Identification of candidate substrates for poly(ADP‐ribose) polymerase‐2 (PARP2) in the absence of DNA damage using high‐density protein microarrays
Troiani, Sonia, Lupi, Rosita, Perego, Rita, Re Depaolini, Stefania, Thieffine, Sandrine, Bosotti, Roberta, Rusconi, Luisa
Published in The FEBS journal (01.10.2011)
Published in The FEBS journal (01.10.2011)
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Optimization of pyrazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)
Huynh, Tram, Chen, Zhong, Pang, Suhong, Geng, Jieping, Bandiera, Tiziano, Bindi, Simona, Vianello, Paola, Roletto, Fulvia, Thieffine, Sandrine, Galvani, Arturo, Vaccaro, Wayne, Poss, Michael A., Trainor, George L., Lorenzi, Matthew V., Gottardis, Marco, Jayaraman, Lata, Purandare, Ashok V.
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
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Cell Division Cycle 7 Kinase Inhibitors: 1H-Pyrrolo[2,3-b]pyridines, Synthesis and Structure−Activity Relationships
Ermoli, Antonella, Bargiotti, Alberto, Brasca, Maria Gabriella, Ciavolella, Antonella, Colombo, Nicoletta, Fachin, Gabriele, Isacchi, Antonella, Menichincheri, Maria, Molinari, Antonio, Montagnoli, Alessia, Pillan, Antonio, Rainoldi, Sonia, Sirtori, Federico Riccardi, Sola, Francesco, Thieffine, Sandrine, Tibolla, Marcellino, Valsasina, Barbara, Volpi, Daniele, Santocanale, Corrado, Vanotti, Ermes
Published in Journal of medicinal chemistry (23.07.2009)
Published in Journal of medicinal chemistry (23.07.2009)
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Natural and synthetic 2-oxoglutarate derivatives are substrates for oncogenic variants of human isocitrate dehydrogenase 1 and 2
Liu, Xiao, Reinbold, Raphael, Liu, Shuang, Herold, Ryan A., Rabe, Patrick, Duclos, Stéphanie, Yadav, Rahul B., Abboud, Martine I., Thieffine, Sandrine, Armstrong, Fraser A., Brewitz, Lennart, Schofield, Christopher J.
Published in The Journal of biological chemistry (01.02.2023)
Published in The Journal of biological chemistry (01.02.2023)
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Structural basis for CARM1 inhibition by indole and pyrazole inhibitors
Sack, John S, Thieffine, Sandrine, Bandiera, Tiziano, Fasolini, Marina, Duke, Gerald J, Jayaraman, Lata, Kish, Kevin F, Klei, Herbert E, Purandare, Ashok V, Rosettani, Pamela, Troiani, Sonia, Xie, Dianlin, Bertrand, Jay A
Published in Biochemical journal (01.06.2011)
Published in Biochemical journal (01.06.2011)
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Insights into PARP Inhibitors' Selectivity Using Fluorescence Polarization and Surface Plasmon Resonance Binding Assays
Papeo, Gianluca, Avanzi, Nilla, Bettoni, Serena, Leone, Antonella, Paolucci, Mauro, Perego, Rita, Quartieri, Francesca, Riccardi-Sirtori, Federico, Thieffine, Sandrine, Montagnoli, Alessia, Lupi, Rosita
Published in Journal of biomolecular screening (01.09.2014)
Published in Journal of biomolecular screening (01.09.2014)
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Abstract 691: In vitro and in vivo characterization of selective orally available Parp-1 inhibitors with demonstrated antitumor efficacy in BRCA negative cancer models
Papeo, Gianluca, Rainoldi, Sonia, Gianellini, Laura, Ciavolella, Antonella, Leone, Antonella, Lupi, Rosita, Sola, Francesco, Caprera, Francesco, Paolucci, Mauro, Thieffine, Sandrine, Perego, Rita, Albanese, Clara, Casale, Elena, Forte, Barbara, Guanci, Marco, Orsini, Paolo, Posteri, Helena, Scolaro, Alessandra, Riccardi-Sirtori, Federico, Zuccotto, Fabio, Donati, Daniele, Moll, Jurgen, Montagnoli, Alessia
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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Cell Division Cycle 7 Kinase Inhibitors: 1 H -Pyrrolo[2,3- b ]pyridines, Synthesis and Structure−Activity Relationships
Ermoli, Antonella, Bargiotti, Alberto, Brasca, Maria Gabriella, Ciavolella, Antonella, Colombo, Nicoletta, Fachin, Gabriele, Isacchi, Antonella, Menichincheri, Maria, Molinari, Antonio, Montagnoli, Alessia, Pillan, Antonio, Rainoldi, Sonia, Sirtori, Federico Riccardi, Sola, Francesco, Thieffine, Sandrine, Tibolla, Marcellino, Valsasina, Barbara, Volpi, Daniele, Santocanale, Corrado, Vanotti, Ermes
Published in Journal of medicinal chemistry (23.07.2009)
Published in Journal of medicinal chemistry (23.07.2009)
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TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF
VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE
Year of Publication 03.03.2005
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Year of Publication 03.03.2005
Patent
TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF
VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE
Year of Publication 20.01.2005
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Year of Publication 20.01.2005
Patent
TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF
VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE
Year of Publication 18.11.2004
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Year of Publication 18.11.2004
Patent
TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF
VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, KALISZ, HENRYK, PEREGO, RITA, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE
Year of Publication 18.11.2004
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Year of Publication 18.11.2004
Patent
TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF
VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE
Year of Publication 08.02.2006
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Year of Publication 08.02.2006
Patent