Optimization of Alkylidene Hydrazide Based Human Glucagon Receptor Antagonists. Discovery of the Highly Potent and Orally Available 3-Cyano-4-hydroxybenzoic Acid [1-(2,3,5,6-Tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide
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Published in Journal of medicinal chemistry (19.12.2002)
Published in Journal of medicinal chemistry (19.12.2002)
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Glucagon antagonists/inverse agonists
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Year of Publication 02.09.2003
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Glucagon antagonists/inverse agonists
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Year of Publication 02.09.2003
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Glucagon antagonists/inverse agonists
ATSUO KUKI, ANTHONY LING, MIN TENG, MICHAEL BRUNO PLEWE, JESPER LAU, LOTTE BJERRE KNUDSEN, KIMBERLY ANN TESTON, PETER MADSEN, VLAD GREGOR, ULLA GROVE SIDELMANN, CHRISTIAN SAMS, MICHAEL DAVID JOHNSON, JUN FENG, JAVIER GONZALES, DAN KIEL, LARS NAERUM, YUFENG HONG, SHENGHUA SHI
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Year of Publication 20.06.2002
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GLUCAGON ANTAGONISTS/INVERSE AGONISTS
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Year of Publication 17.05.2001
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GLUCAGON ANTAGONISTS/INVERSE AGONISTS
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Year of Publication 28.10.2000
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ANTAGONISTS AND REVERSE ANTAGONISTS OF GLUCOGENE
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Year of Publication 11.09.2000
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GLUCAGON ANTAGONISTS/INVERSE AGONISTS
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Year of Publication 26.04.2000
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Year of Publication 26.04.2000
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Glucagon antagonists/inverse agonists
ATSUO KUKI, ANTHONY LING, MIN TENG, MICHAEL BRUNO PLEWE, JESPER LAU, LOTTE BJERRE KNUDSEN, KIMBERLY ANN TESTON, PETER MADSEN, VLAD GREGOR, ULLA GROVE SIDELMANN, CHRISTIAN SAMS, MICHAEL DAVID JOHNSON, JUN FENG, JAVIER GONZALES, DAN KIEL, LARS NAERUM, YUFENG HONG, SHENGHUA SHI
Year of Publication 25.01.1999
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Year of Publication 25.01.1999
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GLUCAGON ANTAGONISTS/INVERSE AGONISTS
SHI, SHENGHUA, GREGOR, VLAD, PLEWE, MICHAEL BRUNO, KNUDSEN, LOTTE BJERRE, SIDELMANN, ULLA GROVE, SAMS, CHRISTIAN, LAU, JESPER, FENG, JUN, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, NAERUM, LARS, LING, ANTHONY, GONZALES, JAVIER, MADSEN, PETER, TENG, MIN, JOHNSON, MICHAEL DAVID, TESTON, KIMBERLY ANN
Year of Publication 14.01.1999
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Year of Publication 14.01.1999
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GLUCAGON ANTAGONISTS/INVERSE AGONISTS
GREGOR, VLAD, SHI, SHENGHUA, PLEWE, MICHAEL, BRUNO, TESTON, KIMBERLY, ANN, JOHNSON, MICHAEL, DAVID, SAMS, CHRISTIAN, KNUDSEN, LOTTE, BJERRE, LAU, JESPER, FENG, JUN, KUKI, ATSUO, HONG, YUFENG, KIEL, DAN, NAERUM, LARS, SIDELMANN, ULLA, GROVE, GONZALES, JAVIER, LING, ANTHONY, MADSEN, PETER, TENG, MIN
Year of Publication 14.01.1999
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Year of Publication 14.01.1999
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Glucagon antagonists/inverse agonists
ATSUO KUKI, ANTHONY LAI LING, MIN TENG, MICHAEL BRUNO PLEWE, JESPER LAU, LOTTE BJERRE KNUDSEN, KIMBERLY ANN TESTON, PETER MADSEN, VLAD GREGOR, ULLA GROVE SIDELMANN, CHRISTIAN SAMS, MICHAEL DAVID JOHNSON, JUN FENG, JAVIER GONZALEZ, DAN KIEL, LARS NAERUM, YUFENG HONG, SHENGHUA SHI
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Year of Publication 25.01.1999
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Composto,uso do mesmo, composição farmacêutica, e, processos de tratar a diabete do tipo i ou do tipo ii, de tratar a hiperglicemia, e de diminuir a glicose do sangue em um mamìfero
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Year of Publication 29.08.2000
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Year of Publication 29.08.2000
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Glucagon antagonists/inversion agonists
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Year of Publication 12.07.2000
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Year of Publication 29.02.2000
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Year of Publication 29.02.2000
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