Highly Diastereoselective Arylations of Substituted Piperidines
Seel, Stephanie, Thaler, Tobias, Takatsu, Keishi, Zhang, Cong, Zipse, Hendrik, Straub, Bernd F, Mayer, Peter, Knochel, Paul
Published in Journal of the American Chemical Society (06.04.2011)
Published in Journal of the American Chemical Society (06.04.2011)
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Journal Article
Highly Diastereoselective Iron-Mediated C(sp2)C(sp3) Cross-Coupling Reactions between Aryl Grignard Reagents and Cyclic Iodohydrine Derivatives
Steib, Andreas K., Thaler, Tobias, Komeyama, Kimihiro, Mayer, Peter, Knochel, Paul
Published in Angewandte Chemie (International ed.) (28.03.2011)
Published in Angewandte Chemie (International ed.) (28.03.2011)
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Journal Article
Potent and Selective Human Prostaglandin F (FP) Receptor Antagonist (BAY-6672) for the Treatment of Idiopathic Pulmonary Fibrosis (IPF)
Beck, Hartmut, Thaler, Tobias, Meibom, Daniel, Meininghaus, Mark, Jörißen, Hannah, Dietz, Lisa, Terjung, Carsten, Bairlein, Michaela, von Bühler, Clemens-Jeremias, Anlauf, Sonja, Fürstner, Chantal, Stellfeld, Timo, Schneider, Dirk, Gericke, Kersten M, Buyck, Thomas, Lovis, Kai, Münster, Uwe, Anlahr, Johanna, Kersten, Elisabeth, Levilain, Guillaume, Marossek, Virginia, Kast, Raimund
Published in Journal of medicinal chemistry (22.10.2020)
Published in Journal of medicinal chemistry (22.10.2020)
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Journal Article
Highly Diastereoselective C(sp³)C(sp) Cross-Coupling Reactions between 1,3- and 1,4-Substituted Cyclohexylzinc Reagents and Bromoalkynes through Remote Stereocontrol
Thaler, Tobias, Guo, Li-Na, Mayer, Peter, Knochel, Paul
Published in Angewandte Chemie (International ed.) (25.02.2011)
Published in Angewandte Chemie (International ed.) (25.02.2011)
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Journal Article
Discovery of IRAK4 Inhibitors BAY1834845 (Zabedosertib) and BAY1830839
Bothe, Ulrich, Günther, Judith, Nubbemeyer, Reinhard, Siebeneicher, Holger, Ring, Sven, Bömer, Ulf, Peters, Michaele, Rausch, Alexandra, Denner, Karsten, Himmel, Herbert, Sutter, Andreas, Terebesi, Ildiko, Lange, Martin, Wengner, Antje M., Guimond, Nicolas, Thaler, Tobias, Platzek, Johannes, Eberspächer, Uwe, Schäfer, Martina, Steuber, Holger, Zollner, Thomas M., Steinmeyer, Andreas, Schmidt, Nicole
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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Journal Article
Highly diastereoselective Csp₃-Csp₂ Negishi cross-coupling with 1,2-, 1,3- and 1,4-substituted cycloalkylzinc compounds
Thaler, Tobias, Haag, Benjamin, Gavryushin, Andrei, Schober, Katrin, Hartmann, Evelyn, Gschwind, Ruth M, Zipse, Hendrik, Mayer, Peter, Knochel, Paul
Published in Nature chemistry (01.02.2010)
Published in Nature chemistry (01.02.2010)
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Journal Article
Preparation of Stereodefined Secondary Alkyllithium Compounds
Seel, Stephanie, Dagousset, Guillaume, Thaler, Tobias, Frischmuth, Annette, Karaghiosoff, Konstantin, Zipse, Hendrik, Knochel, Paul
Published in Chemistry : a European journal (02.04.2013)
Published in Chemistry : a European journal (02.04.2013)
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Journal Article
Sulfoxide–Alkene Hybrids: A New Class of Chiral Ligands for the Hayashi–Miyaura Reaction
Thaler, Tobias, Guo, Li-Na, Steib, Andreas K, Raducan, Mihai, Karaghiosoff, Konstantin, Mayer, Peter, Knochel, Paul
Published in Organic letters (17.06.2011)
Published in Organic letters (17.06.2011)
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Journal Article
Highly diastereoselective Csp 3–Csp 2 Negishi cross-coupling with 1,2-, 1,3- and 1,4-substituted cycloalkylzinc compounds
Thaler, Tobias, Haag, Benjamin, Gavryushin, Andrei, Schober, Katrin, Hartmann, Evelyn, Gschwind, Ruth M, Zipse, Hendrik, Mayer, Peter, Knochel, Paul
Published in Nature chemistry (01.02.2010)
Published in Nature chemistry (01.02.2010)
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