Detection of Weak Organic Anion-Transporting Polypeptide 1B Inhibition by Probenecid with Plasma-Based Coproporphyrin in Humans
Zhang, Yueping, Holenarsipur, Vinay K, Kandoussi, Hamza, Zeng, Jianing, Mariappan, T Thanga, Sinz, Michael, Shen, Hong
Published in Drug metabolism and disposition (01.10.2020)
Published in Drug metabolism and disposition (01.10.2020)
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Evidence for the Validity of Pyridoxic Acid (PDA) as a Plasma-Based Endogenous Probe for OAT1 and OAT3 Function in Healthy Subjects
Shen, Hong, Holenarsipur, Vinay K, Mariappan, T Thanga, Drexler, Dieter M, Cantone, Joseph L, Rajanna, Prabhakar, Singh Gautam, Shashyendra, Zhang, Yueping, Gan, Jinping, Shipkova, Petia A, Marathe, Punit, Humphreys, W Griffith
Published in The Journal of pharmacology and experimental therapeutics (01.01.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2019)
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Transporter Activity Changes in Nonalcoholic Steatohepatitis: Assessment with Plasma Coproporphyrin I and III
Chatterjee, Sagnik, Mukherjee, Sambuddho, Sankara Sivaprasad, L V J, Naik, Tanvi, Gautam, Shashyendra Singh, Murali, Bokka Venkata, Hadambar, Avinash Annasao, Gunti, Gowtham Raj, Kuchibhotla, Vijaykumar, Deyati, Avisek, Basavanthappa, Sushma, Ramarao, Manjunath, Mariappan, T Thanga, Zinker, Bradley A, Zhang, Yueping, Sinz, Michael, Shen, Hong
Published in The Journal of pharmacology and experimental therapeutics (01.01.2021)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2021)
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Journal Article
Selective IRAK4 Inhibition Attenuates Disease in Murine Lupus Models and Demonstrates Steroid Sparing Activity
Dudhgaonkar, Shailesh, Ranade, Sourabh, Nagar, Jignesh, Subramani, Siva, Prasad, Durga Shiv, Karunanithi, Preethi, Srivastava, Ratika, Venkatesh, Kamala, Selvam, Sabariya, Krishnamurthy, Prasad, Mariappan, T Thanga, Saxena, Ajay, Fan, Li, Stetsko, Dawn K, Holloway, Deborah A, Li, Xin, Zhu, Jun, Yang, Wen-Pin, Ruepp, Stefan, Nair, Satheesh, Santella, Joseph, Duncia, John, Hynes, John, McIntyre, Kim W, Carman, Julie A
Published in The Journal of immunology (1950) (01.02.2017)
Published in The Journal of immunology (1950) (01.02.2017)
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Insight into tissue unbound concentration: utility in drug discovery and development
Mariappan, T Thanga, Mandlekar, Sandhya, Marathe, Punit
Published in Current drug metabolism (01.03.2013)
Published in Current drug metabolism (01.03.2013)
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Estimation of the Unbound Brain Concentration of P‑Glycoprotein Substrates or Nonsubstrates by a Serial Cerebrospinal Fluid Sampling Technique in Rats
Mariappan, T. Thanga, Kurawattimath, Vishwanath, Gautam, Shashyendra Singh, Kulkarni, Chetan P, Kallem, Rajareddy, Taskar, Kunal S, Marathe, Punit H, Mandlekar, Sandhya
Published in Molecular pharmaceutics (03.02.2014)
Published in Molecular pharmaceutics (03.02.2014)
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Journal Article
A modified serial blood sampling technique and utility of dried-blood spot technique in estimation of blood concentration: application in mouse pharmacokinetics
Kurawattimath, Vishwanath, Pocha, Krishna, Thanga Mariappan, T., Trivedi, Ravi Kumar, Mandlekar, Sandhya
Published in European journal of drug metabolism and pharmacokinetics (01.03.2012)
