The G Protein-Coupled Receptor GPR17: Overview and Update
Marucci, Gabriella, Dal Ben, Diego, Lambertucci, Catia, Santinelli, Claudia, Spinaci, Andrea, Thomas, Ajiroghene, Volpini, Rosaria, Buccioni, Michela
Published in ChemMedChem (06.12.2016)
Published in ChemMedChem (06.12.2016)
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Journal Article
Antiproliferative Evaluation of Isofuranodiene on Breast and Prostate Cancer Cell Lines
Marucci, Gabriella, Thomas, Ajiroghene, Papa, Fabrizio, Maggi, Filippo, Lambertucci, Catia, Dal Ben, Diego, Buccioni, Michela, Volpini, Rosaria
Published in TheScientificWorld (01.01.2014)
Published in TheScientificWorld (01.01.2014)
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Journal Article
2′,3′-O-Substituted ATP derivatives as potent antagonists of purinergic P2X3 receptors and potential analgesic agents
Dal Ben, Diego, Marchenkova, Anna, Thomas, Ajiroghene, Lambertucci, Catia, Spinaci, Andrea, Marucci, Gabriella, Nistri, Andrea, Volpini, Rosaria
Published in Purinergic signalling (01.03.2017)
Published in Purinergic signalling (01.03.2017)
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Journal Article
Overview on Radiolabel-Free in vitro Assays for GPCRs
Buccioni, Michela, Santinelli, Claudia, Angeli, Piero, Dal Ben, Diego, Lambertucci, Catia, Thomas, Ajiroghene, Volpini, Rosaria, Marucci, Gabriella
Published in Mini reviews in medicinal chemistry (01.01.2017)
Published in Mini reviews in medicinal chemistry (01.01.2017)
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Journal Article
Innovative functional cAMP assay for studying G protein-coupled receptors: application to the pharmacological characterization of GPR17
Buccioni, Michela, Marucci, Gabriella, Dal Ben, Diego, Giacobbe, Dania, Lambertucci, Catia, Soverchia, Laura, Thomas, Ajiroghene, Volpini, Rosaria, Cristalli, Gloria
Published in Purinergic signalling (01.12.2011)
Published in Purinergic signalling (01.12.2011)
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Journal Article
Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A(3) receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation
Varano, Flavia, Catarzi, Daniela, Squarcialupi, Lucia, Betti, Marco, Vincenzi, Fabrizio, Ravani, Annalisa, Varani, Katia, Dal Ben, Diego, Thomas, Ajiroghene, Volpini, Rosaria, Colotta, Vittoria
Published in European journal of medicinal chemistry (26.05.2015)
Published in European journal of medicinal chemistry (26.05.2015)
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Journal Article
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A3 receptor antagonists. Synthesis, structure–affinity relationships and molecular modeling studies
Catarzi, Daniela, Varano, Flavia, Poli, Daniela, Squarcialupi, Lucia, Betti, Marco, Trincavelli, Letizia, Martini, Claudia, Dal Ben, Diego, Thomas, Ajiroghene, Volpini, Rosaria, Colotta, Vittoria
Published in Bioorganic & medicinal chemistry (01.01.2015)
Published in Bioorganic & medicinal chemistry (01.01.2015)
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Journal Article
Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation
Varano, Flavia, Catarzi, Daniela, Squarcialupi, Lucia, Betti, Marco, Vincenzi, Fabrizio, Ravani, Annalisa, Varani, Katia, Dal Ben, Diego, Thomas, Ajiroghene, Volpini, Rosaria, Colotta, Vittoria
Published in European journal of medicinal chemistry (26.05.2015)
Published in European journal of medicinal chemistry (26.05.2015)
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Journal Article
1,2,4-Triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A(3) receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies
Catarzi, Daniela, Varano, Flavia, Poli, Daniela, Squarcialupi, Lucia, Betti, Marco, Trincavelli, Letizia, Martini, Claudia, Dal Ben, Diego, Thomas, Ajiroghene, Volpini, Rosaria, Colotta, Vittoria
