Structural insights into inhibitor regulation of the DNA repair protein DNA-PKcs
Liang, Shikang, Thomas, Sherine E, Chaplin, Amanda K, Hardwick, Steven W, Chirgadze, Dimitri Y, Blundell, Tom L
Published in Nature (London) (27.01.2022)
Published in Nature (London) (27.01.2022)
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Journal Article
Arginine-deprivation–induced oxidative damage sterilizes Mycobacterium tuberculosis
Tiwari, Sangeeta, van Tonder, Andries J., Vilchèze, Catherine, Mendes, Vitor, Thomas, Sherine E., Malek, Adel, Chen, Bing, Chen, Mei, Kim, John, Blundell, Tom L., Parkhill, Julian, Weinrick, Brian, Berney, Michael, Jacobs, William R.
Published in Proceedings of the National Academy of Sciences - PNAS (25.09.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (25.09.2018)
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Journal Article
Structural Biology and the Design of New Therapeutics: From HIV and Cancer to Mycobacterial Infections: A Paper Dedicated to John Kendrew
Thomas, Sherine E, Mendes, Vitor, Kim, So Yeon, Malhotra, Sony, Ochoa-Montaño, Bernardo, Blaszczyk, Michal, Blundell, Tom L
Published in Journal of molecular biology (18.08.2017)
Published in Journal of molecular biology (18.08.2017)
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Journal Article
Structure-guided fragment-based drug discovery at the synchrotron: screening binding sites and correlations with hotspot mapping
Thomas, Sherine E, Collins, Patrick, James, Rory Hennell, Mendes, Vitor, Charoensutthivarakul, Sitthivut, Radoux, Chris, Abell, Chris, Coyne, Anthony G, Floto, R Andres, von Delft, Frank, Blundell, Tom L
Published in Philosophical transactions of the Royal Society of London. Series A: Mathematical, physical, and engineering sciences (17.06.2019)
Published in Philosophical transactions of the Royal Society of London. Series A: Mathematical, physical, and engineering sciences (17.06.2019)
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Journal Article
A Fragment‐Based Competitive 19F LB‐NMR Platform For Hotspot‐Directed Ligand Profiling
McCarthy, William J., Thomas, Sherine E., Olaleye, Tayo, Boland, Jennifer A., Floto, R. Andres, Williams, Glyn, Blundell, Tom L., Coyne, Anthony G., Abell, Chris
Published in Angewandte Chemie International Edition (09.09.2024)
Published in Angewandte Chemie International Edition (09.09.2024)
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Journal Article
Genomes, structural biology and drug discovery: combating the impacts of mutations in genetic disease and antibiotic resistance
Pandurangan, Arun Prasad, Ascher, David B, Thomas, Sherine E, Blundell, Tom L
Published in Biochemical Society transactions (15.04.2017)
Published in Biochemical Society transactions (15.04.2017)
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Journal Article
Development of Inhibitors against Mycobacterium abscessus tRNA (m1G37) Methyltransferase (TrmD) Using Fragment-Based Approaches
Whitehouse, Andrew J, Thomas, Sherine E, Brown, Karen P, Fanourakis, Alexander, Chan, Daniel S.-H, Libardo, M. Daben J, Mendes, Vitor, Boshoff, Helena I. M, Floto, R. Andres, Abell, Chris, Blundell, Tom L, Coyne, Anthony G
Published in Journal of medicinal chemistry (08.08.2019)
Published in Journal of medicinal chemistry (08.08.2019)
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Journal Article
Fragment-based discovery of a new class of inhibitors targeting mycobacterial tRNA modification
Thomas, Sherine E, Whitehouse, Andrew J, Brown, Karen, Burbaud, Sophie, Belardinelli, Juan M, Sangen, Jasper, Lahiri, Ramanuj, Libardo, Mark Daben J, Gupta, Pooja, Malhotra, Sony, Boshoff, Helena I M, Jackson, Mary, Abell, Chris, Coyne, Anthony G, Blundell, Tom L, Floto, Rodrigo Andres, Mendes, Vítor
Published in Nucleic acids research (20.08.2020)
Published in Nucleic acids research (20.08.2020)
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Journal Article
SARS-CoV-2 3D database: understanding the coronavirus proteome and evaluating possible drug targets
Alsulami, Ali F, Thomas, Sherine E, Jamasb, Arian R, Beaudoin, Christopher A, Moghul, Ismail, Bannerman, Bridget, Copoiu, Liviu, Vedithi, Sundeep Chaitanya, Torres, Pedro, Blundell, Tom L
Published in Briefings in bioinformatics (22.03.2021)
Published in Briefings in bioinformatics (22.03.2021)
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Journal Article
Predicted structural mimicry of spike receptor-binding motifs from highly pathogenic human coronaviruses
Beaudoin, Christopher A., Jamasb, Arian R., Alsulami, Ali F., Copoiu, Liviu, van Tonder, Andries J., Hala, Sharif, Bannerman, Bridget P., Thomas, Sherine E., Vedithi, Sundeep Chaitanya, Torres, Pedro H.M., Blundell, Tom L.
