Central Mechanisms Regulating Penile Erection in Conscious Rats: The Dopaminergic Systems Related to the Proerectile Effect of Apomorphine
Hsieh, Gin C, Hollingsworth, Peter R, Martino, Brenda, Chang, Renjie, Terranova, Marc A, O'Neill, Alyssa B, Lynch, James J, Moreland, Robert B, Donnelly-Roberts, Diana L, Kolasa, Teodozyi, Mikusa, Joseph P, McVey, Jill M, Marsh, Kennan C, Sullivan, James P, Brioni, Jorge D
Published in The Journal of pharmacology and experimental therapeutics (01.01.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2004)
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Discovery of 2-(4-Pyridin-2-ylpiperazin-1-ylmethyl)-1H-benzimidazole (ABT-724), a Dopaminergic Agent with a Novel Mode of Action for the Potential Treatment of Erectile Dysfunction
Cowart, Marlon, Latshaw, Steven P, Bhatia, Pramila, Daanen, Jerome F, Rohde, Jeffrey, Nelson, Sherry L, Patel, Meena, Kolasa, Teodozyi, Nakane, Masaki, Uchic, Marie E, Miller, Loan N, Terranova, Marc A, Chang, Renjie, Donnelly-Roberts, Diana L, Namovic, Marian T, Hollingsworth, Peter R, Martino, Brenda R, Lynch, James J, Sullivan, James P, Hsieh, Gin C, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Journal of medicinal chemistry (15.07.2004)
Published in Journal of medicinal chemistry (15.07.2004)
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Dopamine D-4 ligands and models of receptor activation: 2-(4-pyridin-2-ylpiperazin-1-ylmethyl)-1H-benzimidazole and related heteroarylmethylarylpiperazines exhibit a substituent effect responsible for additional efficacy tuning
Stewart, AO, Cowart, MD, Moreland, RB, Latshaw, SP, Matulenko, MA, Bhatia, PA, Wang, XQ, Daanen, JF, Nelson, SL, Terranova, MA, Namovic, MT, Donnelly-Roberts, DL, Miller, LN, Nakane, M, Sullivan, JP, Brioni, JD
Published in Journal of medicinal chemistry (22.04.2004)
Published in Journal of medicinal chemistry (22.04.2004)
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Synthesis and functional activity of (2-aryl-1-piperazinyl)- N-(3-methylphenyl)acetamides: selective dopamine D 4 receptor agonists
Matulenko, Mark A, Hakeem, Ahmed A, Kolasa, Teodozyi, Nakane, Masaki, Terranova, Marc A, Uchic, Marie E, Miller, Loan N, Chang, Renjie, Donnelly-Roberts, Diana L, Namovic, Marian T, Moreland, Robert B, Brioni, Jorge D, Stewart, Andrew O
Published in Bioorganic & medicinal chemistry (01.07.2004)
Published in Bioorganic & medicinal chemistry (01.07.2004)
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2-[4-(3,4-Dimethylphenyl)piperazin-1-ylmethyl]-1H benzoimidazole (A-381393), a selective dopamine D 4 receptor antagonist
Nakane, Masaki, Cowart, Marlon D., Hsieh, Gin C., Miller, Loan, Uchic, Marie E., Chang, Renjie, Terranova, Marc A., Donnelly-Roberts, Diana L., Namovic, Marian T., Miller, Thomas R., Wetter, Jill M., Marsh, Kennan, Stewart, Andrew O., Brioni, Jorge D., Moreland, Robert B.
Published in Neuropharmacology (01.07.2005)
Published in Neuropharmacology (01.07.2005)
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Discovery of 3-Methyl-N-(1-oxy-3',4',5',6'-tetrahydro-2' H-[2,4'-bipyridine]-1'-ylmethyl)benzamide (ABT-670), an Orally Bioavailable Dopamine D sub(4) Agonist for the Treatment of Erectile Dysfunction
Patel, M V, Kolasa, T, Mortell, K, Matulenko, MA, Hakeem, A A, Rohde, J J, Nelson, S L, Cowart, MD, Nakane, M, Miller, L N, Uchic, ME, Terranova, MA, El-Kouhen, O F, Donnelly-Roberts, D L
Published in Journal of medicinal chemistry (14.12.2006)
Published in Journal of medicinal chemistry (14.12.2006)
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Activation of soluble guanylate cyclase causes relaxation of corpus cavernosum tissue: Synergism of nitric oxide and YC-1
NAKANE, M, HSIEH, G, MILLER, L. N, CHANG, R, TERRANOVA, M. A, MORELAND, R. B, KOLASA, T, BRIONI, J. D
Published in International journal of impotence research (01.04.2002)
Published in International journal of impotence research (01.04.2002)
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Journal Article
2-[4-(3, 4-Dimethylphenyl)piperazin-1-ylmethyl]-1H benzoimidazole (A-381393), a selective dopamine D sub(4) receptor antagonist
Nakane, M, Cowart, MD, Hsieh, G C, Miller, L, Uchic, ME, Chang, R, Terranova, MA, Donnelly-Roberts, D L, Namovic, M T, Miller, T R, Wetter, J M, Marsh, K, Stewart, A O, Brioni, J D, Moreland, R B
Published in Neuropharmacology (01.07.2005)
Published in Neuropharmacology (01.07.2005)
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