Published in Bioorganic & medicinal chemistry (01.01.2015)
Published in Bioorganic & medicinal chemistry (01.01.2015)
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Journal Article
Imidazo[1,2-a]pyrazin-8-amine core for the design of new adenosine receptor antagonists: Structural exploration to target the A(3) and A(2A) subtypes
Poli, Daniela, Falsini, Matteo, Varano, Flavia, Betti, Marco, Varani, Katia, Vincenzi, Fabrizio, Pugliese, Anna Maria, Pedata, Felicita, Dal Ben, Diego, Thomas, Ajiroghene, Palchetti, Ilaria, Bettazzi, Francesca, Catarzi, Daniela, Colotta, Vittoria
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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Journal Article
8-(2-Furyl)adenine derivatives as A(2A) adenosine receptor ligands
Dal Ben, Diego, Buccioni, Michela, Lambertucci, Catia, Thomas, Ajiroghene, Klotz, Karl-Norbert, Federico, Stephanie, Cacciari, Barbara, Spalluto, Giampiero, Volpini, Rosaria
Published in European journal of medicinal chemistry (01.12.2013)
Published in European journal of medicinal chemistry (01.12.2013)
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Journal Article
The GProtein-Coupled Receptor GPR17: Overview and Update
Marucci, Gabriella, DalBen, Diego, Lambertucci, Catia, Santinelli, Claudia, Spinaci, Andrea, Thomas, Ajiroghene, Volpini, Rosaria, Buccioni, Michela
Published in ChemMedChem (01.12.2016)
Published in ChemMedChem (01.12.2016)
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Journal Article
The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A(2A) Adenosine Receptor
Thomas, Ajiroghene, Buccioni, Michela, Dal Ben, Diego, Lambertucci, Catia, Marucci, Gabriella, Santinelli, Claudia, Spinaci, Andrea, Kachler, Sonja, Klotz, Karl-Norbert, Volpini, Rosaria
Published in ChemMedChem (19.08.2016)
Published in ChemMedChem (19.08.2016)
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Journal Article
Molecular modeling study on potent and selective adenosine A(3) receptor agonists
Dal Ben, Diego, Buccioni, Michela, Lambertucci, Catia, Marucci, Gabriella, Thomas, Ajiroghene, Volpini, Rosaria, Cristalli, Gloria
Published in Bioorganic & medicinal chemistry (15.11.2010)
Published in Bioorganic & medicinal chemistry (15.11.2010)
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Journal Article
Simulation and Comparative Analysis of Different Binding Modes of Non-nucleoside Agonists at the A2A Adenosine Receptor
Dal Ben, Diego, Buccioni, Michela, Lambertucci, Catia, Marucci, Gabriella, Santinelli, Claudia, Spinaci, Andrea, Thomas, Ajiroghene, Volpini, Rosaria
Published in Molecular informatics (01.09.2016)
Published in Molecular informatics (01.09.2016)
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Journal Article
Evidence for the Existence of a Specific G Protein-Coupled Receptor Activated by Guanosine
Volpini, Rosaria, Marucci, Gabriella, Buccioni, Michela, Dal Ben, Diego, Lambertucci, Catia, Lammi, Carmen, Mishra, Ram C., Thomas, Ajiroghene, Cristalli, Gloria
Published in ChemMedChem (06.06.2011)
Published in ChemMedChem (06.06.2011)
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Journal Article
Imidazo[1,2-a]pyrazin-8-amine core for the design of new adenosine receptor antagonists: Structural exploration to target the A3 and A2A subtypes
Poli, Daniela, Falsini, Matteo, Varano, Flavia, Betti, Marco, Varani, Katia, Vincenzi, Fabrizio, Pugliese, Anna Maria, Pedata, Felicita, Dal Ben, Diego, Thomas, Ajiroghene, Palchetti, Ilaria, Bettazzi, Francesca, Catarzi, Daniela, Colotta, Vittoria
Published in European journal of medicinal chemistry (05.01.2017)
Published in European journal of medicinal chemistry (05.01.2017)
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Journal Article