Central Mechanisms Regulating Penile Erection in Conscious Rats: The Dopaminergic Systems Related to the Proerectile Effect of Apomorphine
Hsieh, Gin C, Hollingsworth, Peter R, Martino, Brenda, Chang, Renjie, Terranova, Marc A, O'Neill, Alyssa B, Lynch, James J, Moreland, Robert B, Donnelly-Roberts, Diana L, Kolasa, Teodozyi, Mikusa, Joseph P, McVey, Jill M, Marsh, Kennan C, Sullivan, James P, Brioni, Jorge D
Published in The Journal of pharmacology and experimental therapeutics (01.01.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2004)
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Journal Article
Synthesis and functional activity of (2-aryl-1-piperazinyl)-N-(3-methylphenyl)acetamides: selective dopamine D4 receptor agonists
Matulenko, Mark A, Hakeem, Ahmed A, Kolasa, Teodozyi, Nakane, Masaki, Terranova, Marc A, Uchic, Marie E, Miller, Loan N, Chang, Renjie, Donnelly-Roberts, Diana L, Namovic, Marian T, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Bioorganic & medicinal chemistry (01.07.2004)
Published in Bioorganic & medicinal chemistry (01.07.2004)
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Journal Article
Discovery of 3-Methyl-N-(1-oxy-3‘,4‘,5‘,6‘-tetrahydro-2‘H-[2,4‘-bipyridine]-1‘-ylmethyl)benzamide (ABT-670), an Orally Bioavailable Dopamine D4 Agonist for the Treatment of Erectile Dysfunction
Patel, Meena V, Kolasa, Teodozyj, Mortell, Kathleen, Matulenko, Mark A, Hakeem, Ahmed A, Rohde, Jeffrey J, Nelson, Sherry L, Cowart, Marlon D, Nakane, Masaki, Miller, Loan N, Uchic, Marie E, Terranova, Marc A, El-Kouhen, Odile F, Donnelly-Roberts, Diana L, Namovic, Marian T, Hollingsworth, Peter R, Chang, Renjie, Martino, Brenda R, Wetter, Jill M, Marsh, Kennan C, Martin, Ruth, Darbyshire, John F, Gintant, Gary, Hsieh, Gin C, Moreland, Robert B, Sullivan, James P, Brioni, Jorge D, Stewart, Andrew O
Published in Journal of medicinal chemistry (14.12.2006)
Published in Journal of medicinal chemistry (14.12.2006)
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Journal Article
Discovery of 2-(4-Pyridin-2-ylpiperazin-1-ylmethyl)-1H-benzimidazole (ABT-724), a Dopaminergic Agent with a Novel Mode of Action for the Potential Treatment of Erectile Dysfunction
Cowart, Marlon, Latshaw, Steven P, Bhatia, Pramila, Daanen, Jerome F, Rohde, Jeffrey, Nelson, Sherry L, Patel, Meena, Kolasa, Teodozyi, Nakane, Masaki, Uchic, Marie E, Miller, Loan N, Terranova, Marc A, Chang, Renjie, Donnelly-Roberts, Diana L, Namovic, Marian T, Hollingsworth, Peter R, Martino, Brenda R, Lynch, James J, Sullivan, James P, Hsieh, Gin C, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Journal of medicinal chemistry (15.07.2004)
Published in Journal of medicinal chemistry (15.07.2004)
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Journal Article
Comparative pharmacology of human dopamine D2-like receptor stable cell lines coupled to calcium flux through Gαqo5
MORELAND, Robert B, NAKANE, Masaki, EL-KOUHEN, Odile F, MASTERS, Jeffrey N, BRIONI, Jorge D, DONNELLY-ROBERTS, Diana L, MILLER, Loan N, CHANG, Renjie, UCHIC, Marie E, TERRANOVA, Marc A, GUBBINS, Earl J, HELFRICH, Rosalind J, NAMOVIC, Marian T
Published in Biochemical pharmacology (15.08.2004)
Published in Biochemical pharmacology (15.08.2004)
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Journal Article
1-Aryl-3-(4-pyridine-2-ylpiperazin-1-yl)propan-1-one Oximes as Potent Dopamine D4 Receptor Agonists for the Treatment of Erectile Dysfunction
Kolasa, Teodozyj, Matulenko, Mark A, Hakeem, Ahmed A, Patel, Meena V, Mortell, Kathleen, Bhatia, Pramila, Henry, Rodger, Nakane, Masaki, Hsieh, Gin C, Terranova, Marc A, Uchic, Marie E, Miller, Loan N, Chang, Renje, Donnelly-Roberts, Diana L, Namovic, Marian T, Hollingsworth, Peter R, Martino, Brenda, El Kouhen, Odile, Marsh, Kennan C, Wetter, Jill M, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Journal of medicinal chemistry (24.08.2006)
