-azabicyclo[3.2.1]octan-3-yloxy-benzamides as selective antagonists of the kappa opioid receptor. Part 1
Brugel, Todd A., Smith, Reed W., Balestra, Michael, Becker, Christopher, Daniels, Thalia, Hoerter, Tiffany N., Koether, Gerard M., Throner, Scott R., Panko, Laura M., Folmer, James J., Cacciola, Joseph, Hunter, Angela M., Liu, Ruifeng, Edwards, Philip D., Brown, Dean G., Gordon, John, Ledonne, Norman C., Pietras, Mark, Schroeder, Patricia, Sygowski, Linda A., Hirata, Lee T., Zacco, Anna, Peters, Matthew F.
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
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Azepines and Piperidines with Dual Norepinephrine Dopamine Uptake Inhibition and Antidepressant Activity
Brown, Dean G, Bernstein, Peter R, Wu, Ye, Urbanek, Rebecca A, Becker, Christopher W, Throner, Scott R, Dembofsky, Bruce T, Steelman, Gary B, Lazor, Lois A, Scott, Clay W, Wood, Michael W, Wesolowski, Steven S, Nugiel, David A, Koch, Stephanie, Yu, Jian, Pivonka, Donald E, Li, Shuang, Thompson, Carol, Zacco, Anna, Elmore, Charles S, Schroeder, Patricia, Liu, JianWei, Hurley, Christopher A, Ward, Stuart, Hunt, Hazel J, Williams, Karen, McLaughlin, Joseph, Hoesch, Valerie, Sydserff, Simon, Maier, Donna, Aharony, David
Published in ACS medicinal chemistry letters (10.01.2013)
Published in ACS medicinal chemistry letters (10.01.2013)
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Discovery of AZD9833, a Potent and Orally Bioavailable Selective Estrogen Receptor Degrader and Antagonist
Scott, James S, Moss, Thomas A, Balazs, Amber, Barlaam, Bernard, Breed, Jason, Carbajo, Rodrigo J, Chiarparin, Elisabetta, Davey, Paul R. J, Delpuech, Oona, Fawell, Stephen, Fisher, David I, Gagrica, Sladjana, Gangl, Eric T, Grebe, Tyler, Greenwood, Ryan D, Hande, Sudhir, Hatoum-Mokdad, Holia, Herlihy, Kara, Hughes, Samantha, Hunt, Thomas A, Huynh, Hoan, Janbon, Sophie L. M, Johnson, Tony, Kavanagh, Stefan, Klinowska, Teresa, Lawson, Mandy, Lister, Andrew S, Marden, Stacey, McGinnity, Dermot F, Morrow, Christopher J, Nissink, J. Willem M, O’Donovan, Daniel H, Peng, Bo, Polanski, Radoslaw, Stead, Darren S, Stokes, Stephen, Thakur, Kumar, Throner, Scott R, Tucker, Michael J, Varnes, Jeffrey, Wang, Haixia, Wilson, David M, Wu, Dedong, Wu, Ye, Yang, Bin, Yang, Wenzhan
Published in Journal of medicinal chemistry (10.12.2020)
Published in Journal of medicinal chemistry (10.12.2020)
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