Published in European journal of drug metabolism and pharmacokinetics (01.03.2012)
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Journal Article
In Vitro Stimulation of Multidrug Resistance-Associated Protein 2 Function Is Not Reproduced In Vivo in Rats
Gilibili, Ravindranath Reddy, Kurawattimath, Vishwanath, Murali, Bokka Venkata, Lai, Yurong, Mariappan, T Thanga, Shen, Hong, Chatterjee, Sagnik
Published in Pharmaceutics (08.08.2018)
Published in Pharmaceutics (08.08.2018)
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Journal Article
Role of hepatic blood flow and metabolism in the pharmacokinetics of ten drugs in lean, aged and obese rats
Subramanian, Murali, Kurawattimath, Vishwanath, Pocha, Krishna, Freeden, Chris, Rao, Indranil, Thanga Mariappan, T., Marathe, Punit H., Vikramadithyan, Reeba K., Abraham, Pamela, Kulkarni, Chetan P., Katnapally, Prasanna, Nutakki, Ravikumar, Paruchury, Sundeep, Bhutani, Priyadeep, Mandlekar, Sandhya
Published in Xenobiotica (01.12.2014)
Published in Xenobiotica (01.12.2014)
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Journal Article
Coproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition Assay
Gilibili, Ravindranath Reddy, Chatterjee, Sagnik, Bagul, Pravin, Mosure, Kathleen W, Murali, Bokka Venkata, Mariappan, T Thanga, Mandlekar, Sandhya, Lai, Yurong
Published in Drug metabolism and disposition (01.06.2017)
Published in Drug metabolism and disposition (01.06.2017)
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Journal Article
Unmasking the Role of Uptake Transporters for Digoxin Uptake Across the Barriers of the Central Nervous System in Rat
Taskar, Kunal S, Mariappan, T Thanga, Kurawattimath, Vishwanath, Singh Gautam, Shashyendra, Radhakrishna Mullapudi, TV, Sridhar, Srikanth K, Kallem, Raja Reddy, Marathe, Punit, Mandlekar, Sandhya
Published in Journal of central nervous system disease (01.01.2017)
Published in Journal of central nervous system disease (01.01.2017)
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Journal Article
Endogenous Plasma Kynurenic Acid in Human: A Newly Discovered Biomarker for Drug-Drug Interactions Involving Organic Anion Transporter 1 and 3 Inhibition
Tang, Jennifer, Shen, Hong, Zhao, Xiaofeng, Holenarsipur, Vinay K, Mariappan, T Thanga, Zhang, Yueping, Panfen, Erika, Zheng, Jim, Humphreys, W Griffith, Lai, Yurong
Published in Drug metabolism and disposition (01.12.2021)
Published in Drug metabolism and disposition (01.12.2021)
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Journal Article
A Tribute to Professor Saranjit Singh - A Critical Thinker, Innovator, Mentor, and Educator
Ladumor, Mayur K., Paudel, Amrit, Modhave, Dattatray, Sharma, Sheena, Balhara, Ankit, Singh, Dilip K., Ramalingam, Manikandan, Shah, Ravi, Pavankumarraju, Surapuraju, Kurmi, Moolchand, Mariappan, T. Thanga, Bhutani, Hemant, Prasad, Bhagwat
Published in Journal of pharmaceutical sciences (01.05.2022)
Published in Journal of pharmaceutical sciences (01.05.2022)
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Oral bioavailability, efficacy and gastric tolerability of P2026, a novel nitric oxide-releasing diclofenac in rat
Pathan, Asif R., Karwa, Manoj, Pamidiboina, Venu, Deshattiwar, Jagannath J., Deshmukh, Nitin J., Gaikwad, Parikshit P., Mali, Sunil V., Desai, Dattatraya C., Dhiman, Mini, Thanga Mariappan, T., Sharma, Somesh D., Satyam, Apparao, Nemmani, Kumar V. S.
