Substrate-biased activity-based probes identify proteases that cleave receptor CDCP1
Kryza, Thomas, Khan, Tashbib, Lovell, Scott, Harrington, Brittney S, Yin, Julia, Porazinski, Sean, Pajic, Marina, Koistinen, Hannu, Rantala, Juha K, Dreyer, Tobias, Magdolen, Viktor, Reuning, Ute, He, Yaowu, Tate, Edward W, Hooper, John D
Published in Nature chemical biology (01.07.2021)
Published in Nature chemical biology (01.07.2021)
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Journal Article
100: EXOME SEQUENCING OF A FAMILY WITH A SEVERE COLITIS PHENOTYPE IDENTIFIES A RARE MISSENSE MUTATION IN A NOVEL IBD GENE
Giri, Rabina, Gordon, Robert, Magor, Graham W., He, Yaowu, Kryza, Thomas, Khan, Tashbib, Schreiber, Veronika, Hasnain, Sumaira Z., Ewing, Adam, Hooper, John, Florin, Timothy H., Perkins, Andrew, Gala, Manish, Begun, Jakob
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2022)
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2022)
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Inhibition of Aurora B kinase (AURKB) enhances the effectiveness of 5-fluorouracil chemotherapy against colorectal cancer cells
Shah, Esha T, Molloy, Christopher, Gough, Madeline, Kryza, Thomas, Samuel, Selwin G, Tucker, Amos, Bhatia, Maneet, Ferguson, Genevieve, Heyman, Rebecca, Vora, Shivam, Monkman, James, Bolderson, Emma, Kulasinghe, Arutha, He, Yaowu, Gabrielli, Brian, Hooper, John D, Richard, Derek J, O'Byrne, Kenneth J, Adams, Mark N
Published in British journal of cancer (20.04.2024)
Published in British journal of cancer (20.04.2024)
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Journal Article
Tissue factor pathway inhibitor 2 is a potent kallikrein-related protease 12 inhibitor
Lavergne, Marion, Guillon-Munos, Audrey, Lenga Ma Bonda, Woodys, Attucci, Sylvie, Kryza, Thomas, Barascu, Aurélia, Moreau, Thierry, Petit-Courty, Agnès, Sizaret, Damien, Courty, Yves, Iochmann, Sophie, Reverdiau, Pascale
Published in Biological chemistry (27.09.2021)
Published in Biological chemistry (27.09.2021)
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Journal Article
Abstract P4-07-26: Development of CDCP1-targeting antibody-drug conjugate for Triple negative and metastatic breast cancer
Gough, Madeline, Khan, Tashbib, Kwah, Kayden, He, Yaowu, Ratnayake, Gishan, Pyke, Christopher, Snell, Cameron, Hooper, John, Kryza, Thomas
Published in Cancer research (Chicago, Ill.) (01.03.2023)
Published in Cancer research (Chicago, Ill.) (01.03.2023)
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Journal Article
In vitro engineering of a bone metastases model allows for study of the effects of antiandrogen therapies in advanced prostate cancer
Bock, Nathalie, Kryza, Thomas, Shokoohmand, Ali, Röhl, Joan, Ravichandran, Akhilandeshwari, Wille, Marie-Luise, Nelson, Colleen C, Hutmacher, Dietmar W, Clements, Judith A
Published in Science advances (01.06.2021)
Published in Science advances (01.06.2021)
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Journal Article
Downregulation of the neonatal Fc receptor expression in non-small cell lung cancer tissue is associated with a poor prognosis