Published in Journal of medicinal chemistry (24.08.2006)
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Journal Article
Dopamine D4 Ligands and Models of Receptor Activation: 2-(4-Pyridin-2-ylpiperazin-1-ylmethyl)-1H-benzimidazole and Related Heteroarylmethylarylpiperazines Exhibit a Substituent Effect Responsible for Additional Efficacy Tuning
Stewart, Andrew O, Cowart, Marlon D, Moreland, Robert B, Latshaw, Steve P, Matulenko, Mark A, Bhatia, Pramila A, Wang, Xueqing, Daanen, Jerome F, Nelson, Sherry L, Terranova, Marc A, Namovic, Marian T, Donnelly-Roberts, Diana L, Miller, Loan N, Nakane, Masaki, Sullivan, James P, Brioni, Jorge D
Published in Journal of medicinal chemistry (22.04.2004)
Published in Journal of medicinal chemistry (22.04.2004)
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Journal Article
2-[4-(3,4-Dimethylphenyl)piperazin-1-ylmethyl]-1H benzoimidazole (A-381393), a selective dopamine D4 receptor antagonist
Nakane, Masaki, Cowart, Marlon D, Hsieh, Gin C, Miller, Loan, Uchic, Marie E, Chang, Renjie, Terranova, Marc A, Donnelly-Roberts, Diana L, Namovic, Marian T, Miller, Thomas R, Wetter, Jill M, Marsh, Kennan, Stewart, Andrew O, Brioni, Jorge D, Moreland, Robert B
Published in Neuropharmacology (01.07.2005)
Published in Neuropharmacology (01.07.2005)
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Journal Article
3H] A-369508 ([2-[4-(2-cyanophenyl)-1-piperazinyl]-N-(3-methylphenyl) acetamide): an agonist radioligand selective for the dopamine D4 receptor
MORELAND, Robert B, TERRANOVA, Marc A, CHANG, Renjie, UCHIC, Marie E, MATULENKO, Mark A, SURBER, Bruce W, STEWART, Andrew O, BRIONI, Jorge D
Published in European journal of pharmacology (23.08.2004)
Published in European journal of pharmacology (23.08.2004)
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Journal Article
Synthesis and activity of 2-[4-(4-[3H]-2-cyanophenyl)piperazinyl]-N-(2,4,6-[3H]3-3-methylphenyl)acetamide: a selective dopamine D4 receptor agonist and radioligand
Matulenko, Mark A., Surber, Bruce, Fan, Leimin, Kolasa, Teodozyi, Nakane, Masaki, Terranova, Marc A., Uchic, Marie E., Miller, Loan N., Chang, Renjie, Donnelly-Roberts, Diana L., Namovic, Marian T., Moreland, Robert B., Brioni, Jorge D., Stewart, Andrew O.
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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Journal Article
Discovery of 3-methyl-N-(1-oxy-3 ',4 ',5 ',6 '-tetrahydro-2 ' H-[2,4 '-bipyridine]-1 '-ylmethyl)benzamide (ABT-670), an orally bioavailable dopamine D-4 agonist for the treatment of erectile dysfunction
Patel, Meena V., Kolasa, Teodozyj, Mortell, Kathleen, Matulenko, Mark A., Hakeem, Ahmed A., Rohde, Jeffrey J., Nelson, Sherry L., Cowart, Marlon D., Nakane, Masaki, Miller, Loan N., Uchic, Marie E., Terranova, Marc A., El-Kouhen, Odile F., Donnelly-Roberts, Diana L., Namovic, Marian T., Hollingsworth, Peter R., Chang, Renjie, Martino, Brenda R., Wetter, Jill M., Marsh, Kennan C., Martin, Ruth, Darbyshire, John F., Gintant, Gary, Hsieh, Gin C., Moreland, Robert B., Sullivan, James P., Brioni, Jorge D., Stewart, Andrew O.
Published in Journal of medicinal chemistry (14.12.2006)
Published in Journal of medicinal chemistry (14.12.2006)
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Journal Article
1-Aryl-3-(4-pyridine-2-ylpiperazin-1-yl)propan-1-one oximes as potent dopamine D-4 receptor agonists for the treatment of erectile dysfunction
Kolasa, Teodozyj, Matulenko, Mark A., Hakeem, Ahmed A., Patel, Meena V., Mortell, Kathleen, Bhatia, Pramila, Henry, Rodger, Nakane, Masaki, Hsieh, Gin C., Terranova, Marc A., Uchic, Marie E., Miller, Loan N., Chang, Renje, Donnelly-Roberts, Diana L., Namovic, Marian T., Hollingsworth, Peter R., Martino, Brenda, El Kouhen, Odile, Marsh, Kennan C., Wetter, Jill M., Moreland, Robert B., Brioni, Jorge D., Stewart, Andrew O.