Published in Computational and structural biotechnology journal (01.01.2021)
Published in Computational and structural biotechnology journal (01.01.2021)
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Journal Article
Ribavirin for Crimean-Congo hemorrhagic fever: systematic review and meta-analysis
Soares-Weiser, Karla, Thomas, Sherine, Thomson, Gail, Garner, Paul
Published in BMC infectious diseases (13.07.2010)
Published in BMC infectious diseases (13.07.2010)
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Journal Article
Mycobacterial genomics and structural bioinformatics: opportunities and challenges in drug discovery
Waman, Vaishali P., Vedithi, Sundeep Chaitanya, Thomas, Sherine E., Bannerman, Bridget P., Munir, Asma, Skwark, Marcin J., Malhotra, Sony, Blundell, Tom L.
Published in Emerging microbes & infections (01.01.2019)
Published in Emerging microbes & infections (01.01.2019)
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Journal Article
A fragment-based approach to assess the ligandability of ArgB, ArgC, ArgD and ArgF in the L-arginine biosynthetic pathway of Mycobacterium tuberculosis
Gupta, Pooja, Thomas, Sherine E., Zaidan, Shaymaa A., Pasillas, Maria A., Cory-Wright, James, Sebastián-Pérez, Víctor, Burgess, Ailidh, Cattermole, Emma, Meghir, Clio, Abell, Chris, Coyne, Anthony G., Jacobs, William R., Blundell, Tom L., Tiwari, Sangeeta, Mendes, Vítor
Published in Computational and structural biotechnology journal (01.01.2021)
Published in Computational and structural biotechnology journal (01.01.2021)
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Journal Article
Structural insights into the EthR-DNA interaction using native mass spectrometry
Shiu-Hin Chan, Daniel, Seetoh, Wei-Guang, McConnell, Brendan N, Matak-Vinković, Dijana, Thomas, Sherine E, Mendes, Vitor, Blaszczyk, Michal, Coyne, Anthony G, Blundell, Tom L, Abell, Chris
Published in Chemical communications (Cambridge, England) (23.03.2017)
Published in Chemical communications (Cambridge, England) (23.03.2017)
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Journal Article
Fragment Screening against the EthR–DNA Interaction by Native Mass Spectrometry
Chan, Daniel Shiu‐Hin, Mendes, Vitor, Thomas, Sherine E., McConnell, Brendan N., Matak‐Vinković, Dijana, Coyne, Anthony G., Blundell, Tom L., Abell, Chris
Published in Angewandte Chemie International Edition (19.06.2017)
Published in Angewandte Chemie International Edition (19.06.2017)
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Journal Article
Structural Characterization of Mycobacterium abscessus Phosphopantetheine Adenylyl Transferase Ligand Interactions: Implications for Fragment-Based Drug Design
Thomas, Sherine E, McCarthy, William J, El Bakali, Jamal, Brown, Karen P, Kim, So Yeon, Blaszczyk, Michal, Mendes, Vítor, Abell, Chris, Floto, R Andres, Coyne, Anthony G, Blundell, Tom L
Published in Frontiers in molecular biosciences (30.05.2022)
Published in Frontiers in molecular biosciences (30.05.2022)
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Journal Article
A Fragment‐Based Competitive 19F LB‐NMR Platform For Hotspot‐Directed Ligand Profiling
McCarthy, William J., Thomas, Sherine E., Olaleye, Tayo, Boland, Jennifer A., Floto, R. Andres, Williams, Glyn, Blundell, Tom L., Coyne, Anthony G., Abell, Chris
Published in Angewandte Chemie (09.09.2024)
Published in Angewandte Chemie (09.09.2024)
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Journal Article
Development of Inhibitors of SAICAR Synthetase (PurC) from Mycobacterium abscessus Using a Fragment-Based Approach
Charoensutthivarakul, Sitthivut, Thomas, Sherine E, Curran, Amy, Brown, Karen P, Belardinelli, Juan M, Whitehouse, Andrew J, Acebrón-García-de-Eulate, Marta, Sangan, Jaspar, Gramani, Subramanian G, Jackson, Mary, Mendes, Vitor, Floto, R. Andres, Blundell, Tom L, Coyne, Anthony G, Abell, Chris
Published in ACS infectious diseases (11.02.2022)
Published in ACS infectious diseases (11.02.2022)
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Journal Article
Glycemia and Cognitive Function in Metabolic Syndrome and Coronary Heart Disease
Avadhani, Radhika, MS, Fowler, Kristen, RN, Barbato, Corinne, BS, Thomas, Sherine, BA, Wong, Winnie, BA, Paul, Camille, BA, Aksakal, Mehmet, MD, Hauser, Thomas H., MMSC, MPH, MD, Weinger, Katie, EdD, RN, Goldfine, Allison B., MD
Published in The American journal of medicine (01.01.2015)
Published in The American journal of medicine (01.01.2015)
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