Dalloneau, Emilie, Baroukh, Nadine, Mavridis, Konstantinos, Maillet, Agnès, Gueugnon, Fabien, Courty, Yves, Petit, Agnès, Kryza, Thomas, Del Rio, Maguy, Guyetant, Serge, Cadena Castaneda, Diana Carolina, Dhommée, Christine, Arnoult, Christophe, Scorilas, Andreas, Gouilleux-Gruart, Valérie, Heuzé-Vourc'h, Nathalie
Published in Oncotarget (23.08.2016)
Published in Oncotarget (23.08.2016)
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Journal Article
Angiogenesis stimulated by human kallikrein-related peptidase 12 acting via a platelet-derived growth factor B-dependent paracrine pathway
Kryza, Thomas, Achard, Carole, Parent, Christelle, Marchand-Adam, Sylvain, Guillon-Munos, Audrey, Iochmann, Sophie, Korkmaz, Brice, Respaud, Renaud, Courty, Yves, Heuzé-Vourc'h, Nathalie
Published in The FASEB journal (01.02.2014)
Published in The FASEB journal (01.02.2014)
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Journal Article
Preclinical Evaluation of a Fluorescent Probe Targeting Receptor CDCP1 for Identification of Ovarian Cancer
He, Yaowu, Khan, Tashbib, Kryza, Thomas, Jones, Martina L, Goh, Justin B, Lyons, Nicholas J, Pearce, Lesley A, Lee, Michael D, Gough, Madeline, Rogers, Rebecca, Davies, Claire M, Gilks, C. Blake, Hodgkinson, Thomas, Lourie, Rohan, Barry, Sinead C, Perrin, Lewis C, Williams, Charlotte C, Puttick, Simon, Adams, Timothy E, Munro, Trent P, Hooper, John D, Chetty, Naven
Published in Molecular pharmaceutics (06.09.2021)
Published in Molecular pharmaceutics (06.09.2021)
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Journal Article
Engineering osteoblastic metastases to delineate the adaptive response of androgen-deprived prostate cancer in the bone metastatic microenvironment
Bock, Nathalie, Shokoohmand, Ali, Kryza, Thomas, Röhl, Joan, Meijer, Jonelle, Tran, Phong A, Nelson, Colleen C, Clements, Judith A, Hutmacher, Dietmar W
Published in Bone research (25.04.2019)
Published in Bone research (25.04.2019)
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Journal Article
Effective targeting of intact and proteolysed CDCP1 for imaging and treatment of pancreatic ductal adenocarcinoma
Kryza, Thomas, Khan, Tashbib, Puttick, Simon, Li, Chao, Sokolowski, Kamil A, Tse, Brian Wc, Cuda, Tahleesa, Lyons, Nicholas, Gough, Madeline, Yin, Julia, Parkin, Ashleigh, Deryugina, Elena I, Quigley, James P, Law, Ruby H P, Whisstock, James C, Riddell, Andrew D, Barbour, Andrew P, Wyld, David K, Thomas, Paul A, Rose, Stephen, Snell, Cameron E, Pajic, Marina, He, Yaowu, Hooper, John D
Published in Theranostics (01.01.2020)
Published in Theranostics (01.01.2020)
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Journal Article
Kallikrein‐related peptidase 4 induces cancer‐associated fibroblast features in prostate‐derived stromal cells
Kryza, Thomas, Silva, Lakmali M., Bock, Nathalie, Fuhrman‐Luck, Ruth A., Stephens, Carson R., Gao, Jin, Samaratunga, Hema, Lawrence, Mitchell G., Hooper, John D., Dong, Ying, Risbridger, Gail P., Clements, Judith A.