Published in Journal of medicinal chemistry (24.08.2006)
Published in Journal of medicinal chemistry (24.08.2006)
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Journal Article
Synthesis and functional activity of (2-aryl-1-piperazinyl)- N-(3-methylphenyl)acetamides: selective dopamine D 4 receptor agonists
Matulenko, Mark A, Hakeem, Ahmed A, Kolasa, Teodozyi, Nakane, Masaki, Terranova, Marc A, Uchic, Marie E, Miller, Loan N, Chang, Renjie, Donnelly-Roberts, Diana L, Namovic, Marian T, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Bioorganic & medicinal chemistry (01.07.2004)
Published in Bioorganic & medicinal chemistry (01.07.2004)
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Journal Article
2-[4-(3,4-Dimethylphenyl)piperazin-1-ylmethyl]-1H benzoimidazole (A-381393), a selective dopamine D 4 receptor antagonist
Nakane, Masaki, Cowart, Marlon D., Hsieh, Gin C., Miller, Loan, Uchic, Marie E., Chang, Renjie, Terranova, Marc A., Donnelly-Roberts, Diana L., Namovic, Marian T., Miller, Thomas R., Wetter, Jill M., Marsh, Kennan, Stewart, Andrew O., Brioni, Jorge D., Moreland, Robert B.
Published in Neuropharmacology (01.07.2005)
Published in Neuropharmacology (01.07.2005)
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Journal Article
3 H] A-369508 ([2-[4-(2-cyanophenyl)-1-piperazinyl]- N-(3-methylphenyl) acetamide): an agonist radioligand selective for the dopamine D 4 receptor
Moreland, Robert B., Terranova, Marc A., Chang, Renjie, Uchic, Marie E., Matulenko, Mark A., Surber, Bruce W., Stewart, Andrew O., Brioni, Jorge D.
Published in European journal of pharmacology (2004)
Published in European journal of pharmacology (2004)
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Journal Article
Comparative pharmacology of human dopamine D(2)-like receptor stable cell lines coupled to calcium flux through Galpha(qo5)
Moreland, Robert B, Nakane, Masaki, Donnelly-Roberts, Diana L, Miller, Loan N, Chang, Renjie, Uchic, Marie E, Terranova, Marc A, Gubbins, Earl J, Helfrich, Rosalind J, Namovic, Marian T, El-Kouhen, Odile F, Masters, Jeffrey N, Brioni, Jorge D
Published in Biochemical pharmacology (15.08.2004)
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Published in Biochemical pharmacology (15.08.2004)
Journal Article
Synthesis and functional activity of (2-aryl-1-piperazinyl)-N-(3-methylphenyl)acetamides: selective dopamine D4 receptor agonists
MATULENKO, Mark A, HAKEEM, Ahmed A, MORELAND, Robert B, BRIONI, Jorge D, STEWART, Andrew O, KOLASA, Teodozyi, NAKANE, Masaki, TERRANOVA, Marc A, UCHIC, Marie E, MILLER, Loan N, CHANG, Renjie, DONNELLY-ROBERTS, Diana L, NAMOVIC, Marian T
Published in Bioorganic & medicinal chemistry (01.07.2004)
Published in Bioorganic & medicinal chemistry (01.07.2004)
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Journal Article
Comparative pharmacology of human dopamine D 2-like receptor stable cell lines coupled to calcium flux through Gα qo5
Moreland, Robert B, Nakane, Masaki, Donnelly-Roberts, Diana L, Miller, Loan N, Chang, Renjie, Uchic, Marie E, Terranova, Marc A, Gubbins, Earl J, Helfrich, Rosalind J, Namovic, Marian T, El-Kouhen, Odile F, Masters, Jeffrey N, Brioni, Jorge D
Published in Biochemical pharmacology (2004)
Published in Biochemical pharmacology (2004)
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Journal Article
Discovery of 2-(4-Pyridin-2-ylpiperazin-1-ylmethyl)-1 H -benzimidazole (ABT-724), a Dopaminergic Agent with a Novel Mode of Action for the Potential Treatment of Erectile Dysfunction
Cowart, Marlon, Latshaw, Steven P., Bhatia, Pramila, Daanen, Jerome F., Rohde, Jeffrey, Nelson, Sherry L., Patel, Meena, Kolasa, Teodozyi, Nakane, Masaki, Uchic, Marie E., Miller, Loan N., Terranova, Marc A., Chang, Renjie, Donnelly-Roberts, Diana L., Namovic, Marian T., Hollingsworth, Peter R., Martino, Brenda R., Lynch, James J., Sullivan, James P., Hsieh, Gin C., Moreland, Robert B., Brioni, Jorge D., Stewart, Andrew O.
Published in Journal of medicinal chemistry (01.07.2004)
Published in Journal of medicinal chemistry (01.07.2004)
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Journal Article
Dopamine D 4 Ligands and Models of Receptor Activation: 2-(4-Pyridin-2-ylpiperazin-1-ylmethyl)-1 H -benzimidazole and Related Heteroarylmethylarylpiperazines Exhibit a Substituent Effect Responsible for Additional Efficacy Tuning
Stewart, Andrew O., Cowart, Marlon D., Moreland, Robert B., Latshaw, Steve P., Matulenko, Mark A., Bhatia, Pramila A., Wang, Xueqing, Daanen, Jerome F., Nelson, Sherry L., Terranova, Marc A., Namovic, Marian T., Donnelly-Roberts, Diana L., Miller, Loan N., Nakane, Masaki, Sullivan, James P., Brioni, Jorge D.
Published in Journal of medicinal chemistry (01.04.2004)
Published in Journal of medicinal chemistry (01.04.2004)
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Journal Article