Search Results - "Terry A. Hauser" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Comparison of acetylcholine receptor interactions of the marine toxins, 13-desmethylspirolide C and gymnodimine

Comparison of acetylcholine receptor interactions of the marine toxins, 13-desmethylspirolide C and gymnodimine

by Hauser, Terry A., Hepler, Christopher D., Kombo, David C., Grinevich, Vladimir P., Kiser, Melanie N., Hooker, Dawn N., Zhang, Jiahui, Mountfort, Douglas, Selwood, Andrew, Akireddy, S. Rao, Letchworth, Sharon R., Yohannes, Daniel
Published in Neuropharmacology (01.06.2012)

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3D Molecular Descriptors Important for Clinical Success

3D Molecular Descriptors Important for Clinical Success

by Kombo, David C, Tallapragada, Kartik, Jain, Rachit, Chewning, Joseph, Mazurov, Anatoly A, Speake, Jason D, Hauser, Terry A, Toler, Steve
Published in Journal of chemical information and modeling (25.02.2013)

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An α7 Nicotinic Acetylcholine Receptor-Selective Agonist Reduces Weight Gain and Metabolic Changes in a Mouse Model of Diabetes

An α7 Nicotinic Acetylcholine Receptor-Selective Agonist Reduces Weight Gain and Metabolic Changes in a Mouse Model of Diabetes

by Marrero, Mario B., Lucas, Rudolf, Salet, Christina, Hauser, Terry A., Mazurov, Anatoly, Lippiello, Patrick M., Bencherif, Merouane
Published in The Journal of pharmacology and experimental therapeutics (01.01.2010)

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Discovery of (2S,3R)‑N‑[2-(Pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]oct-3-yl]benzo[b]furan-2-carboxamide (TC-5619), a Selective α7 Nicotinic Acetylcholine Receptor Agonist, for the Treatment of Cognitive Disorders

Discovery of (2S,3R)‑N‑[2-(Pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]oct-3-yl]benzo[b]furan-2-carboxamide (TC-5619), a Selective α7 Nicotinic Acetylcholine Receptor Agonist, for the Treatment of Cognitive Disorders

by Mazurov, Anatoly A, Kombo, David C, Hauser, Terry A, Miao, Lan, Dull, Gary, Genus, John F, Fedorov, Nikolai B, Benson, Lisa, Sidach, Serguei, Xiao, Yunde, Hammond, Philip S, James, John W, Miller, Craig H, Yohannes, Daniel
Published in Journal of medicinal chemistry (26.11.2012)

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The effect of food and liquid pH on the integrity of enteric-coated beads from cysteamine bitartrate delayed-release capsules

The effect of food and liquid pH on the integrity of enteric-coated beads from cysteamine bitartrate delayed-release capsules

by Pavloff, Nadine, Hauser, Terry A, Williams, Chris, Isbell, Sara Louis, Cadieux, Ben, Johnson, Mark
Published in Drug design, development and therapy (01.01.2018)

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QM-polarized ligand docking accurately predicts the trend in binding affinity of a series of arylmethylene quinuclidine-like derivatives at the α4β2 and α3β4 nicotinic acetylcholine receptors (nAChRs)

QM-polarized ligand docking accurately predicts the trend in binding affinity of a series of arylmethylene quinuclidine-like derivatives at the α4β2 and α3β4 nicotinic acetylcholine receptors (nAChRs)

by Kombo, David C., Grinevich, Vladimir P., Hauser, Terry A., Sidach, Serguei, Bencherif, Merouane
Published in Bioorganic & medicinal chemistry letters (01.09.2013)

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Discovery of 3‑(5-Chloro-2-furoyl)-3,7-diazabicyclo[3.3.0]octane (TC-6683, AZD1446), a Novel Highly Selective α4β2 Nicotinic Acetylcholine Receptor Agonist for the Treatment of Cognitive Disorders

