Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity
Gerninghaus, Joshua, Zhubi, Rezart, Kraemer, Andreas, Marwah Karim, Do Hoang Nhu Tran, Joerger, Andreas C, Schreiber, Christian, Berger, Lena M, Berger, Benedict Tilman, Theresa Al Ehret, Elson, Lewis, Lenz, Christopher, Saxena, Krishna, Mueller, Susanne, Einav, Shirit, Knapp, Stefan, Hanke, Thomas
Published in bioRxiv (18.02.2024)
Published in bioRxiv (18.02.2024)
Get full text
Paper
Journal Article