Published in Inflammopharmacology (01.08.2010)
Published in Inflammopharmacology (01.08.2010)
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Effect of pretreatment regimens of 1-aminobenzotriazole on metabolism and gastric emptying of probe compounds in rat
Padmanabhan, Shweta, Kaur, Harbeer, Rao, Abhijith, Saxena, Ajay, Gupta, Yogesh Kumar, Mariappan, T. Thanga, Holenarsipur, Vinay K.
Published in Xenobiotica (03.06.2019)
Published in Xenobiotica (03.06.2019)
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Journal Article
Coproporphyrin-I: A Fluorescent, Endogenous Optimal Probe Substrate for ABCC2 (MRP2) Suitable for Vesicle-Based MRP2 Inhibition Assay
Gilibili, Ravindranath Reddy, Chatterjee, Sagnik, Bagul, Pravin, Mosure, Kathleen W., Murali, Bokka Venkata, Mariappan, T. Thanga, Mandlekar, Sandhya, Lai, Yurong
Published in Drug metabolism and disposition (01.06.2017)
Published in Drug metabolism and disposition (01.06.2017)
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Journal Article
Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors
Cherney, Emily C, Zhang, Liping, Guo, Weiwei, Huang, Audris, Williams, David, Seitz, Steven, Shan, Weifang, Zhu, Xiao, Gullo-Brown, Johnni, Maley, Derrick, Lin, Tai-an, Hunt, John T, Huang, Christine, Yang, Zheng, D’Arienzo, Celia J, Discenza, Lorell N, Ranasinghe, Asoka, Grubb, Mary F, Traeger, Sarah C, Li, Xin, Johnston, Kathy A, Kopcho, Lisa, Fereshteh, Mark, Foster, Kimberly A, Stefanski, Kevin, Delpy, Diane, Dhar, Gopal, Anandam, Aravind, Mahankali, Sandeep, Padmanabhan, Shweta, Rajanna, Prabhakar, Murali, Venkata, Mariappan, T. Thanga, Pattasseri, Shabeerali, Nimje, Roshan Y, Hong, Zhenqiu, Kempson, James, Rampulla, Richard, Mathur, Arvind, Gupta, Anuradha, Borzilleri, Robert, Vite, Gregory, Balog, Aaron
Published in ACS medicinal chemistry letters (08.07.2021)
Published in ACS medicinal chemistry letters (08.07.2021)
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Optimization of Nicotinamides as Potent and Selective IRAK4 Inhibitors with Efficacy in a Murine Model of Psoriasis
Nair, Satheesh, Kumar, Sreekantha Ratna, Paidi, Venkatram Reddy, Sistla, Ramesh, Kantheti, Durgarao, Polimera, Subba Rao, Thangavel, Soodamani, Mukherjee, Amrita Jha, Das, Mitalee, Bhide, Rajeev S, Pitts, William J, Murugesan, Natesan, Dudhgoankar, Shailesh, Nagar, Jignesh, Subramani, Siva, Mazumder, Debarati, Carman, Julie A, Holloway, Deborah A, Li, Xin, Fereshteh, Mark P, Ruepp, Stefan, Palanisamy, Kamalavenkatesh, Mariappan, T. Thanga, Maddi, Srinivas, Saxena, Ajay, Elzinga, Paul, Chimalakonda, Anjaneya, Ruan, Qian, Ghosh, Kaushik, Bose, Sucharita, Sack, John, Yan, Chunhong, Kiefer, Susan E, Xie, Dianlin, Newitt, John A, Saravanakumar, S. Pon, Rampulla, Richard A, Barrish, Joel C, Carter, Percy H, Hynes, John
Published in ACS medicinal chemistry letters (09.07.2020)
Published in ACS medicinal chemistry letters (09.07.2020)
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Erratum to: A modified serial blood sampling technique and utility of dried-blood spot technique in estimation of blood concentration: application in mouse pharmacokinetics
Kurawattimath, Vishwanath, Pocha, Krishna, Thanga Mariappan, T., Trivedi, Ravi Kumar, Mandlekar, Sandhya
Published in European journal of drug metabolism and pharmacokinetics (01.12.2011)
Published in European journal of drug metabolism and pharmacokinetics (01.12.2011)
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