Discovery of 3‑(5-Chloro-2-furoyl)-3,7-diazabicyclo[3.3.0]octane (TC-6683, AZD1446), a Novel Highly Selective α4β2 Nicotinic Acetylcholine Receptor Agonist for the Treatment of Cognitive Disorders

by Mazurov, Anatoly A, Miao, Lan, Bhatti, Balwinder S, Strachan, Jon-Paul, Akireddy, Srinivasa, Murthy, Srinivasa, Kombo, David, Xiao, Yun-de, Hammond, Philip, Zhang, Jenny, Hauser, Terry A, Jordan, Kristen G, Miller, Craig H, Speake, Jason D, Gatto, Gregory J, Yohannes, Daniel
Published in Journal of medicinal chemistry (08.11.2012)

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Novel nicotinic acetylcholine receptor agonists containing carbonyl moiety as a hydrogen bond acceptor

Novel nicotinic acetylcholine receptor agonists containing carbonyl moiety as a hydrogen bond acceptor

by Mazurov, Anatoly A., Kombo, David C., Akireddy, Srinivasa, Murthy, Srinivasa, Hauser, Terry A., Jordan, Kristen G., Gatto, Gregory J., Yohannes, Daniel
Published in Bioorganic & medicinal chemistry letters (01.07.2013)

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Discovery of novel alpha 7 nicotinic acetylcholine receptor ligands via pharmacophoric and docking studies of benzylidene anabaseine analogs

Discovery of novel alpha 7 nicotinic acetylcholine receptor ligands via pharmacophoric and docking studies of benzylidene anabaseine analogs

by Kombo, David C, Mazurov, Anatoly A, Chewning, Joseph, Hammond, Philip S, Tallapragada, Kartik, Hauser, Terry A, Speake, Jason, Yohannes, Daniel, Caldwell, William S
Published in Bioorganic & medicinal chemistry letters (15.01.2012)

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Discovery of novel α7 nicotinic acetylcholine receptor ligands via pharmacophoric and docking studies of benzylidene anabaseine analogs

Discovery of novel α7 nicotinic acetylcholine receptor ligands via pharmacophoric and docking studies of benzylidene anabaseine analogs

by Kombo, David C., Mazurov, Anatoly A., Chewning, Joseph, Hammond, Philip S., Tallapragada, Kartik, Hauser, Terry A., Speake, Jason, Yohannes, Daniel, Caldwell, William S.
Published in Bioorganic & medicinal chemistry letters (15.01.2012)

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Docking studies of benzylidene anabaseine interactions with α7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related α7 selective ligands

Docking studies of benzylidene anabaseine interactions with α7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related α7 selective ligands

by Kombo, David C., Mazurov, Anatoly, Tallapragada, Kartik, Hammond, Philip S., Chewning, Joseph, Hauser, Terry A., Vasquez-Valdivieso, Montserrat, Yohannes, Daniel, Talley, Todd T., Taylor, Palmer, Caldwell, William S.
Published in European journal of medicinal chemistry (01.11.2011)

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Analgesic effects mediated by neuronal nicotinic acetylcholine receptor agonists: Correlation with desensitization of α4β2 receptors

Analgesic effects mediated by neuronal nicotinic acetylcholine receptor agonists: Correlation with desensitization of α4β2 receptors

by Zhang, Jiahui, Xiao, Yun-De, Jordan, Kristen G., Hammond, Phil S., Van Dyke, Katherine M., Mazurov, Anatoly A., Speake, Jason D., Lippiello, Patrick M., James, John W., Letchworth, Sharon R., Bencherif, Merouane, Hauser, Terry A.
Published in European journal of pharmaceutical sciences (18.12.2012)

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Pharmacological properties and predicted binding mode of arylmethylene quinuclidine-like derivatives at the α3β4 nicotinic acetylcholine receptor (nAChR)

Pharmacological properties and predicted binding mode of arylmethylene quinuclidine-like derivatives at the α3β4 nicotinic acetylcholine receptor (nAChR)

by Kombo, David C., Hauser, Terry A., Grinevich, Vladimir P., Melvin, Matthew S., Strachan, Jon-Paul, Sidach, Serguei S., Chewning, Joseph, Fedorov, Nikolai, Tallapragada, Kartik, Breining, Scott R., Miller, Craig H.
Published in Bioorganic & medicinal chemistry letters (01.03.2013)

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2-(Arylmethyl)-3-substituted quinuclidines as selective α7 nicotinic receptor ligands

