Toxoflavins and Deazaflavins as the First Reported Selective Small Molecule Inhibitors of Tyrosyl-DNA Phosphodiesterase II
Raoof, Ali, Depledge, Paul, Hamilton, Niall M, Hamilton, Nicola S, Hitchin, James R, Hopkins, Gemma V, Jordan, Allan M, Maguire, Laura A, McGonagle, Alison E, Mould, Daniel P, Rushbrooke, Mathew, Small, Helen F, Smith, Kate M, Thomson, Graeme J, Turlais, Fabrice, Waddell, Ian D, Waszkowycz, Bohdan, Watson, Amanda J, Ogilvie, Donald J
Published in Journal of medicinal chemistry (22.08.2013)
Published in Journal of medicinal chemistry (22.08.2013)
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Small-Molecule Inhibition of UBE2T/FANCL-Mediated Ubiquitylation in the Fanconi Anemia Pathway
Cornwell, Matthew J, Thomson, Graeme J, Coates, Julia, Belotserkovskaya, Rimma, Waddell, Ian D, Jackson, Stephen P, Galanty, Yaron
Published in ACS chemical biology (18.10.2019)
Published in ACS chemical biology (18.10.2019)
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The discovery of 2-substituted phenol quinazolines as potent RET kinase inhibitors with improved KDR selectivity
Newton, Rebecca, Bowler, Katherine A., Burns, Emily M., Chapman, Philip J., Fairweather, Emma E., Fritzl, Samantha J.R., Goldberg, Kristin M., Hamilton, Niall M., Holt, Sarah V., Hopkins, Gemma V., Jones, Stuart D., Jordan, Allan M., Lyons, Amanda J., Nikki March, H., McDonald, Neil Q., Maguire, Laura A., Mould, Daniel P., Purkiss, Andrew G., Small, Helen F., Stowell, Alexandra I.J., Thomson, Graeme J., Waddell, Ian D., Waszkowycz, Bohdan, Watson, Amanda J., Ogilvie, Donald J.
Published in European journal of medicinal chemistry (13.04.2016)
Published in European journal of medicinal chemistry (13.04.2016)
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Novel Steroid Inhibitors of Glucose 6-Phosphate Dehydrogenase
Hamilton, Niall M, Dawson, Martin, Fairweather, Emma E, Hamilton, Nicola S, Hitchin, James R, James, Dominic I, Jones, Stuart D, Jordan, Allan M, Lyons, Amanda J, Small, Helen F, Thomson, Graeme J, Waddell, Ian D, Ogilvie, Donald J
Published in Journal of medicinal chemistry (10.05.2012)
Published in Journal of medicinal chemistry (10.05.2012)
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Development and evaluation of selective, reversible LSD1 inhibitors derived from fragments
Hitchin, James R., Blagg, Julian, Burke, Rosemary, Burns, Samantha, Cockerill, Mark J., Fairweather, Emma E., Hutton, Colin, Jordan, Allan M., McAndrew, Craig, Mirza, Amin, Mould, Daniel, Thomson, Graeme J., Waddell, Ian, Ogilvie, Donald J.
Published in MedChemComm (01.11.2013)
Published in MedChemComm (01.11.2013)
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A fluorescence-based assay for the apurinic/apyrimidinic-site cleavage activity of human tyrosyl-DNA phosphodiesterase 1
Thomson, Graeme J., Hamilton, Nicola S., Hopkins, Gemma V., Waddell, Ian D., Watson, Amanda J., Ogilvie, Donald J.
Published in Analytical biochemistry (01.09.2013)
Published in Analytical biochemistry (01.09.2013)
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Abstract 1139: Novel, cellular active inhibitors of G6PD, a key mediator of ROS-induced cellular stress
Jordan, Allan M., Hamilton, Niall M., Hamilton, Nicola S., Hitchin, James R., James, Dominic I., Jones, Stuart D., Lyons, Amanda J., March, H. Nikki, Thomson, Graeme J., Waddell, Ian D., Ogilvie, Donald J.
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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Development and evaluation of selective, reversible LSD1 inhibitors derived from fragmentsElectronic supplementary information (ESI) available. See DOI: 10.1039/c3md00226h
Hitchin, James R, Blagg, Julian, Burke, Rosemary, Burns, Samantha, Cockerill, Mark J, Fairweather, Emma E, Hutton, Colin, Jordan, Allan M, McAndrew, Craig, Mirza, Amin, Mould, Daniel, Thomson, Graeme J, Waddell, Ian, Ogilvie, Donald J
Year of Publication 23.10.2013
Year of Publication 23.10.2013
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Single-center study comparing computed tomography colonography with conventional colonoscopy
Roberts-Thomson, Ian C, Tucker, Graeme R, Hewett, Peter J, Cheung, Peter, Sebben, Ruben A, Khoo, E E Win, Marker, Julie D, Clapton, Wayne K
Published in World journal of gastroenterology : WJG (21.01.2008)
Published in World journal of gastroenterology : WJG (21.01.2008)
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