Published in Molecular oncology (01.10.2017)
Published in Molecular oncology (01.10.2017)
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Journal Article
Anti-CDCP1 immuno-conjugates for detection and inhibition of ovarian cancer
Harrington, Brittney S, He, Yaowu, Khan, Tashbib, Puttick, Simon, Conroy, Paul J, Kryza, Thomas, Cuda, Tahleesa, Sokolowski, Kamil A, Tse, Brian Wc, Robbins, Katherine K, Arachchige, Buddhika J, Stehbens, Samantha J, Pollock, Pamela M, Reed, Sarah, Weroha, S John, Haluska, Paul, Salomon, Carlos, Lourie, Rohan, Perrin, Lewis C, Law, Ruby H P, Whisstock, James C, Hooper, John D
Published in Theranostics (01.01.2020)
Published in Theranostics (01.01.2020)
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Journal Article
MUC13 Cell Surface Mucin Limits Salmonella Typhimurium Infection by Protecting the Mucosal Epithelial BarrierSummary
Michael A. McGuckin, Julie M. Davies, Pascal Felgner, Kuan Yau Wong, Rabina Giri, Yaowu He, Md Moniruzzaman, Thomas Kryza, Haressh Sajiir, John D. Hooper, Timothy H. Florin, Jakob Begun, Abderrahim Oussalah, Sumaira Z. Hasnain, Michael Hensel, Yong H. Sheng
Published in Cellular and molecular gastroenterology and hepatology (01.01.2023)
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Published in Cellular and molecular gastroenterology and hepatology (01.01.2023)
Journal Article
CUB Domain-Containing Protein 1 (CDCP1) is a rational target for the development of imaging tracers and antibody-drug conjugates for cancer detection and therapy
Khan, Tashbib, Lyons, Nicholas J, Gough, Madeline, Kwah, Kayden K X, Cuda, Tahleesa J, Snell, Cameron E, Tse, Brian W, Sokolowski, Kamil A, Pearce, Lesley A, Adams, Timothy E, Rose, Stephen E, Puttick, Simon, Pajic, Marina, Adams, Mark N, He, Yaowu, Hooper, John D, Kryza, Thomas
Published in Theranostics (01.01.2022)
Published in Theranostics (01.01.2022)
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Journal Article
MUC13 Cell Surface Mucin Limits Salmonella Typhimurium Infection by Protecting the Mucosal Epithelial Barrier
McGuckin, Michael A, Davies, Julie M, Felgner, Pascal, Wong, Kuan Yau, Giri, Rabina, He, Yaowu, Moniruzzaman, Md, Kryza, Thomas, Sajiir, Haressh, Hooper, John D, Florin, Timothy H, Begun, Jakob, Oussalah, Abderrahim, Hasnain, Sumaira Z, Hensel, Michael, Sheng, Yong H
Published in Cellular and molecular gastroenterology and hepatology (2023)
Published in Cellular and molecular gastroenterology and hepatology (2023)
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Journal Article
Preclinical Molecular PET-CT Imaging Targeting CDCP1 in Colorectal Cancer
Cuda, Tahleesa J., He, Yaowu, Kryza, Thomas, Khan, Tashbib, Tse, Brian W., Sokolowski, Kamil A., Liu, Cheng, Lyons, Nicholas, Gough, Madeline, Snell, Cameron E., Wyld, David K., Rose, Stephen, Riddell, Andrew D., Stevenson, Andrew R. L., Thomas, Paul A., Clark, David A., Puttick, Simon, Hooper, John D.
Published in Contrast media and molecular imaging (2021)
Published in Contrast media and molecular imaging (2021)
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Journal Article
Pro-angiogenic effect of human kallikrein-related peptidase 12 (KLK12) in lung endothelial cells does not depend on kinin-mediated activation of B2 receptor
Kryza, Thomas, Lalmanach, Gilles, Lavergne, Marion, Lecaille, Fabien, Reverdiau, Pascale, Courty, Yves, Heuzé-Vourc’h, Nathalie
Published in Biological chemistry (01.03.2013)
Published in Biological chemistry (01.03.2013)
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Journal Article
Engineering osteoblastic metastases to delineate the adaptive response of androgen-deprived prostate cancer in the bone metastatic microenvironment
Nathalie Bock, Ali Shokoohmand, Thomas Kryza, Joan R?hl, Jonelle Meijer, Phong A. Tran, Colleen C. Nelson, Judith A. Clements, Dietmar W. Hutmacher
Published in 骨研究(英文版) (2019)
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Published in 骨研究(英文版) (2019)
Journal Article
Integration of Two In-depth Quantitative Proteomics Approaches Determines the Kallikrein-related Peptidase 7 (KLK7) Degradome in Ovarian Cancer Cell Secretome
Silva, Lakmali Munasinghage, Kryza, Thomas, Stoll, Thomas, Hoogland, Christine, Dong, Ying, Stephens, Carson Ryan, Hastie, Marcus Lachlan, Magdolen, Viktor, Kleifeld, Oded, Gorman, Jeffrey John, Clements, Judith Ann
Published in Molecular & cellular proteomics (01.05.2019)
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Published in Molecular & cellular proteomics (01.05.2019)
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