2-(Arylmethyl)-3-substituted quinuclidines as selective α7 nicotinic receptor ligands

by Mazurov, Anatoly, Klucik, Jozef, Miao, Lan, Phillips, Teresa Y., Seamans, Angela, Schmitt, Jeffrey D., Hauser, Terry A., Johnson, Raymond T., Miller, Craig
Published in Bioorganic & medicinal chemistry letters (15.04.2005)

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First Total Synthesis of (±)-3-Hydroxy-11-norcytisine: Structure Confirmation and Biological Characterization

First Total Synthesis of (±)-3-Hydroxy-11-norcytisine: Structure Confirmation and Biological Characterization

by Yohannes, Daniel, Hansen, Camilla P, Akireddy, Srinivasa Rao, Hauser, Terry A, Kiser, Melanie N, Gurnon, Nicholas J, Day, Cynthia S, Bhatti, Balwinder, Caldwell, William S
Published in Organic letters (04.12.2008)

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Therapeutic potential of novel selective drugs targeting nicotinic acetylcholine receptors

Therapeutic potential of novel selective drugs targeting nicotinic acetylcholine receptors

by Bencherif, Merouane, Hauser, Terry A, Jordan, Kristen G, Gatto, Gregory J
Published in Journal of molecular neuroscience (01.01.2006)

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Discovery of (2S,3R)-N-[2-(Pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]oct-3-yl]benzo[b]furan-2-carboxamide (TC-5619), a Selective alpha 7 Nicotinic Acetylcholine Receptor Agonist, for the Treatment of Cognitive Disorders

Discovery of (2S,3R)-N-[2-(Pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]oct-3-yl]benzo[b]furan-2-carboxamide (TC-5619), a Selective alpha 7 Nicotinic Acetylcholine Receptor Agonist, for the Treatment of Cognitive Disorders

by Mazurov, Anatoly A., Kombo, David C., Hauser, Terry A., Miao, Lan, Dull, Gary, Genus, John F., Fedorov, Nikolai B., Benson, Lisa, Sidach, Serguei, Xiao, Yunde, Hammond, Philip S., James, John W., Miller, Craig H., Yohannes, Daniel
Published in Journal of medicinal chemistry (22.11.2012)

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Discovery of 3-(5-Chloro-2-furoyl)-3,7-diazabicyclo[3.3.0]octane (TC-6683, AZD1446), a Novel Highly Selective alpha 4 beta 2 Nicotinic Acetylcholine Receptor Agonist for the Treatment of Cognitive Disorders

Discovery of 3-(5-Chloro-2-furoyl)-3,7-diazabicyclo[3.3.0]octane (TC-6683, AZD1446), a Novel Highly Selective alpha 4 beta 2 Nicotinic Acetylcholine Receptor Agonist for the Treatment of Cognitive Disorders

by Mazurov, Anatoly A., Miao, Lan, Bhatti, Balwinder S., Strachan, Jon-Paul, Akireddy, Srinivasa, Murthy, Srinivasa, Kombo, David, Xiao, Yun-de, Hammond, Philip, Zhang, Jenny, Hauser, Terry A., Jordan, Kristen G., Miller, Craig H., Speake, Jason D., Gatto, Gregory J., Yohannes, Daniel
Published in Journal of medicinal chemistry (08.11.2012)

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Docking studies of benzylidene anabaseine interactions with alpha 7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related alpha 7 selective ligands

Docking studies of benzylidene anabaseine interactions with alpha 7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related alpha 7 selective ligands

by Kombo, David C., Mazurov, Anatoly, Tallapragada, Kartik, Hammond, Philip S., Chewning, Joseph, Hauser, Terry A., Vasquez-Valdivieso, Montserrat, Yohannes, Daniel, Talley, Todd T., Taylor, Palmer, Caldwell, William S.
Published in European journal of medicinal chemistry (01.11.2011)

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Conformation Dependence of MHC Class I in the Modulation of Target Cell Sensitivity to Natural Killing

Conformation Dependence of MHC Class I in the Modulation of Target Cell Sensitivity to Natural Killing

by Hauser, Terry A, Malyguine, Anatoli M, Dawson, Jeffrey R
Published in Human immunology (01.02.1998)

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